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Titolo Data di pubblicazione Autore(i) Rivista Editore
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2015 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies 1-gen-2015 Ruiu, S; Anzani, N; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Alcaro, S; Maccioni, Elias; Distinto, Simona; Cottiglia, Filippo JOURNAL OF NATURAL PRODUCTS -
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) enlighten the mechanism of action of a new Ribonuclease H/DNA polymerase RT dual inhibitor 1-gen-2014 Esposito, Francesca; Corona, Angela; Meleddu, Rita; Distinto, Simona; Giulia, Bianco; Maccioni, Elias; Stuart JF Le Grice, ; Enzo, Tramontano - -
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2014 Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, C; Esposito, Francesca; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Artese, A; Scalise, D; Fresta, M; Arridu, A; Ortuso, F; Maccioni, Elias; Tramontano, Enzo CHEMMEDCHEM -
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 RT. 1-gen-2013 Esposito, Francesca; Meleddu, R; Cannas, V; Distinto, Simona; Del Vecchio, C; Biano, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo - -
Synthesis and biological activity evaluation of new dual-inhibitors of both associated functions of HIV-1 RT 1-gen-2013 Meleddu, R.; Distinto, Simona; Corona, Angela; Bianco, Giulia; Arridu, A.; Cannas, V.; Tramontano, Enzo; Alcaro, S.; Matyus, P.; Maccioni, Elias - -
MD protocol validation for the study of MAOB-inhibitor complexes 1-gen-2013 Bianco, Giulia; Cossu, P.; Distinto, Simona; Meleddu, R.; Arridu, A.; Ortuso, F.; Alcaro, S.; Maccioni, Elias - -
In search of new antitumor agents through the combination of individually active moieties: construction of a [3,5-diaryl-(4,5- dihydropyrazol-1-yl)-4-oxo-1,3-thiazol-5-ylidene]- 1H-indol-2-ones library 1-gen-2013 Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; Bogdan, D.; Matyus, P.; Maccioni, Elias - -
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents 1-gen-2013 Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias - -
Towards the total block of HIV-1 Reverse Transcriptase: the dual-inhibitors approach 1-gen-2013 Meleddu, R.; Arridu, A.; Bianco, Giulia; Tramontano, Enzo; Distinto, Simona; Matyus, P.; Maccioni, Elias - -
N-alkylamides from Otanthus maritimus: structure elucidation, binding affinity for cannabinoid receptors and computational study 1-gen-2013 Anzani, N.; Ruiu, S.; Orrù, A.; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S.; Cottiglia, Filippo - -
Molecular Aspects of the RT/drug Interactions. Perspective of Dual Inhibitors 1-gen-2013 Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Corona, Angela; Alcaro, S; Tramontano, Enzo CURRENT PHARMACEUTICAL DESIGN -
Identification and characterization of new DNA G-quadruplex binders selected by a combination of ligand and structure based virtual screening approaches 1-gen-2013 Alcaro, S.; Musetti, C.; Distinto, Simona; Casatti, M.; Zagotto, G.; Artese, A.; Parrotta, L.; Moraca, F.; Costa, G.; Ortuso, F.; Maccioni, Elias; Sissi, C. JOURNAL OF MEDICINAL CHEMISTRY -
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Single Site Dual Inhibitors of HIV-1 RT 1-gen-2013 Esposito, Francesca; Meleddu, R; Cannas, Valeria; Distinto, Simona; Del Vecchio, C; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo VIROLOGIE -
Design, synthesis and biological activity evaluation of c-myc proto-oncogene binders as potential antitumor agents 1-gen-2013 Meleddu, R.; Distinto, S; Sissi, C.; Musetti, C.; Arridu, A.; Bianco, Giulia; Parrotta, L.; Ortuso, F.; Alcaro, S.; Maccioni, Elias - -
New dual inhibitors of RT associated functions: investigation on their mechanism and mode of action 1-gen-2013 Distinto, Simona; Bianco, Giulia; Meleddu, R.; Cannas, C.; Del Vecchio, C.; Cottiglia, Filippo; Alcaro, S.; Parolin, C.; Tramontano, Enzo; Maccioni, Elias - -
Investigation on the mechanism of action of new dual inhibitors of HIV-1 RT 1-gen-2013 Bianco, Giulia; Distinto, Simona; Meleddu, R.; Cannas, C.; Del Vecchio, C.; Cottiglia, Filippo; Alcaro, S.; Parolin, C.; Tramontano, Enzo; Maccioni, Elias - -
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors 1-gen-2013 Ruiu, S; Anzani, Nicola; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S; Cottiglia, Filippo BIOORGANIC & MEDICINAL CHEMISTRY -
A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition 1-gen-2013 Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Distinto, Simona; Yañez, M.; Viña, D.; Lamela, M.; Maccioni, Elias JOURNAL OF HETEROCYCLIC CHEMISTRY -
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) shed light on the mechanism of action of a new Ribonuclease H/ DNA polymerase RT dual inhibitor 1-gen-2013 Corona, Angela; Meleddu, Rita; Esposito, Francesca; Distinto, Simona; Bianco, Giulia; Maccioni, Elias; Le Grice, S.; Tramontano, Enzo RETROVIROLOGY BioMed Central Ltd
Mostrati risultati da 41 a 60 di 163
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