MACCIONI, ELIAS
MACCIONI, ELIAS
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
1-acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties
2008-01-01 Vigo, S.; Alcaro, S.; Bolasco, A.; Cardia, C.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Sanna, M. L.; Secci, D.; Yanez, M.
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors
2008-01-01 Sanna, M. L.; Alcaro, S.; Bolasco, A.; Cardia, C.; Cirilli, R.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Secci, D.; Vigo, S.; Yanez, M.
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents
2013-01-01 Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function
2011-01-01 Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona
38. A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone
2009-01-01 Franco, Chimenti; Bruna, Bizzarri; Maccioni, Elias; Daniela, Secci; Adriana, Bolasco; Paola, Chimenti; Rossella, Fioravanti; Arianna, Granese; Simone, Carradori; Federica, Tosi; Paola, Ballario; Stefano, Vernarecci; AND PATRIZIA, Filatici
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias
9-fluorenones as new scaffolds for G-quadruplex DNA
2012-01-01 Meleddu, R.; Distinto, Simona; Parrotta, L.; Maccioni, Elias; Musetti, C.; Sissi, C; Sanna, M. L.; Alcaro, S.
A combined shape-, 2D-fingerprint-and pharmacophore-based virtual screening for the identification of dual inhibitors targeting HIV-1 reverse transcriptase.
2011-01-01 Esposito, Francesca; Distinto, Simona; J., Kirchmair; C. M., Cardia; Maccioni, Elias; S., Alcaro; L., Zinzula; E., Tramontano
AN INVESTIGATION INTO THE ELECTRON-IONIZATION-INDUCED MASS-SPECTROMETRIC BEHAVIOR OF SOME TRANS-SUBSTITUTED AND CIS-SUBSTITUTED CYCLOALKYLAMINES OF PHARMACEUTICAL INTEREST
1993-01-01 Anchisi, C; Fadda, ANNA MARIA; Maccioni, Am; Maccioni, Elias; Favretto, D; Traldi, P.
Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions
2006-01-01 Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, A; Chimenti, P; Secci, D; Maccioni, Elias; LA TORRE, F.
Application of an immobilised amylose-based chiral stationary phase to the development of new monoamine oxidase B inhibitors
2010-01-01 Sanna, MARIA LUISA; Maccioni, Elias; Sara, Vigo; Cristina, Faggi; Roberto, Cirilli
Attività di un derivato isotiosemicarbazonico ciclico nei confronti di biofilm di Candida albicans FLC-S e FLC-R in combinazione con AMB
2006-01-01 Saddi, M; Chisu, L; Cardia, Mc; Saddi, B; Maccioni, Elias; DE LOGU, Alessandro
Aumento della sensibilità all’AmB di biofilm di Candida albicans fluconazolo-resistente nell’impiego combinato con derivati ciclici isotiosemicarbazonici
2006-01-01 Saddi, M; Cardia, Mc; Chisu, L; Borgna, R; Maccioni, Elias; Saddi, B; DE LOGU, Alessandro
Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitors
2016-01-01 Schneider, Anna; Corona, Angela; Spöring, Imke; Jordan, Mareike; Buchholz, Bernd; Maccioni, Elias; Di Santo, Roberto; Bodem, Jochen; Tramontano, Enzo; Wöhrl, Birgitta M.
Brain delivery of the NK3 receptor agonist senktide by immunoliposome: an in vivo microdialysis study
2010-01-01 DE LUCA, MARIA ANTONIETTA; Lai, Francesco; Bimpisidis, Zisis; Manca, MARIA LETIZIA; Maccioni, Elias; Caboni, Pierluigi; Fadda, ANNA MARIA; DI CHIARA, Gaetano
Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase
2011-01-01 Meleddu, Rita; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Distinto, Simona; Sanna, M. L.; Cardia, C.; Alcaro, S.; Maccioni, Elias
Characterization of 2,5-diaryl-1,3,4-oxadiazolines by multinuclear magnetic resonance and density functional theory calculations. Investigation on a case of very remote Hammett correlation
2009-01-01 Cerioni, Giovanni; Maccioni, Elias; Cardia, MARIA CRISTINA; Vigo, Sara; Mocci, Francesca
Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity
2019-01-01 Esposito, F.; Ambrosio, F. A.; Maleddu, R.; Costa, G.; Rocca, R.; Maccioni, E.; Catalano, R.; Romeo, I.; Eleftheriou, P.; Karia, D. C.; Tsirides, P.; Godvani, N.; Pandya, H.; Corona, A.; Alcaro, S.; Artese, A.; Geronikaki, A.; Tramontano, E.
Combining induced fit docking and molecular dynamics simulations to predict the binding mode of new monoamine oxidase B inhibitors
2008-01-01 Distinto, Simona; Maccioni, Elias; Alcaro, S.; Orallo, F.; Wolber, G.; Cardia, M. C.; Secci, D.; Bolasco, A.; Ortuso, F.; Sanna, M. L.; Vigo, S.; Yanez, M.; Kirchmair, J.; Markt, P.; Chimenti, F.
