MELEDDU, RITA
MELEDDU, RITA
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis and microbiological evaluation
2009-01-01 Biava, M; Porretta, Gc; Poce, G; DE LOGU, Alessandro; Meleddu, Rita; DE ROSSI, E; Manetti, F; Botta, M.
1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings
2008-01-01 Biava, M; Porretta, Gc; Poce, G; DE LOGU, Alessandro; Saddi, M; Meleddu, Rita; Manetti, F; DE ROSSI, E; Botta, M.
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents
2013-01-01 Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias
2-Acylhydrazino-5-arylpyrrole derivatives: Synthesis and antifungal activity evaluation
2009-01-01 Onnis, Valentina; DE LOGU, Alessandro; Cocco, Mt; Fadda, R; Meleddu, Rita; Congiu, Cenzo
2-methoxynaphthalen thiazole derivate : a new HIV-1 RT Ribonuclease H/DNA polymerase dual inhibitor active on viral replication
2014-01-01 Corona, Angela; Meleddu, R.; Esposito, E.; Distinto, S.; Bianco, G.; Maccioni, E.; Tramontano, E. .
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function
2011-01-01 Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona
A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition
2013-01-01 Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Distinto, Simona; Yañez, M.; Viña, D.; Lamela, M.; Maccioni, Elias
Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase
2011-01-01 Meleddu, Rita; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Distinto, Simona; Sanna, M. L.; Cardia, C.; Alcaro, S.; Maccioni, Elias
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation
2020-01-01 Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F.
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents
2008-01-01 Biava, M; Porretta G., C; Poce, G; DE LOGU, Alessandro; Meleddu, Rita; De Rossi, E; Manetti, F; Botta, M.
Design and synthesis of new isatin derivatives as HIV-1 reverse transcriptase associated ribonuclease H inhibitors
2011-01-01 Esposito, Francesca; Meleddu, R.; Sanna, MARIA LUISA; Distinto, Simona; Corona, Angela; Cannas, Valeria; Tramontano, Enzo; Cardia, MARIA CRISTINA
Design and synthesis of new Isatin derivatives as HIV-1 Reverse Transcriptase associated Ribonuclease H inhibitors twenty-fourth
2011-01-01 Esposito, Francesca; Meleddu, Rita; Sanna M., L; Distinto, S; Corona, Angela; Cannas, V; Tramontano, Enzo; Cardia, M. C.
Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach
2010-01-01 Meleddu, Rita; Sanna, M. L.; Distinto, Simona; Esposito, Francesca; Corona, Angela; Ortuso, F.; Alcaro, S.; Maccioni, Elias; Cardia, M. C.; Tramontano, Enzo
Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors
2011-01-01 Meleddu, Rita; Corona, Angela; Sanna M., L; Esposito, Francesca; Cardia M., C; Tramontano, Enzo; Maccioni, Elias
Design, synthesis and biological activity evaluation of new HIV-1 reverse transcriptase dual inhibitors
2011-01-01 Meleddu, R.; Corona, Angela; Distinto, Simona; Sanna, M. L.; Esposito, Francesca; Cardia, M. C.; Tramontano, Enzo; Maccioni, Elias
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 RT.
