Sfoglia per Autore
Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors
2011-01-01 Meleddu, Rita; Corona, Angela; Sanna M., L; Esposito, Francesca; Cardia M., C; Tramontano, Enzo; Maccioni, Elias
Isatin derivatives as new scaffolds for HIV-1 reverse transcriptase associated RNase H and RDDP dual inhibitors
2011-01-01 Corona, Angela; Meleddu, Rita; Esposito, Francesca; Sanna, M. L.; Distinto, Simona; Maccioni, Elias; Tramontano, Enzo
Exploring new scaffolds for the inibition of the Ribonuclease H function of RT HIV-1
2011-01-01 Meleddu, Rita; Corona, Angela; Distinto, S; Esposito, Francesca; Sanna M., L; Cardia M., C; Tramontano, Enzo; Maccioni, Elias
A combined shape-, 2D-fingerprint-and pharmacophore-based virtual screening for the identification of dual inhibitors targeting HIV-1 reverse transcriptase.
2011-01-01 Esposito, Francesca; Distinto, Simona; J., Kirchmair; C. M., Cardia; Maccioni, Elias; S., Alcaro; L., Zinzula; E., Tramontano
Identification of HIV-1 reverse transcriptase dual inhibitors by a combined shape-, 2D-fingerprint- and pharmacophore-based virtual screening approach
2011-01-01 Distinto, S; Esposito, Francesca; Kirchmair, J; Cardia, Cm; Maccioni, Elias; Alcaro, S; Zinzula, Luca; Tramontano, Enzo
Semicarbazide-sensitive amine oxidase/vascular adhesion protein-1: a patent survey
2011-01-01 Dunkel, P; Balogh, B; Meleddu, Rita; Maccioni, Elias; Gyires, K; Mátyus, P.
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona
SYNTHESIS, MOLECULAR MODELLING, INHIBITORY ACTIVITY, AND SELECTIVITY TOWARDS MONOAMINE OXIDASE OF NEW HETEROCYCLIC SCAFFOLDS
2010-01-01 Sanna M., L; Maccioni, Elias; Alcaro, S; Cirilli, R; Ferretti, R; Yanez, M; Cardia M., C; Distinto, S; Meleddu, Rita; Vigo, S; Ortuso, F.
Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach
2010-01-01 Meleddu, Rita; Sanna, M. L.; Distinto, Simona; Esposito, Francesca; Corona, Angela; Ortuso, F.; Alcaro, S.; Maccioni, Elias; Cardia, M. C.; Tramontano, Enzo
Shape based computer aided similarity screening: a valid tool in the discovery of new scaffolds for the inhibition of HIV-1 reverse transcriptase associated ribonuclease H function
2010-01-01 Distinto, Simona; Esposito, Francesca; Maccioni, Elias; Cardia, M. C.; Markt, P.; Tramontano, Enzo
Brain delivery of the NK3 receptor agonist senktide by immunoliposome: an in vivo microdialysis study
2010-01-01 DE LUCA, MARIA ANTONIETTA; Lai, Francesco; Bimpisidis, Zisis; Manca, MARIA LETIZIA; Maccioni, Elias; Caboni, Pierluigi; Fadda, ANNA MARIA; DI CHIARA, Gaetano
Synthesis, molecular modelling, inhibitory acivity, and selectivity towards monoamine oxidase of new heterocyclic scaffold
2010-01-01 Sanna, M. L.; Maccioni, Elias; Alcaro, S.; Cirilli, R.; Ferretti, R.; Yañez, M.; Cardia, M. C.; Distinto, Simona; Meleddu, R.; Vigo, S.; Ortuso, F.
Identification of new scaffolds for the inhibition of HIV-1 Reverse Transcriptase associated Ribonuclease H function by means of shape based similarity screening
2010-01-01 Distinto, Simona; Esposito, Francesca; Maccioni, Elias; Cardia, M. C.; Markt, P.; Tramontano, Enzo; Sanna, M. L.; Meleddu, Rita
Semipreparative HPLC enantioseparation, chiroptical properties, and absolute configuration of two novel cyclooxygenase-2 inhibitors
2010-01-01 Cirilli, R; Fiore, S; LA TORRE, F; Maccioni, Elias; Secci, D; Sanna, MARIA LUISA; Faggi, C.
