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Titolo Data di pubblicazione Autore(i) Rivista Editore
Off‑target activity of NBOMes and NBOMe analogs at the µ opioid receptor 1-gen-2023 Deventer, Marie H.; Persson, Mattias; Laus, Antonio; Pottie, Eline; Cannaert, Annelies; Tocco, Graziella; Gréen, Henrik; Stove, Christophe P. ARCHIVES OF TOXICOLOGY -
In silico characterization of ligand–receptor interactions for U-47700, N,N-didesmethyl-U-47700, U-50488 at mu- and kappa-opioid receptors 1-gen-2023 Laus, A; Kumar, A; Caboni, P; DE LUCA, MARIA ANTONIETTA; Baumann, Mh; Pieroni, E; Tocco, G. ARCHIV DER PHARMAZIE -
Structural Elucidation of Relevant Gibberellic Acid Impurities and In Silico Investigation of Their Interaction with Soluble Gibberellin Receptor GID1 1-gen-2023 Caboni, Pierluigi; Laus, Antonio; Eloh, Kodjo; Ntalli, Nikoletta G.; Casula, Mattia; Di Giorgi, Sabrina; Tocco, Graziella ACS OMEGA -
Dihydroxyphenyl- and Heteroaromatic-Based Thienopyrimidinones to Tackle HIV-1 LEDGF/p75-Dependent IN Activity 1-gen-2023 Tocco, G.; Canton, S.; Laus, A.; Caboni, P.; Le Grice, S. F. J.; Tramontano, E.; Esposito, F. MOLECULES -
Mukaiyama reagent: An efficient reaction mediator for rapid synthesis of 1,2-disubstituted-1H-benzo[d]imidazoles 1-gen-2022 Tocco, G.; Laus, A.; Caboni, P. TETRAHEDRON LETTERS -
Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists 1-gen-2022 De Luca, Maria Antonietta; Tocco, Graziella; Mostallino, Rafaela; Laus, Antonio; Caria, Francesca; Musa, Aurora; Pintori, Nicholas; Ucha, Marcos; Poza, Celia; Ambrosio, Emilio; Di Chiara, Gaetano; Castelli, M Paola NEUROPHARMACOLOGY -
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists 1-gen-2022 Tocco, Graziella; Laus, Antonio; Vanejevs, Maksims; Ture, Anastasija; Mostallino, Rafaela; Pintori, Nicholas; De Luca, Maria Antonietta; Castelli, M. Paola; Di Chiara, Gaetano ARCHIV DER PHARMAZIE -
U-47700 and its analogs: non-fentanyl synthetic opioids impacting the recreational drug market 1-gen-2020 Baumann, Michael H.; Tocco, Graziella; Papsun, Donna M.; Mohr, Amanda L.; Fogarty, Melissa F.; Krotulski, Alex J. BRAIN SCIENCES -
Electron-Deficient Alkynes as Powerful Tools against Root-Knot Nematode Melodogyne incognita: Nematicidal Activity and Investigation on the Mode of Action 1-gen-2020 Tocco, Graziella; Eloh, Kodjo; Laus, Antonio; Sasanelli, Nicola; Caboni, Pierluigi JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Scaffold hopping and optimisation of 3’,4’-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H 1-gen-2020 Tocco, Graziella; Esposito, Francesca; Caboni, Pierluigi; Laus, Antonio; Beutler, John A.; Wilson, Jennifer A.; Corona, Angela; Le Grice, Stuart F. J.; Tramontano, Enzo JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Uvaria angolensis as a promising source of inhibitors of HIV-1 RT-associated RNA-dependent DNA polymerase and RNase H functions 1-gen-2018 NGOUTANE MFOPA, Alvine; Corona, Angela; Eloh, Kodjo; Tramontano, Enzo; Frau, Aldo; Boyom, Fabrice Fekam; Caboni, Pierluigi; Tocco, Graziella NATURAL PRODUCT RESEARCH -
Haloacetophenones as newly potent nematicides against Meloidogyne incognita 1-gen-2017 Tocco, Graziella; Eloh, Kodjo; Onnis, Valentina; Sasanelli, Nicola; Caboni, Pierluigi INDUSTRIAL CROPS AND PRODUCTS -
Solvent-Free addition of indole to aldehydes: Unexpected synthesis of novel 1-[1-(1h-indol-3-yl) alkyl]-1h-indoles and preliminary evaluation of their cytotoxicity in hepatocarcinoma cells 1-gen-2017 Tocco, Graziella; Zedda, Gloria; Casu, Mariano; Simbula, Gabriella; Begala, Michela MOLECULES -
Nematicidal activity of the volatilome of Eruca sativa on Meloidogyne incognita 1-gen-2015 Aissani, Nadhem; Urgeghe, Pp; Oplos, C; Saba, M; Tocco, Graziella; Petretto, Gl; Eloh, Kodjo; Menkissoglu Spiroudi, U; Ntalli, Nikoletta; Caboni, Pierluigi JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Tulipaline A: Structure–activity aspects as a nematicide and V-ATPase inhibitor 1-gen-2014 Caboni, Pierluigi; Tronci, L; Liori, B; Tocco, Graziella; Sasanelli, N; Diana, Andrea PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY -
ZnO-mediated regioselective C-arylsulfonylation of indoles: A facile solvent-free synthesis of 2- and 3-sulfonylindoles and preliminary evaluation of their activity against drug-resistant mutant HIV-1 reverse transcriptases (RTs) 1-gen-2013 Tocco, Graziella; Begala, Michela; Esposito, Francesca; Caboni, Pierluigi; Cannas, Valeria; Tramontano, Enzo TETRAHEDRON LETTERS -
Potent nematicidal activity of phthalaldehyde, salicylaldehyde, and cinnamic aldehyde against Meloidogyne incognita 1-gen-2013 Caboni, Pierluigi; Aissani, Nadhem; Cabras, Tiziana; Falqui, Andrea; Marotta, R; Liori, B; Ntalli, Nikoletta; Sarais, Giorgia; Sasanelli, N; Tocco, Graziella JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Nematicidal activity of mint aqueous extracts against the root-knot nematode Meloidogyne incognita 1-gen-2013 Caboni, Pierluigi; Saba, M; Tocco, Graziella; Casu, Laura; Murgia, A; Maxia, Andrea; Menkissoglu Spiroudi, U; Ntalli, Nikoletta JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Active site and allosteric inhibitors of the ribonuclease H activity of HIV reverse transcriptase 1-gen-2013 Corona, Angela; Masaoka, T; Tocco, Graziella; Tramontano, Enzo; Le Grice, Sfj FUTURE MEDICINAL CHEMISTRY -
Exploiting drug-resistant enzymes as tools to identify thienopyrimidinone inhibitors of human immunodeficiency virus reverse transcriptase-associated ribonuclease H 1-gen-2013 Masaoka, T; Chung, S; Caboni, Pierluigi; Rausch, Jw; Wilson, Ja; Taskent Sezgin, H; Beutler, Ja; Tocco, Graziella; Le Grice, Sfj JOURNAL OF MEDICINAL CHEMISTRY -
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