2013-01-01 Esposito, Francesca; Meleddu, R; Cannas, V; Distinto, Simona; Del Vecchio, C; Biano, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Single Site Dual Inhibitors of HIV-1 RT
2013-01-01 Esposito, Francesca; Meleddu, R; Cannas, Valeria; Distinto, Simona; Del Vecchio, C; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase
2014-01-01 Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, C; Esposito, Francesca; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Artese, A; Scalise, D; Fresta, M; Arridu, A; Ortuso, F; Maccioni, Elias; Tramontano, Enzo
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| (3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| 1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis and microbiological evaluation | 1-gen-2009 | Biava, M; Porretta, Gc; Poce, G; DE LOGU, Alessandro; Meleddu, Rita; DE ROSSI, E; Manetti, F; Botta, M. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| 1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings | 1-gen-2008 | Biava, M; Porretta, Gc; Poce, G; DE LOGU, Alessandro; Saddi, M; Meleddu, Rita; Manetti, F; DE ROSSI, E; Botta, M. | JOURNAL OF MEDICINAL CHEMISTRY | - |
| 2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents | 1-gen-2013 | Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias | - | - |
| 2-Acylhydrazino-5-arylpyrrole derivatives: Synthesis and antifungal activity evaluation | 1-gen-2009 | Onnis, Valentina; DE LOGU, Alessandro; Cocco, Mt; Fadda, R; Meleddu, Rita; Congiu, Cenzo | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| 2-methoxynaphthalen thiazole derivate : a new HIV-1 RT Ribonuclease H/DNA polymerase dual inhibitor active on viral replication | 1-gen-2014 | Corona, Angela; Meleddu, R.; Esposito, E.; Distinto, S.; Bianco, G.; Maccioni, E.; Tramontano, E. . | - | - |
| 3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias | - | - |
| 3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona | JOURNAL OF MEDICINAL CHEMISTRY | - |
| A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition | 1-gen-2013 | Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Distinto, Simona; Yañez, M.; Viña, D.; Lamela, M.; Maccioni, Elias | JOURNAL OF HETEROCYCLIC CHEMISTRY | - |
| Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Distinto, Simona; Sanna, M. L.; Cardia, C.; Alcaro, S.; Maccioni, Elias | - | - |
| Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation | 1-gen-2020 | Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents | 1-gen-2008 | Biava, M; Porretta G., C; Poce, G; DE LOGU, Alessandro; Meleddu, Rita; De Rossi, E; Manetti, F; Botta, M. | - | - |
| Design and synthesis of new isatin derivatives as HIV-1 reverse transcriptase associated ribonuclease H inhibitors | 1-gen-2011 | Esposito, Francesca; Meleddu, R.; Sanna, MARIA LUISA; Distinto, Simona; Corona, Angela; Cannas, Valeria; Tramontano, Enzo; Cardia, MARIA CRISTINA | ANTIVIRAL RESEARCH | - |
| Design and synthesis of new Isatin derivatives as HIV-1 Reverse Transcriptase associated Ribonuclease H inhibitors twenty-fourth | 1-gen-2011 | Esposito, Francesca; Meleddu, Rita; Sanna M., L; Distinto, S; Corona, Angela; Cannas, V; Tramontano, Enzo; Cardia, M. C. | - | - |
| Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach | 1-gen-2010 | Meleddu, Rita; Sanna, M. L.; Distinto, Simona; Esposito, Francesca; Corona, Angela; Ortuso, F.; Alcaro, S.; Maccioni, Elias; Cardia, M. C.; Tramontano, Enzo | - | - |
| Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Sanna M., L; Esposito, Francesca; Cardia M., C; Tramontano, Enzo; Maccioni, Elias | - | - |
| Design, synthesis and biological activity evaluation of new HIV-1 reverse transcriptase dual inhibitors | 1-gen-2011 | Meleddu, R.; Corona, Angela; Distinto, Simona; Sanna, M. L.; Esposito, Francesca; Cardia, M. C.; Tramontano, Enzo; Maccioni, Elias | - | - |
| Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 RT. | 1-gen-2013 | Esposito, Francesca; Meleddu, R; Cannas, V; Distinto, Simona; Del Vecchio, C; Biano, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo | - | - |
| Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Single Site Dual Inhibitors of HIV-1 RT | 1-gen-2013 | Esposito, Francesca; Meleddu, R; Cannas, Valeria; Distinto, Simona; Del Vecchio, C; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Maccioni, Elias; Tramontano, Enzo | VIROLOGIE | - |
| Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2014 | Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, C; Esposito, Francesca; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Artese, A; Scalise, D; Fresta, M; Arridu, A; Ortuso, F; Maccioni, Elias; Tramontano, Enzo | CHEMMEDCHEM | - |