Sfoglia per Autore
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones
2016-01-01 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, A; Manfredini, S; Pacifico, S; Liekens, S; Balzarini, J.
Potent nematicidal activity of maleimide derivatives on Meloidogyne incognita
2016-01-01 Eloh, Kodjo; Demurtas, Monica; Mura, MANUEL GIACOMO; Deplano, Alessandro; Onnis, Valentina; Sasanelli, N; Maxia, Andrea; Caboni, Pierluigi
Investigation of the mechanism of FAAH inhibition of profen amide derivatives
2015-01-01 Morgillo, Cm; Deplano, Alessandro; Demurtas, Monica; Karlosson, J; Onnis, Valentina; Congiu, Cenzo; Fowler, Cj; Catalanotti, B.
Dihydroquinazoline and Triazinedione Derivatives as Prok1 and Prok2 receptor antagonists in HEK-293 transfected cells
2015-01-01 Balboni, Gianfranco; Congiu, Cenzo; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Sbai, Oualid; Rondard, Philippe; Onnis, Valentina
Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Dedeoglu, Nurcan; Supuran, Claudiu T.
Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties
2015-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Ceruso, Mariangela; Supuran, Claudiu T.
In vitro nematicidal activity of aryl hydrazones and comparative GC-MS metabolomics analysis
2015-01-01 Eloh, Kodjo; Demurtas, Monica; Deplano, Alessandro; Ngoutane Mfopa, A; Murgia, Antonio; Maxia, Andrea; Onnis, Valentina; Caboni, Pierluigi
Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor
2015-01-01 Gouveia Figueira, S; Karlsson, J; Deplano, Alessandro; Hashemian, S; Svensson, M; Fredriksson Sundbom, M; Congiu, Cenzo; Onnis, Valentina; Fowler, Cj
Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel
2015-01-01 Petrocellis, Luciano De; Moriello, Aniello Schiano; Byun, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Vázquez Romero, Ana; Garrido, Maria; Messeguer, Angel; Zhang, Fang Xiong; Zamponi, Gerald W; Deplano, Alessandro; Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Marzo, Vincenzo Di
Interaction of the N-(3-Methylpyridin-2-yl)amide derivatives of flurbiprofen and ibuprofen with FAAH: Enantiomeric selectivity and binding mode
2015-01-01 Karlsson, Jessica; Morgillo, Carmine M; Deplano, Alessandro; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Svensson, Mona; Novellino, Ettore; Congiu, Cenzo; Onnis, Valentina; Catalanotti, Bruno; Fowler, Christopher J.
Design, synthesis and pharmacological investigation on new FAAH inhibitors
2014-01-01 Onnis, Valentina; Congiu, Cenzo; Deplano, Alessandro; Demurtas, M; Cipriano, M; Fowler C., J; Morgillo C., M; Catalanotti, B.
Design, Synthesis and Evaluation of new 2-(Arylidenehydrazino)pyrrole Derivatives as Potential Antitumor Agents
2014-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Demurtas, M; Balboni, Gianfranco
A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists
2014-01-01 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Negri, L; Lattanzi, R; Balboni, Gianfranco
Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization
2014-01-01 Lattanzi, R; Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Francioso, A; Ambrosio, C; Casella, I; Costa, T; Caltabiano, G; Matsoukas M., T; Balboni, Gianfranco; Negri, L.
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones | 1-gen-2016 | Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, A; Manfredini, S; Pacifico, S; Liekens, S; Balzarini, J. | MOLECULES | - |
Potent nematicidal activity of maleimide derivatives on Meloidogyne incognita | 1-gen-2016 | Eloh, Kodjo; Demurtas, Monica; Mura, MANUEL GIACOMO; Deplano, Alessandro; Onnis, Valentina; Sasanelli, N; Maxia, Andrea; Caboni, Pierluigi | JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | - |
Investigation of the mechanism of FAAH inhibition of profen amide derivatives | 1-gen-2015 | Morgillo, Cm; Deplano, Alessandro; Demurtas, Monica; Karlosson, J; Onnis, Valentina; Congiu, Cenzo; Fowler, Cj; Catalanotti, B. | - | - |
Dihydroquinazoline and Triazinedione Derivatives as Prok1 and Prok2 receptor antagonists in HEK-293 transfected cells | 1-gen-2015 | Balboni, Gianfranco; Congiu, Cenzo; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Sbai, Oualid; Rondard, Philippe; Onnis, Valentina | - | - |
Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Dedeoglu, Nurcan; Supuran, Claudiu T. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties | 1-gen-2015 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Balboni, Gianfranco; Ceruso, Mariangela; Supuran, Claudiu T. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
In vitro nematicidal activity of aryl hydrazones and comparative GC-MS metabolomics analysis | 1-gen-2015 | Eloh, Kodjo; Demurtas, Monica; Deplano, Alessandro; Ngoutane Mfopa, A; Murgia, Antonio; Maxia, Andrea; Onnis, Valentina; Caboni, Pierluigi | JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | - |
Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor | 1-gen-2015 | Gouveia Figueira, S; Karlsson, J; Deplano, Alessandro; Hashemian, S; Svensson, M; Fredriksson Sundbom, M; Congiu, Cenzo; Onnis, Valentina; Fowler, Cj | PLOS ONE | - |
Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel | 1-gen-2015 | Petrocellis, Luciano De; Moriello, Aniello Schiano; Byun, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Vázquez Romero, Ana; Garrido, Maria; Messeguer, Angel; Zhang, Fang Xiong; Zamponi, Gerald W; Deplano, Alessandro; Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Marzo, Vincenzo Di | PHARMACOLOGICAL RESEARCH | - |
Interaction of the N-(3-Methylpyridin-2-yl)amide derivatives of flurbiprofen and ibuprofen with FAAH: Enantiomeric selectivity and binding mode | 1-gen-2015 | Karlsson, Jessica; Morgillo, Carmine M; Deplano, Alessandro; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Svensson, Mona; Novellino, Ettore; Congiu, Cenzo; Onnis, Valentina; Catalanotti, Bruno; Fowler, Christopher J. | PLOS ONE | - |
Design, synthesis and pharmacological investigation on new FAAH inhibitors | 1-gen-2014 | Onnis, Valentina; Congiu, Cenzo; Deplano, Alessandro; Demurtas, M; Cipriano, M; Fowler C., J; Morgillo C., M; Catalanotti, B. | CHEMMEDCHEM | - |
Design, Synthesis and Evaluation of new 2-(Arylidenehydrazino)pyrrole Derivatives as Potential Antitumor Agents | 1-gen-2014 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Demurtas, M; Balboni, Gianfranco | CHEMMEDCHEM | - |
A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists | 1-gen-2014 | Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Negri, L; Lattanzi, R; Balboni, Gianfranco | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization | 1-gen-2014 | Lattanzi, R; Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Francioso, A; Ambrosio, C; Casella, I; Costa, T; Caltabiano, G; Matsoukas M., T; Balboni, Gianfranco; Negri, L. | INTERNATIONAL JOURNAL OF PHARMACEUTICAL SCIENCES AND RESEARCH | - |
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