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| 1-acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties | 1-gen-2008 | Vigo, S.; Alcaro, S.; Bolasco, A.; Cardia, C.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Sanna, M. L.; Secci, D.; Yanez, M. | - | - |
| 1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors | 1-gen-2008 | Sanna, M. L.; Alcaro, S.; Bolasco, A.; Cardia, C.; Cirilli, R.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Secci, D.; Vigo, S.; Yanez, M. | - | - |
| 2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents | 1-gen-2013 | Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias | - | - |
| 3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias | - | - |
| 3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona | JOURNAL OF MEDICINAL CHEMISTRY | - |
| 38. A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone | 1-gen-2009 | Franco, Chimenti; Bruna, Bizzarri; Maccioni, Elias; Daniela, Secci; Adriana, Bolasco; Paola, Chimenti; Rossella, Fioravanti; Arianna, Granese; Simone, Carradori; Federica, Tosi; Paola, Ballario; Stefano, Vernarecci; AND PATRIZIA, Filatici | JOURNAL OF MEDICINAL CHEMISTRY | - |
| (3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| 9-fluorenones as new scaffolds for G-quadruplex DNA | 1-gen-2012 | Meleddu, R.; Distinto, Simona; Parrotta, L.; Maccioni, Elias; Musetti, C.; Sissi, C; Sanna, M. L.; Alcaro, S. | - | - |
| A combined shape-, 2D-fingerprint-and pharmacophore-based virtual screening for the identification of dual inhibitors targeting HIV-1 reverse transcriptase. | 1-gen-2011 | Esposito, Francesca; Distinto, Simona; J., Kirchmair; C. M., Cardia; Maccioni, Elias; S., Alcaro; L., Zinzula; E., Tramontano | - | - |
| AN INVESTIGATION INTO THE ELECTRON-IONIZATION-INDUCED MASS-SPECTROMETRIC BEHAVIOR OF SOME TRANS-SUBSTITUTED AND CIS-SUBSTITUTED CYCLOALKYLAMINES OF PHARMACEUTICAL INTEREST | 1-gen-1993 | Anchisi, C; Fadda, ANNA MARIA; Maccioni, Am; Maccioni, Elias; Favretto, D; Traldi, P. | RAPID COMMUNICATIONS IN MASS SPECTROMETRY | - |
| Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions | 1-gen-2006 | Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, A; Chimenti, P; Secci, D; Maccioni, Elias; LA TORRE, F. | JOURNAL OF CHROMATOGRAPHY A | - |
| Application of an immobilised amylose-based chiral stationary phase to the development of new monoamine oxidase B inhibitors | 1-gen-2010 | Sanna, MARIA LUISA; Maccioni, Elias; Sara, Vigo; Cristina, Faggi; Roberto, Cirilli | TALANTA | - |
| Attività di un derivato isotiosemicarbazonico ciclico nei confronti di biofilm di Candida albicans FLC-S e FLC-R in combinazione con AMB | 1-gen-2006 | Saddi, M; Chisu, L; Cardia, Mc; Saddi, B; Maccioni, Elias; DE LOGU, Alessandro | - | - |
| Aumento della sensibilità all’AmB di biofilm di Candida albicans fluconazolo-resistente nell’impiego combinato con derivati ciclici isotiosemicarbazonici | 1-gen-2006 | Saddi, M; Cardia, Mc; Chisu, L; Borgna, R; Maccioni, Elias; Saddi, B; DE LOGU, Alessandro | - | - |
| Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitors | 1-gen-2016 | Schneider, Anna; Corona, Angela; Spöring, Imke; Jordan, Mareike; Buchholz, Bernd; Maccioni, Elias; Di Santo, Roberto; Bodem, Jochen; Tramontano, Enzo; Wöhrl, Birgitta M. | NUCLEIC ACIDS RESEARCH | - |
| Brain delivery of the NK3 receptor agonist senktide by immunoliposome: an in vivo microdialysis study | 1-gen-2010 | DE LUCA, MARIA ANTONIETTA; Lai, Francesco; Bimpisidis, Zisis; Manca, MARIA LETIZIA; Maccioni, Elias; Caboni, Pierluigi; Fadda, ANNA MARIA; DI CHIARA, Gaetano | MONITORING MOLECULES IN NEUROSCIENCE | B Westerink, R Clinckers, I Smolders, Y Michotte |
| Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2011 | Meleddu, Rita; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Distinto, Simona; Sanna, M. L.; Cardia, C.; Alcaro, S.; Maccioni, Elias | - | - |
| Characterization of 2,5-diaryl-1,3,4-oxadiazolines by multinuclear magnetic resonance and density functional theory calculations. Investigation on a case of very remote Hammett correlation | 1-gen-2009 | Cerioni, Giovanni; Maccioni, Elias; Cardia, MARIA CRISTINA; Vigo, Sara; Mocci, Francesca | MAGNETIC RESONANCE IN CHEMISTRY | - |
| Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity | 1-gen-2019 | Esposito, F.; Ambrosio, F. A.; Maleddu, R.; Costa, G.; Rocca, R.; Maccioni, E.; Catalano, R.; Romeo, I.; Eleftheriou, P.; Karia, D. C.; Tsirides, P.; Godvani, N.; Pandya, H.; Corona, A.; Alcaro, S.; Artese, A.; Geronikaki, A.; Tramontano, E. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Combining induced fit docking and molecular dynamics simulations to predict the binding mode of new monoamine oxidase B inhibitors | 1-gen-2008 | Distinto, Simona; Maccioni, Elias; Alcaro, S.; Orallo, F.; Wolber, G.; Cardia, M. C.; Secci, D.; Bolasco, A.; Ortuso, F.; Sanna, M. L.; Vigo, S.; Yanez, M.; Kirchmair, J.; Markt, P.; Chimenti, F. | - | - |