Sfoglia per Autore
Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2020-01-01 Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Treatment With the Delta Opioid Agonist UFP-512 Alleviates Chronic Inflammatory and Neuropathic Pain: Mechanisms Implicated
2019-01-01 Polo, Sara; Díaz, Andrés Felipe; Gallardo, Núria; Leánez, Sergi; Balboni, Gianfranco; Pol, Olga
δ-Opioid Receptor Activation Attenuates Hypoxia/MPP+-Induced Downregulation of PINK1: a Novel Mechanism of Neuroprotection Against Parkinsonian Injury
2019-01-01 Xu, Yuan; Zhi, Feng; Peng, Ya; Shao, Naiyuan; Khiati, Dhiaedin; Balboni, Gianfranco; Yang, Yilin; Xia, Ying
The prokineticin receptor antagonist PC1 rescues memory impairment induced by β amyloid administration through the modulation of prokineticin system
2019-01-01 Maftei, Daniela; Ratano, Patrizia; Fusco, Ilaria; Marconi, Veronica; Squillace, Silvia; Negri, Lucia; Severini, Cinzia; Balboni, Gianfranco; Steardo, Luca; Bronzuoli, Maria Rosanna; Scuderi, Caterina; Campolongo, Patrizia; Lattanzi, Roberta
Antagonistic Activity of Naphthoquinone-Based Hybrids toward Amyloids Associated with Alzheimer's Disease and Type-2 Diabetes
2019-01-01 Tyrrell, PAUL ANTHONY; Viswanathan, G. K.; Mahapatra, S.; Balboni, G.; Pacifico, S.; Gazit, E.; Segal, D.
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation
2019-01-01 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Targeting prokineticin system counteracts hypersensitivity, neuroinflammation, and tissue damage in a mouse model of bortezomib-induced peripheral neuropathy
2019-01-01 Moschetti, Giorgia; Amodeo, Giada; Maftei, Daniela; Lattanzi, Roberta; Procacci, Patrizia; Sartori, Patrizia; Balboni, Gianfranco; Onnis, Valentina; Conte, Vincenzo; Panerai, Alberto; Sacerdote, Paola; Franchi, Silvia
Prokineticin 2 promotes and sustains neuroinflammation in vincristine treated mice: Focus on pain and emotional like behavior
2019-01-01 Moschetti, G.; Amodeo, G.; Paladini, M. S.; Molteni, R.; Balboni, G.; Panerai, A.; Sacerdote, P.; Franchi, S.
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors
2019-01-01 Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gianfranco; Onnis, Valentina; Potter, Barry V. L.
Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones
2019-01-01 Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity
2018-01-01 Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2018-01-01 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T.
Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy
2018-01-01 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T.
Antagonism of EG-VEGF receptors is a novel targeted therapy for choriocarcinoma progression: in vitro, in vivo and in clinical studies
2017-01-01 Traboulsi, Wael; Sergent, Fréderic; Brouillet, Sophie; Boufettal, Houssine; Hoffmann, Pascale; Zhou, Qun yong; Balboni, Gianfranco; Aboussaouira, Touria; Feige, Jean jacques; Benharouga, Mohamed; Alfaidy, Nadia
3,4-Dihydroquinazoline derivatives inhibit the activities of cholinesterase enzymes
2017-01-01 Park, Byeongyeon; Nam, Ji Hye; Kim, Jin Han; Kim, Hyoung Ja; Onnis, Valentina; Balboni, Gianfranco; Lee, Kyung Tae; Park, Jeong Ho; Catto, Marco; Carotti, Angelo; Lee, Jae Yeol
Antagonism of EG-VEGF receptors as targeted therapy for choriocarcinoma progression in vitro and in vivo
