TRAMONTANO, ENZO

TRAMONTANO, ENZO  

DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE  

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Titolo Data di pubblicazione Autore(i) Rivista Editore
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity 1-gen-2020 Desantis, Jenny; Massari, Serena; Corona, Angela; Astolfi, Andrea; Sabatini, Stefano; Manfroni, Giuseppe; Palazzotti, Deborah; Cecchetti, Violetta; Pannecouque, Christophe; Tramontano, Enzo; Tabarrini, Oriana MOLECULES -
2,6-Bis (3,4,5 - trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays 1-gen-2004 Costi, R; DI SANTO, R; Artico, M; Massa, S; Ragno, R; Loddo, Roberta; LA COLLA, M; Tramontano, Enzo; LA COLLA, P; Pani, Alessandra BIOORGANIC & MEDICINAL CHEMISTRY -
2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication 1-gen-2020 Corona, Angela; Onnis, Valentina; Del Vecchio, Claudia; Esposito, Francesca; Cheng, Yung-Chi; Tramontano, Enzo MOLECULES -
3,4-Dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs): a new class of specific inhibitors of human immunodeficiency virus type 1 1-gen-1993 Artico, M; Massa, S; Mai, A; Marongiu, Me; Piras, G; Tramontano, Enzo; LA COLLA, P. ANTIVIRAL CHEMISTRY & CHEMOTHERAPY -
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function 1-gen-2011 Meleddu, Rita; Corona, Angela; Distinto, Simona; Esposito, Francesca; Sanna, M. L.; Cardia, C.; Tramontano, Enzo; Maccioni, Elias - -
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2015 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
5-alkyl-2-(alkylthio)-6-(2,6-dihalophenyl-methyl)-3,4-dihydropyrimidin-4(3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives 1-gen-1999 Mai, A; Artico, M; Sbardella, G; Massa, S; Novellino, E; Greco, G; Loi, Ag; Tramontano, Enzo; Marongiu, Me; LA COLLA, P. JOURNAL OF MEDICINAL CHEMISTRY -
5-arylaminouracil derivatives as potential dual-action agents 1-gen-2015 Matyugina, Es; Novikov, Ms; Babkov, Da; Valuev Elliston, Vt; Vanpouille, C; Zicari, S; Corona, Angela; Tramontano, Enzo; Margolis, Lb; Khandazhinskaya, Al; Kochetkov, Sn ACTA NATURAE -
6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach 1-gen-2013 Costi, R; Métifiot, M; Esposito, Francesca; Cuzzucoli Crucitti, G; Pescatori, L; Messore, A; Scipione, L; Tortorella, S; Zinzula, Luca; Novellino, E; Pommier, Y; Tramontano, Enzo; Marchand, C; Di Santo, R. JOURNAL OF MEDICINAL CHEMISTRY -
6-[1-(4-fluorophenyl)methyl-1H-pyrrol-2-y1)]-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro 1-gen-2005 Tramontano, Enzo; Esposito, Francesca; Badas, R; DI SANTO, R; Costi, R; La, Colla ANTIVIRAL RESEARCH -
6-Aryl-2,4-dioxo-5-hexenoic acids, novel integrase inhibitors active against HIV-1 multiplication in cell-based assays 1-gen-2004 Costi, R; DI SANTO, R; Artico, M; Roux, A; Ragno, R; Massa, S; Tramontano, Enzo; LA COLLA, M; Loddo, Roberta; Marongiu, Me; Pani, Alessandra; LA COLLA, P. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS -
A review on the in vitro activity of phosphorothioate oligonucleotides against human immunodeficiency viruses 1-gen-1993 De Falco, S; Iacomino, G; Galderisi, U; Cipollaro, M; De Rienzo, A; Galano G., Cascino A; Loi, Ag; Spiga, Mg; Basile, T; Musu, D; DE MONTIS, Antonella; Tramontano, Enzo; Marongiu, Me; La Colla, P. MINERVA BIOTECNOLOGICA -
A single conservative amino acid substitution in the reverse transcriptase of human immunodeficiency virus type 1 confers resistance to (+)-(5S)-4,5,6,7-tetrahydro-5-methyl-6-(3-methyl-2butenyl)imidazo[4,5,1,jk][1,4] benzodiazepin-2(1H)-thione (TIBO R82150) 1-gen-1993 Mellors, J; Im, Gj; Tramontano, Enzo; Winkler, Sr; Medina, Dj; Dutschman, Ge; Bazmi, Hz; Piras, G; Gonzales, Cj; Cheng, Y. C. MOLECULAR PHARMACOLOGY -
Active site and allosteric inhibitors of the ribonuclease H activity of HIV reverse transcriptase 1-gen-2013 Corona, Angela; Masaoka, T; Tocco, Graziella; Tramontano, Enzo; Le Grice, Sfj FUTURE MEDICINAL CHEMISTRY -
Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase (RT) -associated DNA polymerase and Ribonuclease H (RNase H) activities effective also on the RNase H activity of non-nucleoside resistant RTs 1-gen-2010 Esposito, F.; Kharlamova, T.; Distinto, S.; Zinzula, L.; Cheng, Y-C.; Dutschman, G.; Floris, G.; Markt, P.; Tramontano, E. - -
Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and Ribonuclease H activities effective also on non-nucleoside resistant RTs 1-gen-2010 Esposito, F; Kharlamova, T.; Distinto, S.; Zinzula, L.; Floris, G.; Sanna Randaccio, L.; Deutschman, G.; Cheng, Y-C.; Tramontano, E. - -
Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and RNase H activities effective also on the RNase H activity of non-nucleoside resistant reverse transcriptases 1-gen-2011 Esposito, Francesca; Kharlamova, T; Distinto, Simona; Zinzula, Luca; Cheng Y., C; Dutschman, G; Floris, G; Markt, P; Corona, Angela; Tramontano, Enzo THE FEBS JOURNAL -
ANALYSIS OF 98 HERV-K(HML-2) CONTAINING PROVIRUSES IDENTIFIED IN THE HUMAN GENOME ASSEMBLY GRCH37/HG19 BY RETROTECTOR AND THEIR GENOMIC CONTEXT 1-gen-2014 Cadeddu, Marta; Grandi, Nicole; L., Vargiu; P., Rodriguez Tomè; J., Blomberg; Tramontano, Enzo - -
Anti-AIDS agents, 6. Salaspermic acid, an anti-HIV principle from tripterygium wilfordii, and the structure-activity correlation with its relared compounds 1-gen-1992 Chen, K; Shi, Q; Kashiwada, Y; ZHANG D., C; HU C., Q; JIN J., Q; Nozaki, H; Tramontano, Enzo; CHENG Y., C; Mcphail, Dr; Mcphail, At; Lee, K. H. JOURNAL OF NATURAL PRODUCTS -
Anti-HIV-1 activity of compounds isolated from Hypericum hircinum. 1-gen-2012 Sanna, Cinzia; Esposito, Francesca; Del Vecchio, C; Mandas, D; Ballero, Mauro; Bianco, A; Parolin, C; Tramontano, Enzo - -