COTTIGLIA, FILIPPO

COTTIGLIA, FILIPPO  

DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE  

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Risultati 1 - 20 di 75 (tempo di esecuzione: 0.027 secondi).
Titolo Data di pubblicazione Autore(i) Rivista Editore
Limonoids from Melia azeradach fruits as inhibitors of Flaviviruses In corso di stampa Sanna, Giuseppina; Madeddu, S; Giliberti, G; La Colla, P; Cottiglia, Filippo; Ntali, N; Caboni, Pierluigi ANTIVIRAL RESEARCH -
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPβ phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea 1-gen-2024 Huang, Shiu-Wen; Hsu, Ming Jen; Chen, Hsiu-Chen; Meleddu, Rita; Distinto, Simona; Maccioni, Elias; Cottiglia, Filippo JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action 1-gen-2023 Corona, A.; Meleddu, R.; Delelis, O.; Subra, F.; Cottiglia, F.; Esposito, F.; Distinto, S.; Maccioni, E.; Tramontano, E. FRONTIERS IN CELLULAR AND INFECTION MICROBIOLOGY -
Effects of docosanyl ferulate, a constituent of Withania somnifera, on ethanol- and morphine-elicited conditioned place preference and ERK phosphorylation in the accumbens shell of CD1 mice 1-gen-2022 Maccioni, R.; Serra, M.; Marongiu, J.; Cottiglia, F.; Maccioni, E.; Bassareo, V.; Morelli, M.; Kasture, S. B.; Acquas, E. PSYCHOPHARMACOLOGY -
Formulation and In Vitro Efficacy Assessment of Teucrium marum Extract Loading Hyalurosomes Enriched with Tween 80 and Glycerol 1-gen-2022 Firoznezhad, M.; Castangia, I.; Tuberoso, C. I. G.; Cottiglia, F.; Marongiu, F.; Porceddu, M.; Usach, I.; Escribano-Ferrer, E.; Manca, M. L.; Manconi, M. NANOMATERIALS -
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions 1-gen-2021 Meleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Mátyus, Péter; Maccioni, Elias MOLECULES -
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function 1-gen-2021 Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives 1-gen-2021 Meleddu, R.; Deplano, S.; Maccioni, E.; Ortuso, F.; Cottiglia, F.; Secci, D.; Onali, A.; Sanna, E.; Angeli, A.; Angius, R.; Alcaro, S.; Supuran, C. T.; Distinto, S. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
The biologically active compound of Withania somnifera (L.) Dunal, docosanyl ferulate, is endowed with potent anxiolytic properties but devoid of typical benzodiazepine-like side effects 1-gen-2021 Maccioni, R.; Cottiglia, F.; Maccioni, E.; Talani, G.; Sanna, E.; Bassareo, V.; Kasture, S. B.; Acquas, E. JOURNAL OF PSYCHOPHARMACOLOGY -
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation 1-gen-2020 Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII 1-gen-2020 Meleddu, R.; Distinto, S.; Cottiglia, F.; Angius, R.; Caboni, P.; Angeli, A.; Melis, C.; Deplano, S.; Alcaro, S.; Ortuso, F.; Supuran, C. T.; Maccioni, E. ACS MEDICINAL CHEMISTRY LETTERS -
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases 1-gen-2019 Distinto, S.; Meleddu, R.; Ortuso, F.; Cottiglia, F.; Deplano, S.; SOUSA SEQUEIRA, ANA LISA; Melis, C.; Fois, B.; Angeli, A.; Capasso, C.; Angius, Riccardo; Alcaro, S.; Supuran, C. T.; Maccioni, E. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators 1-gen-2019 Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACCHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe JOURNAL OF NATURAL PRODUCTS -
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids 1-gen-2019 Meleddu, Rita; Petrikaite, Vilma; Distinto, Simona; Arridu, Antonella; Angius, Rossella; Serusi, Lorenzo; Škarnulytė, Laura; Endriulaitytė, Ugnė; Paškevičiu̅tė, Miglė; Cottiglia, Filippo; Gaspari, Marco; Taverna, Domenico; Deplano, Serenella; Fois, Benedetta; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS -
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors 1-gen-2018 Melis, Claudia; Distinto, Simona; Bianco, Giulia; Meleddu, Rita; Cottiglia, Filippo; Fois, Benedetta; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS -
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides 1-gen-2018 Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Gaspari, Marco; Taverna, Domenico; Melis, Claudia; Angeli, Andrea; Bianco, Giulia; Deplano, Serenella; Fois, Benedetta; Del Prete, Sonia; Capasso, Clemente; Alcaro, Stefano; Ortuso, Francesco; Yanez, Matilde; Supuran Claudiu, T.; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS -
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2017 Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia; Cottiglia, Filippo; Maccioni, Elias JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors 1-gen-2017 Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clemente; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, Elias JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action 1-gen-2017 Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo PATHOGENS AND DISEASE -
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms 1-gen-2017 Bianco, Giulia; Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Gaspari, Marco; Melis, Claudia; Corona, Angela; Angius, Rossella; Angeli, Andrea; Taverna, Domenico; Alcaro, Stefano; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T.; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS -