PORCU, ALESSANDRA
PORCU, ALESSANDRA
DIPARTIMENTO DI SCIENZE BIOMEDICHE
COR758, a negative allosteric modulator of GABAB receptors
2021-01-01 Porcu, A.; Mostallino, R.; Serra, V.; Melis, M.; Sogos, V.; Beggiato, S.; Ferraro, L.; Manetti, F.; Gianibbi, B.; Bettler, B.; Corelli, F.; Mugnaini, C.; Castelli, M. P.
Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a G alpha(i/o) protein inhibitor
2018-01-01 Porcu, Alessandra; Melis, Miriam; Turecek, Rostislav; Ullrich, Celine; Mocci, Ignazia; Bettler, Bernhard; Luigi Gessa, Gian; Castelli, MARIA PAOLA
Cannabis and the Use of Amphetamine-Like Substances
2017-01-01 Porcu, Alessandra; Castelli, MARIA PAOLA
Characterization of Rimonabant effects on G protein activity
2016-03-08
In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator
2016-01-01 Porcu, Alessandra; Lobina, Carla; Giunta, Daniela; Solinas, Maurizio; Mugnaini, Claudia; Castelli, MARIA PAOLA
Native CB1 receptor affinity, intrinsic activity and accumbens shell dopamine stimulant properties of third generation SPICE/K2 cannabinoids: BB-22, 5F-PB-22, 5F-AKB-48 and STS-135
2016-01-01 DE LUCA, MARIA ANTONIETTA; Castelli, MARIA PAOLA; Loi, B; Porcu, Alessandra; Martorelli, Mariella; Miliano, Cristina; Kellett, K; Davidson, C; Stair, Jl; Schifano, F; DI CHIARA, Gaetano
Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor
2013-01-01 Mugnaini, C; Pedani, V; Casu, A; Lobina, C; Casti, Alberto; Maccioni, P; Porcu, Alessandra; Giunta, D; Lamponi, S; Solinas, M; Dragoni, S; Valoti, M; Colombo, G; Castelli, MARIA PAOLA; Gessa, Gl; Corelli, F.
The new compound GET73, N-[(4-trifluoromethyl)benzyl]4-methoxybutyramide, regulates hippocampal aminoacidergic transmission possibly via an allosteric modulation of mGlu5 receptor. Behavioural evidence of its "anti-alcohol" and anxiolytic properties.
2013-01-01 Ferraro, L.; Loche, A.; Beggiato, S.; Tomasini, M. C.; Antonelli, T.; Colombo, G.; Lobina, C.; Carai, M. A. M.; Porcu, Alessandra; Castelli, MARIA PAOLA; Clerici, F.; Borelli, A. C.; Cacciaglia, R.; Tanganelli, S.
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| COR758, a negative allosteric modulator of GABAB receptors | 1-gen-2021 | Porcu, A.; Mostallino, R.; Serra, V.; Melis, M.; Sogos, V.; Beggiato, S.; Ferraro, L.; Manetti, F.; Gianibbi, B.; Bettler, B.; Corelli, F.; Mugnaini, C.; Castelli, M. P. | NEUROPHARMACOLOGY | - |
| Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a G alpha(i/o) protein inhibitor | 1-gen-2018 | Porcu, Alessandra; Melis, Miriam; Turecek, Rostislav; Ullrich, Celine; Mocci, Ignazia; Bettler, Bernhard; Luigi Gessa, Gian; Castelli, MARIA PAOLA | NEUROPHARMACOLOGY | - |
| Cannabis and the Use of Amphetamine-Like Substances | 1-gen-2017 | Porcu, Alessandra; Castelli, MARIA PAOLA | - | Elsevier |
| Characterization of Rimonabant effects on G protein activity | 8-mar-2016 | - | - | Università degli Studi di Cagliari |
| In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator | 1-gen-2016 | Porcu, Alessandra; Lobina, Carla; Giunta, Daniela; Solinas, Maurizio; Mugnaini, Claudia; Castelli, MARIA PAOLA | EUROPEAN JOURNAL OF PHARMACOLOGY | - |
| Native CB1 receptor affinity, intrinsic activity and accumbens shell dopamine stimulant properties of third generation SPICE/K2 cannabinoids: BB-22, 5F-PB-22, 5F-AKB-48 and STS-135 | 1-gen-2016 | DE LUCA, MARIA ANTONIETTA; Castelli, MARIA PAOLA; Loi, B; Porcu, Alessandra; Martorelli, Mariella; Miliano, Cristina; Kellett, K; Davidson, C; Stair, Jl; Schifano, F; DI CHIARA, Gaetano | NEUROPHARMACOLOGY | - |
| Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor | 1-gen-2013 | Mugnaini, C; Pedani, V; Casu, A; Lobina, C; Casti, Alberto; Maccioni, P; Porcu, Alessandra; Giunta, D; Lamponi, S; Solinas, M; Dragoni, S; Valoti, M; Colombo, G; Castelli, MARIA PAOLA; Gessa, Gl; Corelli, F. | JOURNAL OF MEDICINAL CHEMISTRY | - |
| The new compound GET73, N-[(4-trifluoromethyl)benzyl]4-methoxybutyramide, regulates hippocampal aminoacidergic transmission possibly via an allosteric modulation of mGlu5 receptor. Behavioural evidence of its "anti-alcohol" and anxiolytic properties. | 1-gen-2013 | Ferraro, L.; Loche, A.; Beggiato, S.; Tomasini, M. C.; Antonelli, T.; Colombo, G.; Lobina, C.; Carai, M. A. M.; Porcu, Alessandra; Castelli, MARIA PAOLA; Clerici, F.; Borelli, A. C.; Cacciaglia, R.; Tanganelli, S. | CURRENT MEDICINAL CHEMISTRY | - |