Application of an immobilised amylose-based chiral stationary phase to the development of new monoamine oxidase B inhibitors
2010-01-01 Sanna, MARIA LUISA; Maccioni, Elias; Sara, Vigo; Cristina, Faggi; Roberto, Cirilli
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase
2010-01-01 Maccioni, Elias; S., Alcaro; F., Orallo; Cardia, MARIA CRISTINA; Distinto, Simona; G., Costa; M., Yanez; Sanna, MARIA LUISA; S., Vigo; Meleddu, Rita; D., Secci
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, S.; Maccioni, Elias; Cardia, MARIA CRISTINA; Yanez, M.; Orallo, F.; Alcaro, S.; Ortuso, F.; Cirilli, R.; Ferretti, R.; Distinto, Simona; Kirchmair, J.; Langer, T.
Tri-substituted thiazolines as promising scaffolds for the design of efficient COX inhibitors
2009-01-01 Maccioni, Elias; Alcaro, S.; Orallo, F.; Cardia, M. C.; Distinto, Simona; Sanna, M. L.; Vigo, S.; Meleddu, R.; Ortuso, F.; Secci, D.; Yanez, M.; Bolasco, A.
Computational approaches for discovery and optimization of monoamine oxidase B inhibitors
2009-01-01 Distinto, Simona; Maccioni, Elias; Alcaro, S.; Orallo, F.; Wolber, G.; Cardia, M. C.; Secci, D.; Bolasco, A.; Ortuso, F.; Sanna, M. L.; Vigo, S.; Yanez, M.; Kirchmair, J.; Markt, P.; Chimenti, F.
Recent advances in monoamine oxidase B inhibitors design
2009-01-01 Chimenti, F.; Maccioni, Elias; Cardia, MARIA CRISTINA; Secci, D.; Bolasco, A.; Alcaro, S.; Ortuso, F.; Orallo, F.; Kirchmair, J.; Markt, P.; Langer, T.; Distinto, Simona
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Sanna M., L; Esposito, Francesca; Cardia M., C; Tramontano, Enzo; Maccioni, Elias | - | - |
Isatin derivatives as new scaffolds for HIV-1 reverse transcriptase associated RNase H and RDDP dual inhibitors | 1-gen-2011 | Corona, Angela; Meleddu, Rita; Esposito, Francesca; Sanna, M. L.; Distinto, Simona; Maccioni, Elias; Tramontano, Enzo | - | - |
Exploring new scaffolds for the inibition of the Ribonuclease H function of RT HIV-1 | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Distinto, S; Esposito, Francesca; Sanna M., L; Cardia M., C; Tramontano, Enzo; Maccioni, Elias | - | - |
A combined shape-, 2D-fingerprint-and pharmacophore-based virtual screening for the identification of dual inhibitors targeting HIV-1 reverse transcriptase. | 1-gen-2011 | Esposito, Francesca; Distinto, Simona; J., Kirchmair; C. M., Cardia; Maccioni, Elias; S., Alcaro; L., Zinzula; E., Tramontano | - | - |
Identification of HIV-1 reverse transcriptase dual inhibitors by a combined shape-, 2D-fingerprint- and pharmacophore-based virtual screening approach | 1-gen-2011 | Distinto, S; Esposito, Francesca; Kirchmair, J; Cardia, Cm; Maccioni, Elias; Alcaro, S; Zinzula, Luca; Tramontano, Enzo | ANTIVIRAL RESEARCH | - |
Semicarbazide-sensitive amine oxidase/vascular adhesion protein-1: a patent survey | 1-gen-2011 | Dunkel, P; Balogh, B; Meleddu, Rita; Maccioni, Elias; Gyires, K; Mátyus, P. | EXPERT OPINION ON THERAPEUTIC PATENTS | - |
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona | JOURNAL OF MEDICINAL CHEMISTRY | - |
SYNTHESIS, MOLECULAR MODELLING, INHIBITORY ACTIVITY, AND SELECTIVITY TOWARDS MONOAMINE OXIDASE OF NEW HETEROCYCLIC SCAFFOLDS | 1-gen-2010 | Sanna M., L; Maccioni, Elias; Alcaro, S; Cirilli, R; Ferretti, R; Yanez, M; Cardia M., C; Distinto, S; Meleddu, Rita; Vigo, S; Ortuso, F. | - | - |
Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach | 1-gen-2010 | Meleddu, Rita; Sanna, M. L.; Distinto, Simona; Esposito, Francesca; Corona, Angela; Ortuso, F.; Alcaro, S.; Maccioni, Elias; Cardia, M. C.; Tramontano, Enzo | - | - |
Shape based computer aided similarity screening: a valid tool in the discovery of new scaffolds for the inhibition of HIV-1 reverse transcriptase associated ribonuclease H function | 1-gen-2010 | Distinto, Simona; Esposito, Francesca; Maccioni, Elias; Cardia, M. C.; Markt, P.; Tramontano, Enzo | - | - |
Brain delivery of the NK3 receptor agonist senktide by immunoliposome: an in vivo microdialysis study | 1-gen-2010 | DE LUCA, MARIA ANTONIETTA; Lai, Francesco; Bimpisidis, Zisis; Manca, MARIA LETIZIA; Maccioni, Elias; Caboni, Pierluigi; Fadda, ANNA MARIA; DI CHIARA, Gaetano | MONITORING MOLECULES IN NEUROSCIENCE | B Westerink, R Clinckers, I Smolders, Y Michotte |
Synthesis, molecular modelling, inhibitory acivity, and selectivity towards monoamine oxidase of new heterocyclic scaffold | 1-gen-2010 | Sanna, M. L.; Maccioni, Elias; Alcaro, S.; Cirilli, R.; Ferretti, R.; Yañez, M.; Cardia, M. C.; Distinto, Simona; Meleddu, R.; Vigo, S.; Ortuso, F. | - | - |
Identification of new scaffolds for the inhibition of HIV-1 Reverse Transcriptase associated Ribonuclease H function by means of shape based similarity screening | 1-gen-2010 | Distinto, Simona; Esposito, Francesca; Maccioni, Elias; Cardia, M. C.; Markt, P.; Tramontano, Enzo; Sanna, M. L.; Meleddu, Rita | - | - |
Semipreparative HPLC enantioseparation, chiroptical properties, and absolute configuration of two novel cyclooxygenase-2 inhibitors | 1-gen-2010 | Cirilli, R; Fiore, S; LA TORRE, F; Maccioni, Elias; Secci, D; Sanna, MARIA LUISA; Faggi, C. | CHIRALITY | - |
Application of an immobilised amylose-based chiral stationary phase to the development of new monoamine oxidase B inhibitors | 1-gen-2010 | Sanna, MARIA LUISA; Maccioni, Elias; Sara, Vigo; Cristina, Faggi; Roberto, Cirilli | TALANTA | - |
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase | 1-gen-2010 | Maccioni, Elias; S., Alcaro; F., Orallo; Cardia, MARIA CRISTINA; Distinto, Simona; G., Costa; M., Yanez; Sanna, MARIA LUISA; S., Vigo; Meleddu, Rita; D., Secci | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 1-gen-2010 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, S.; Maccioni, Elias; Cardia, MARIA CRISTINA; Yanez, M.; Orallo, F.; Alcaro, S.; Ortuso, F.; Cirilli, R.; Ferretti, R.; Distinto, Simona; Kirchmair, J.; Langer, T. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Tri-substituted thiazolines as promising scaffolds for the design of efficient COX inhibitors | 1-gen-2009 | Maccioni, Elias; Alcaro, S.; Orallo, F.; Cardia, M. C.; Distinto, Simona; Sanna, M. L.; Vigo, S.; Meleddu, R.; Ortuso, F.; Secci, D.; Yanez, M.; Bolasco, A. | - | - |
Computational approaches for discovery and optimization of monoamine oxidase B inhibitors | 1-gen-2009 | Distinto, Simona; Maccioni, Elias; Alcaro, S.; Orallo, F.; Wolber, G.; Cardia, M. C.; Secci, D.; Bolasco, A.; Ortuso, F.; Sanna, M. L.; Vigo, S.; Yanez, M.; Kirchmair, J.; Markt, P.; Chimenti, F. | - | - |
Recent advances in monoamine oxidase B inhibitors design | 1-gen-2009 | Chimenti, F.; Maccioni, Elias; Cardia, MARIA CRISTINA; Secci, D.; Bolasco, A.; Alcaro, S.; Ortuso, F.; Orallo, F.; Kirchmair, J.; Markt, P.; Langer, T.; Distinto, Simona | - | S.C. Pandalai |
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