CONGIU, CENZO
CONGIU, CENZO
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
Antagonism of the prokineticin system prevents and reverses allodynia and inflammation in a mouse model of diabetes
2016-01-01 Castelli, M; Amodeo, G; Negri, L; Lattanzi, R; Maftei, D; Gotti, C; Pistillo, F; Onnis, Valentina; Congiu, Cenzo; Panerai, Ae; Sacerdote, P; Franchi, S.
Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor
2015-01-01 Gouveia Figueira, S; Karlsson, J; Deplano, Alessandro; Hashemian, S; Svensson, M; Fredriksson Sundbom, M; Congiu, Cenzo; Onnis, Valentina; Fowler, Cj
Critical role for prokineticin 2 in CNS autoimmunity
2015-01-01 ABOU HAMDAN, M; Costanza, M; Fontana, E; DI DARIO, M; Musio, S; Congiu, Cenzo; Onnis, Valentina; Lattanzi, R; Radaelli, M; Martinelli, V; Salvadori, S; Negri, L; Poliani, Pl; Farina, C; Balboni, Gianfranco; Steinman, L; Pedotti, R.
Design, synthesis, and anti-HIV-1 activity of 1-substituted 3-(3,5-dimethylbenzyl)triazine derivatives
2015-01-01 Sakakibara, Norikazu; Balboni, Gianfranco; Congiu, Cenzo; Onnis, Valentina; Demizu, Yosuke; Misawa, Takashi; Kurihara, Masaaki; Kato, Yoshihisa; Maruyama, Tokumi; Toyama, Masaaki; Okamoto, Mika; Baba, Masanori
Dihydroquinazoline and Triazinedione Derivatives as Prok1 and Prok2 receptor antagonists in HEK-293 transfected cells
2015-01-01 Balboni, Gianfranco; Congiu, Cenzo; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Sbai, Oualid; Rondard, Philippe; Onnis, Valentina
Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel
2015-01-01 Petrocellis, Luciano De; Moriello, Aniello Schiano; Byun, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Vázquez Romero, Ana; Garrido, Maria; Messeguer, Angel; Zhang, Fang Xiong; Zamponi, Gerald W; Deplano, Alessandro; Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Marzo, Vincenzo Di
Interaction of the N-(3-Methylpyridin-2-yl)amide derivatives of flurbiprofen and ibuprofen with FAAH: Enantiomeric selectivity and binding mode
2015-01-01 Karlsson, Jessica; Morgillo, Carmine M; Deplano, Alessandro; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Svensson, Mona; Novellino, Ettore; Congiu, Cenzo; Onnis, Valentina; Catalanotti, Bruno; Fowler, Christopher J.
Investigation of the mechanism of FAAH inhibition of profen amide derivatives
2015-01-01 Morgillo, Cm; Deplano, Alessandro; Demurtas, Monica; Karlosson, J; Onnis, Valentina; Congiu, Cenzo; Fowler, Cj; Catalanotti, B.
PPAR controls pregnancy outcome through activation of EG-VEGF: new insights into the mechanism of placental development
2015-01-01 Vanessa, Garnier; Wael, Traboulsi; Aude, Salomon; Sophie, Brouillet; Thierry, Fournier; Carine, Winkler; Beatrice, Desvergne; Pascale, Hoffmann; Qun Yong, Zhou; Congiu, Cenzo; Onnis, Valentina; Mohamed, Benharouga; Jean Jacques, Feige; Nadia, Alfaidy
Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Ceruso, Mariangela; Supuran, Claudiu T.
Synthesis and evaluation of new pyrazole-based carboxamides as modulators of the TrPv1 channel
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Allarà, Marco; Schiano Moriello, Aniello; Di Marzo, Vincenzo; De Petrocellis, Luciano
Synthesis and SIRT1 modulation studies of amides and hydrazides of benzoic acid incorporating a (2-trifluoromethylpyridin-4-yl)amino moiety
2015-01-01 Congiu, Cenzo; Balboni, Gianfranco; Onnis, Valentina
Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Dedeoglu, Nurcan; Supuran, Claudiu T.
TRPV1 modulators: synthesis and in vitro evaluation of 1-heteroarylpiperidinecarboxamide and piperazinylurea derivatives
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Schiano Moriello, A; Di Marzo, V; De Petrocellis, L.