2017-01-01 Traboulsi, Wael; Sergent, Frederic; Boufettal, Houssine; Brouillet, Sophie; Slim, Rima; Hoffmann, Pascale; Benlahfid, Mohammed; Zhou, qun yong; Balboni, Gianfranco; Onnis, Valentina; Bolze, Pierre Adrien; Salomon, Aude; Sauthier, Philippe; Mallet, François; Aboussaouira, Touria; Feige, Jean Jacques; Benharouga, Mohamed; Alfaidy, Nadia
Prokineticin system modulation as a new target to counteract the amyloid beta toxicity induced by glutamatergic alterations in an in vitro model of Alzheimer's disease
2017-01-01 Caioli, Silvia; Severini, Cinzia; Ciotti, Teresa; Florenzano, Fulvio; Pimpinella, Domenico; Petrocchi Passeri, Pamela; Balboni, Gianfranco; Polisca, Patrizio; Lattanzi, Roberta; Nisticò, Robert; Negri, Lucia; Zona, Cristina
Genetically Encodable Bacterial Flavin Transferase for Fluorogenic Protein Modification in Mammalian Cells
2017-01-01 Kang, Myeong Gyun; Park, Jumi; Balboni, Gianfranco; Lim, Mi Hee; Lee, Changwook; Rhee, Hyun Woo
DESIGN, SYNTHESIS AND PHARMACOLOGICAL INVESTIGATION OF NEW DNA METHYLTRANSFERASE INHIBITORS
2016-01-01 Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Arimondo, Paola B.; Masson, Veronique; Onnis, Valentina
DIHYDROQUINAZOLINE BENZYLAMIDES AS ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE INHIBITORS
2016-01-01 Onnis, Valentina; Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Catto, Marco; Pisani, Leonardo; Carotti, Angelo
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 1-gen-2020 | Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Treatment With the Delta Opioid Agonist UFP-512 Alleviates Chronic Inflammatory and Neuropathic Pain: Mechanisms Implicated | 1-gen-2019 | Polo, Sara; Díaz, Andrés Felipe; Gallardo, Núria; Leánez, Sergi; Balboni, Gianfranco; Pol, Olga | FRONTIERS IN PHARMACOLOGY | - |
| δ-Opioid Receptor Activation Attenuates Hypoxia/MPP+-Induced Downregulation of PINK1: a Novel Mechanism of Neuroprotection Against Parkinsonian Injury | 1-gen-2019 | Xu, Yuan; Zhi, Feng; Peng, Ya; Shao, Naiyuan; Khiati, Dhiaedin; Balboni, Gianfranco; Yang, Yilin; Xia, Ying | MOLECULAR NEUROBIOLOGY | - |
| The prokineticin receptor antagonist PC1 rescues memory impairment induced by β amyloid administration through the modulation of prokineticin system | 1-gen-2019 | Maftei, Daniela; Ratano, Patrizia; Fusco, Ilaria; Marconi, Veronica; Squillace, Silvia; Negri, Lucia; Severini, Cinzia; Balboni, Gianfranco; Steardo, Luca; Bronzuoli, Maria Rosanna; Scuderi, Caterina; Campolongo, Patrizia; Lattanzi, Roberta | NEUROPHARMACOLOGY | - |
| Antagonistic Activity of Naphthoquinone-Based Hybrids toward Amyloids Associated with Alzheimer's Disease and Type-2 Diabetes | 1-gen-2019 | Tyrrell, PAUL ANTHONY; Viswanathan, G. K.; Mahapatra, S.; Balboni, G.; Pacifico, S.; Gazit, E.; Segal, D. | ACS CHEMICAL NEUROSCIENCE | - |
| Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation | 1-gen-2019 | Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Targeting prokineticin system counteracts hypersensitivity, neuroinflammation, and tissue damage in a mouse model of bortezomib-induced peripheral neuropathy | 1-gen-2019 | Moschetti, Giorgia; Amodeo, Giada; Maftei, Daniela; Lattanzi, Roberta; Procacci, Patrizia; Sartori, Patrizia; Balboni, Gianfranco; Onnis, Valentina; Conte, Vincenzo; Panerai, Alberto; Sacerdote, Paola; Franchi, Silvia | JOURNAL OF NEUROINFLAMMATION | - |
