MACCIONI, ELIAS
MACCIONI, ELIAS
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias
1-acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties
2008-01-01 Vigo, S.; Alcaro, S.; Bolasco, A.; Cardia, C.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Sanna, M. L.; Secci, D.; Yanez, M.
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors
2008-01-01 Sanna, M. L.; Alcaro, S.; Bolasco, A.; Cardia, C.; Cirilli, R.; Distinto, Simona; Maccioni, Elias; Orallo, F.; Ortuso, F.; Secci, D.; Vigo, S.; Yanez, M.
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents
2013-01-01 Arridu, A.; Meleddu, R.; Bianco, Giulia; Distinto, Simona; DE LOGU, Alessandro; Matyus, P.; Maccioni, Elias
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function
2011-01-01 Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, Elias; Alcaro, S.; Cirilli, R.; Vigo, S.; Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Yanez, M.; Costa, G.; Casu, Laura; Matyus, P.; Distinto, Simona
38. A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone
2009-01-01 Franco, Chimenti; Bruna, Bizzarri; Maccioni, Elias; Daniela, Secci; Adriana, Bolasco; Paola, Chimenti; Rossella, Fioravanti; Arianna, Granese; Simone, Carradori; Federica, Tosi; Paola, Ballario; Stefano, Vernarecci; AND PATRIZIA, Filatici
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action
2023-01-01 Corona, A.; Meleddu, R.; Delelis, O.; Subra, F.; Cottiglia, F.; Esposito, F.; Distinto, S.; Maccioni, E.; Tramontano, E.
9-fluorenones as new scaffolds for G-quadruplex DNA
2012-01-01 Meleddu, R.; Distinto, Simona; Parrotta, L.; Maccioni, Elias; Musetti, C.; Sissi, C; Sanna, M. L.; Alcaro, S.
A combined shape-, 2D-fingerprint-and pharmacophore-based virtual screening for the identification of dual inhibitors targeting HIV-1 reverse transcriptase.
2011-01-01 Esposito, Francesca; Distinto, Simona; J., Kirchmair; C. M., Cardia; Maccioni, Elias; S., Alcaro; L., Zinzula; E., Tramontano
A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition
2013-01-01 Cardia, MARIA CRISTINA; Sanna, MARIA LUISA; Meleddu, Rita; Distinto, Simona; Yañez, M.; Viña, D.; Lamela, M.; Maccioni, Elias
AN INVESTIGATION INTO THE ELECTRON-IONIZATION-INDUCED MASS-SPECTROMETRIC BEHAVIOR OF SOME TRANS-SUBSTITUTED AND CIS-SUBSTITUTED CYCLOALKYLAMINES OF PHARMACEUTICAL INTEREST
1993-01-01 Anchisi, C; Fadda, ANNA MARIA; Maccioni, Am; Maccioni, Elias; Favretto, D; Traldi, P.
An investigation of the biological effect of structural modifications of isothiosemicarbazones and their cyclic analogues
2003-01-01 Maccioni, Elias; Cardia, MARIA CRISTINA; Distinto, Simona; Bonsignore, L.; DE LOGU, Alessandro
Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions
2006-01-01 Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, A; Chimenti, P; Secci, D; Maccioni, Elias; LA TORRE, F.
Anticancer Activity of Sunitinib Analogues in Human Pancreatic Cancer Cell Cultures under Normoxia and Hypoxia
2023-01-01 Skaraite, I.; Maccioni, E.; Petrikaite, V.
Application of an immobilised amylose-based chiral stationary phase to the development of new monoamine oxidase B inhibitors
2010-01-01 Sanna, MARIA LUISA; Maccioni, Elias; Sara, Vigo; Cristina, Faggi; Roberto, Cirilli
Attività di un derivato isotiosemicarbazonico ciclico nei confronti di biofilm di Candida albicans FLC-S e FLC-R in combinazione con AMB
2006-01-01 Saddi, M; Chisu, L; Cardia, Mc; Saddi, B; Maccioni, Elias; DE LOGU, Alessandro
Aumento della sensibilità all’AmB di biofilm di Candida albicans fluconazolo-resistente nell’impiego combinato con derivati ciclici isotiosemicarbazonici
2006-01-01 Saddi, M; Cardia, Mc; Chisu, L; Borgna, R; Maccioni, Elias; Saddi, B; DE LOGU, Alessandro
Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitors
2016-01-01 Schneider, Anna; Corona, Angela; Spöring, Imke; Jordan, Mareike; Buchholz, Bernd; Maccioni, Elias; Di Santo, Roberto; Bodem, Jochen; Tramontano, Enzo; Wöhrl, Birgitta M.
Brain delivery of the NK3 receptor agonist senktide by immunoliposome: an in vivo microdialysis study
2010-01-01 DE LUCA, MARIA ANTONIETTA; Lai, Francesco; Bimpisidis, Zisis; Manca, MARIA LETIZIA; Maccioni, Elias; Caboni, Pierluigi; Fadda, ANNA MARIA; DI CHIARA, Gaetano