A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists
2014-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Negri, L; Lattanzi, R; Balboni, Gianfranco
An important role for prokineticin 2 in autoimmune CNS demyelination
2014-01-01 Abou hamdan, M.; Costanza, M.; Fontana, E.; Musio, S.; Di Dario, M.; Congiu, Cenzo; Onnis, Valentina; Lattanzi, R.; Negri, L.; Poliani, P. L.; Farina, C.; Balboni, Gianfranco; Steinman, L.; Pedotti, R.
Design, Synthesis and Evaluation of new 2-(Arylidenehydrazino)pyrrole Derivatives as Potential Antitumor Agents
2014-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Demurtas, M; Balboni, Gianfranco
Design, synthesis and pharmacological investigation on new FAAH inhibitors
2014-01-01 Onnis, Valentina; Congiu, Cenzo; Deplano, Alessandro; Demurtas, M; Cipriano, M; Fowler C., J; Morgillo C., M; Catalanotti, B.
Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization
2014-01-01 Lattanzi, R; Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Francioso, A; Ambrosio, C; Casella, I; Costa, T; Caltabiano, G; Matsoukas M., T; Balboni, Gianfranco; Negri, L.
Interaction and reactivity of synthetic aminoisoflavones with metal-free and metalassociated amyloid-beta
2014-01-01 Detoma, As; Krishnamoorthy, J; Nam, Y; Lee, Hj; Brender, Jr; Kochi, A; Lee, D; Onnis, Valentina; Congiu, Cenzo; Manfredini, S; Vertuani, S; Balboni, Gianfranco; Ramamoorthy, A; Lim, Mh
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Antagonism of the prokineticin system prevents and reverses allodynia and inflammation in a mouse model of diabetes | 1-gen-2016 | Castelli, M; Amodeo, G; Negri, L; Lattanzi, R; Maftei, D; Gotti, C; Pistillo, F; Onnis, Valentina; Congiu, Cenzo; Panerai, Ae; Sacerdote, P; Franchi, S. | PLOS ONE | - |
| Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor | 1-gen-2015 | Gouveia Figueira, S; Karlsson, J; Deplano, Alessandro; Hashemian, S; Svensson, M; Fredriksson Sundbom, M; Congiu, Cenzo; Onnis, Valentina; Fowler, Cj | PLOS ONE | - |
| Critical role for prokineticin 2 in CNS autoimmunity | 1-gen-2015 | ABOU HAMDAN, M; Costanza, M; Fontana, E; DI DARIO, M; Musio, S; Congiu, Cenzo; Onnis, Valentina; Lattanzi, R; Radaelli, M; Martinelli, V; Salvadori, S; Negri, L; Poliani, Pl; Farina, C; Balboni, Gianfranco; Steinman, L; Pedotti, R. | NEUROLOGY® NEUROIMMUNOLOGY & NEUROINFLAMMATION | - |
| Design, synthesis, and anti-HIV-1 activity of 1-substituted 3-(3,5-dimethylbenzyl)triazine derivatives | 1-gen-2015 | Sakakibara, Norikazu; Balboni, Gianfranco; Congiu, Cenzo; Onnis, Valentina; Demizu, Yosuke; Misawa, Takashi; Kurihara, Masaaki; Kato, Yoshihisa; Maruyama, Tokumi; Toyama, Masaaki; Okamoto, Mika; Baba, Masanori | ANTIVIRAL CHEMISTRY & CHEMOTHERAPY | - |
| Dihydroquinazoline and Triazinedione Derivatives as Prok1 and Prok2 receptor antagonists in HEK-293 transfected cells | 1-gen-2015 | Balboni, Gianfranco; Congiu, Cenzo; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Sbai, Oualid; Rondard, Philippe; Onnis, Valentina | - | - |
| Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel | 1-gen-2015 | Petrocellis, Luciano De; Moriello, Aniello Schiano; Byun, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Vázquez Romero, Ana; Garrido, Maria; Messeguer, Angel; Zhang, Fang Xiong; Zamponi, Gerald W; Deplano, Alessandro; Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Marzo, Vincenzo Di | PHARMACOLOGICAL RESEARCH | - |