| Prokineticin 2 promotes and sustains neuroinflammation in vincristine treated mice: Focus on pain and emotional like behavior | 1-gen-2019 | Moschetti, G.; Amodeo, G.; Paladini, M. S.; Molteni, R.; Balboni, G.; Panerai, A.; Sacerdote, P.; Franchi, S. | BRAIN BEHAVIOR AND IMMUNITY | - |
| Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors | 1-gen-2019 | Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gianfranco; Onnis, Valentina; Potter, Barry V. L. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones | 1-gen-2019 | Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | BIOORGANIC CHEMISTRY | - |
| Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity | 1-gen-2018 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 1-gen-2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T. | BIOORGANIC CHEMISTRY | - |
| Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy | 1-gen-2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T. | BIOORGANIC CHEMISTRY | - |
| Antagonism of EG-VEGF receptors is a novel targeted therapy for choriocarcinoma progression: in vitro, in vivo and in clinical studies | 1-gen-2017 | Traboulsi, Wael; Sergent, Fréderic; Brouillet, Sophie; Boufettal, Houssine; Hoffmann, Pascale; Zhou, Qun yong; Balboni, Gianfranco; Aboussaouira, Touria; Feige, Jean jacques; Benharouga, Mohamed; Alfaidy, Nadia | PLACENTA | - |
| 3,4-Dihydroquinazoline derivatives inhibit the activities of cholinesterase enzymes | 1-gen-2017 | Park, Byeongyeon; Nam, Ji Hye; Kim, Jin Han; Kim, Hyoung Ja; Onnis, Valentina; Balboni, Gianfranco; Lee, Kyung Tae; Park, Jeong Ho; Catto, Marco; Carotti, Angelo; Lee, Jae Yeol | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | Elsevier Ltd |
| Antagonism of EG-VEGF receptors as targeted therapy for choriocarcinoma progression in vitro and in vivo | 1-gen-2017 | Traboulsi, Wael; Sergent, Frederic; Boufettal, Houssine; Brouillet, Sophie; Slim, Rima; Hoffmann, Pascale; Benlahfid, Mohammed; Zhou, qun yong; Balboni, Gianfranco; Onnis, Valentina; Bolze, Pierre Adrien; Salomon, Aude; Sauthier, Philippe; Mallet, François; Aboussaouira, Touria; Feige, Jean Jacques; Benharouga, Mohamed; Alfaidy, Nadia | CLINICAL CANCER RESEARCH | - |
| Prokineticin system modulation as a new target to counteract the amyloid beta toxicity induced by glutamatergic alterations in an in vitro model of Alzheimer's disease | 1-gen-2017 | Caioli, Silvia; Severini, Cinzia; Ciotti, Teresa; Florenzano, Fulvio; Pimpinella, Domenico; Petrocchi Passeri, Pamela; Balboni, Gianfranco; Polisca, Patrizio; Lattanzi, Roberta; Nisticò, Robert; Negri, Lucia; Zona, Cristina | NEUROPHARMACOLOGY | - |
| Genetically Encodable Bacterial Flavin Transferase for Fluorogenic Protein Modification in Mammalian Cells | 1-gen-2017 | Kang, Myeong Gyun; Park, Jumi; Balboni, Gianfranco; Lim, Mi Hee; Lee, Changwook; Rhee, Hyun Woo | ACS SYNTHETIC BIOLOGY | - |
| DESIGN, SYNTHESIS AND PHARMACOLOGICAL INVESTIGATION OF NEW DNA METHYLTRANSFERASE INHIBITORS | 1-gen-2016 | Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Arimondo, Paola B.; Masson, Veronique; Onnis, Valentina | - | - |
| DIHYDROQUINAZOLINE BENZYLAMIDES AS ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE INHIBITORS | 1-gen-2016 | Onnis, Valentina; Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Catto, Marco; Pisani, Leonardo; Carotti, Angelo | - | - |
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