CORONA, ANGELA

CORONA, ANGELA  

DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE  

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Risultati 1 - 20 di 119 (tempo di esecuzione: 0.025 secondi).
Titolo Data di pubblicazione Autore(i) Rivista Editore
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2015 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity 1-gen-2020 Desantis, Jenny; Massari, Serena; Corona, Angela; Astolfi, Andrea; Sabatini, Stefano; Manfroni, Giuseppe; Palazzotti, Deborah; Cecchetti, Violetta; Pannecouque, Christophe; Tramontano, Enzo; Tabarrini, Oriana MOLECULES -
2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication 1-gen-2020 Corona, Angela; Onnis, Valentina; Del Vecchio, Claudia; Esposito, Francesca; Cheng, Yung-Chi; Tramontano, Enzo MOLECULES -
2-methoxynaphthalen thiazole derivate : a new HIV-1 RT Ribonuclease H/DNA polymerase dual inhibitor active on viral replication 1-gen-2014 Corona, Angela; Meleddu, R.; Esposito, E.; Distinto, S.; Bianco, G.; Maccioni, E.; Tramontano, E. . - -
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function 1-gen-2011 Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias - -
5-arylaminouracil derivatives as potential dual-action agents 1-gen-2015 Matyugina, Es; Novikov, Ms; Babkov, Da; Valuev Elliston, Vt; Vanpouille, C; Zicari, S; Corona, Angela; Tramontano, Enzo; Margolis, Lb; Khandazhinskaya, Al; Kochetkov, Sn ACTA NATURAE -
A combined cell based and site directed mutagenesis approach defines highly conserved residues involved in the selective inhibition of the HIV-1 ribonuclease H function by diketoacid derivatives 1-gen-2014 Corona, Angela; Cosconati, S; Tierry, S; Pescatore, L; Di Leva F., S; Subra, F.; Delelis, O; Esposito, Francesca; Costi, R; Novellino, E; Di Santo, R; Tramontano, E. - -
A Luciferase Reporter Gene Assay to Measure Ebola Virus Viral Protein 35–Associated Inhibition of Double-Stranded RNA–Stimulated, Retinoic Acid–Inducible Gene 1–Mediated Induction of Interferon β 1-gen-2015 Cannas, V; Daino, Gl; Corona, Angela; Esposito, Francesca; Tramontano, Enzo THE JOURNAL OF INFECTIOUS DISEASES -
A new vinyl selenone-based domino approach to spirocyclopropyl oxindoles endowed with anti-HIV RT activity 1-gen-2016 Palomba, M.; Rossi, L.; Sancineto, L.; Tramontano, E.; Corona, A.; Bagnoli, L.; Santi, C.; Pannecouque, C.; Tabarrini, O.; Marini, F ORGANIC & BIOMOLECULAR CHEMISTRY -
Active site and allosteric inhibitors of the ribonuclease H activity of HIV reverse transcriptase 1-gen-2013 Corona, Angela; Masaoka, T; Tocco, Graziella; Tramontano, Enzo; Le Grice, Sfj FUTURE MEDICINAL CHEMISTRY -
Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and RNase H activities effective also on the RNase H activity of non-nucleoside resistant reverse transcriptases 1-gen-2011 Esposito, Francesca; Kharlamova, T; Distinto, Simona; Zinzula, Luca; Cheng Y., C; Dutschman, G; Floris, G; Markt, P; Corona, Angela; Tramontano, Enzo THE FEBS JOURNAL -
An efficient route to novel uracil-based drug-like molecules 1-gen-2015 Babkov, Da; Chizhov, Ao; Khandazhinskaya, Al; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; SELEY RADTKE, Kl; Novikov, Ms SYNTHESIS -
Antiretroviral activity of metal-chelating HIV-1 integrase inhibitors 1-gen-2014 Carcelli, M; Rogolino, D; Sechi, M; Rispoli, G; Fisicaro, E; Compari, C; Grandi, Nicole; Corona, Angela; Tramontano, Enzo; Pannecouque, C; Naesens, L. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Antityrosinase activity of Euphorbia characias extracts 1-gen-2015 Pintus, Francesca; Spano', Delia; Corona, Angela; Medda, Rosaria PEERJ -
Antiviral Agents Against Ebola Virus Infection: Repositioning Old Drugs and Finding Novel Small Molecules 1-gen-2018 Fanunza, Elisa; Frau, Aldo; Corona, Angela; Tramontano, Enzo ANNUAL REPORTS IN MEDICINAL CHEMISTRY -
Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptase 1-gen-2014 Costi, R; Métifiot, M; Chung, S; CUZZUCOLI CRUCITTI, G; Maddali, K; Pescatori, L; Messore, A; Madia, Vn; Pupo, G; Scipione, L; Tortorella, S; DI LEVA, Fs; Cosconati, S; Marinelli, L; Novellino, E; LE GRICE, Sf; Corona, Angela; Pommier, Y; Marchand, C; DI SANTO, R. JOURNAL OF MEDICINAL CHEMISTRY -
Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitors 1-gen-2016 Schneider, Anna; Corona, Angela; Spöring, Imke; Jordan, Mareike; Buchholz, Bernd; Maccioni, Elias; Di Santo, Roberto; Bodem, Jochen; Tramontano, Enzo; Wöhrl, Birgitta M. NUCLEIC ACIDS RESEARCH -
Biological activities of aerial parts extracts of Euphorbia characias 1-gen-2016 Pisano, MARIA BARBARA; Cosentino, Sofia; Viale, Silvia; Spano', Delia; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Montoro, P; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca BIOMED RESEARCH INTERNATIONAL -
Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination 1-gen-2023 Stefanelli, Irina; Corona, Angela; Cerchia, Carmen; Cassese, Emilia; Improta, Salvatore; Costanzi, Elisa; Pelliccia, Sveva; Morasso, Stefano; Esposito, Francesca; Paulis, Annalaura; Scognamiglio, Sante; Di Leva, Francesco Saverio; Storici, Paola; Brindisi, Margherita; Tramontano, Enzo; Cannalire, Rolando; Summa, Vincenzo EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Can the ever-promising target HIV reverse transcriptase-associated RNase H become a success story for drug development? 1-gen-2014 Corona, Angela; Esposito, Francesca; Tramontano, Enzo FUTURE VIROLOGY -