| Interaction of the N-(3-Methylpyridin-2-yl)amide derivatives of flurbiprofen and ibuprofen with FAAH: Enantiomeric selectivity and binding mode | 1-gen-2015 | Karlsson, Jessica; Morgillo, Carmine M; Deplano, Alessandro; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Svensson, Mona; Novellino, Ettore; Congiu, Cenzo; Onnis, Valentina; Catalanotti, Bruno; Fowler, Christopher J. | PLOS ONE | - |
| Investigation of the mechanism of FAAH inhibition of profen amide derivatives | 1-gen-2015 | Morgillo, Cm; Deplano, Alessandro; Demurtas, Monica; Karlosson, J; Onnis, Valentina; Congiu, Cenzo; Fowler, Cj; Catalanotti, B. | - | - |
| PPAR controls pregnancy outcome through activation of EG-VEGF: new insights into the mechanism of placental development | 1-gen-2015 | Vanessa, Garnier; Wael, Traboulsi; Aude, Salomon; Sophie, Brouillet; Thierry, Fournier; Carine, Winkler; Beatrice, Desvergne; Pascale, Hoffmann; Qun Yong, Zhou; Congiu, Cenzo; Onnis, Valentina; Mohamed, Benharouga; Jean Jacques, Feige; Nadia, Alfaidy | AMERICAN JOURNAL OF PHYSIOLOGY: ENDOCRINOLOGY AND METABOLISM | - |
| Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Ceruso, Mariangela; Supuran, Claudiu T. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Synthesis and evaluation of new pyrazole-based carboxamides as modulators of the TrPv1 channel | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Allarà, Marco; Schiano Moriello, Aniello; Di Marzo, Vincenzo; De Petrocellis, Luciano | - | - |
| Synthesis and SIRT1 modulation studies of amides and hydrazides of benzoic acid incorporating a (2-trifluoromethylpyridin-4-yl)amino moiety | 1-gen-2015 | Congiu, Cenzo; Balboni, Gianfranco; Onnis, Valentina | - | - |
| Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Dedeoglu, Nurcan; Supuran, Claudiu T. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
| TRPV1 modulators: synthesis and in vitro evaluation of 1-heteroarylpiperidinecarboxamide and piperazinylurea derivatives | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Schiano Moriello, A; Di Marzo, V; De Petrocellis, L. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists | 1-gen-2014 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Negri, L; Lattanzi, R; Balboni, Gianfranco | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| An important role for prokineticin 2 in autoimmune CNS demyelination | 1-gen-2014 | Abou hamdan, M.; Costanza, M.; Fontana, E.; Musio, S.; Di Dario, M.; Congiu, Cenzo; Onnis, Valentina; Lattanzi, R.; Negri, L.; Poliani, P. L.; Farina, C.; Balboni, Gianfranco; Steinman, L.; Pedotti, R. | JOURNAL OF NEUROIMMUNOLOGY | - |
| Design, Synthesis and Evaluation of new 2-(Arylidenehydrazino)pyrrole Derivatives as Potential Antitumor Agents | 1-gen-2014 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Demurtas, M; Balboni, Gianfranco | CHEMMEDCHEM | - |
| Design, synthesis and pharmacological investigation on new FAAH inhibitors | 1-gen-2014 | Onnis, Valentina; Congiu, Cenzo; Deplano, Alessandro; Demurtas, M; Cipriano, M; Fowler C., J; Morgillo C., M; Catalanotti, B. | CHEMMEDCHEM | - |
| Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization | 1-gen-2014 | Lattanzi, R; Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Francioso, A; Ambrosio, C; Casella, I; Costa, T; Caltabiano, G; Matsoukas M., T; Balboni, Gianfranco; Negri, L. | INTERNATIONAL JOURNAL OF PHARMACEUTICAL SCIENCES AND RESEARCH | - |
| Interaction and reactivity of synthetic aminoisoflavones with metal-free and metalassociated amyloid-beta | 1-gen-2014 | Detoma, As; Krishnamoorthy, J; Nam, Y; Lee, Hj; Brender, Jr; Kochi, A; Lee, D; Onnis, Valentina; Congiu, Cenzo; Manfredini, S; Vertuani, S; Balboni, Gianfranco; Ramamoorthy, A; Lim, Mh | CHEMICAL SCIENCE | - |