TRAMONTANO, ENZO
TRAMONTANO, ENZO
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
Rational structure-based design and optimization of next-generation biphenyl-piperidine-triazine derivatives as potent non-nucleoside reverse transcriptase inhibitors
2026-01-01 Zhang, Kun; Zhao, Li-Min; Xing, Tianhao; Bu, Yueyue; Wang, Qingyun; Pannecouque, Christophe; De Clercq, Erik; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Wang, Shuai; Chen, Fen-Er
Characterization of SARS-CoV-2 nucleocapsid protein oligomers
2025-01-01 Farci, Domenica; Graça, André T; Hall, Michael; Haniewicz, Patrycja; Kereïche, Sami; Faull, Peter; Kirkpatrick, Joanna; Tramontano, Enzo; Schröder, Wolfgang P; Piano, Dario
Cys44 of SARS-CoV-2 3CLpro affects its catalytic activity
2025-01-01 Iacobucci, I.; Cipollone, I.; Cozzolino, F.; Iaconis, D.; Talarico, C.; Coppola, G.; Morasso, S.; Costanzi, E.; Malune, Paolo; Storici, P.; Tramontano, E.; Esposito, Francesca; Monti, M.
Design, and synthesis of 2,4-thiazolidinedione substituted 1–3-5-triazine derivatives as anti-HIV agent via inhibition of reverse transcriptase along with anti-SARS CoV-2, antibacterial and antibiofilm activity
2025-01-01 Singh, Saumya; Srivastava, Kumar Saurabh; Gahtori, Prashant; Anand, Ananya Anurag; Samanta, Sintu Kumar; Kumawat, Mukesh Kumar; Bhat, Hans Raj; Corona, Angela; Tramontano, Enzo; Mitra, Debashis; Singh, Udaya Pratap
Design, Synthesis and Biological Evaluation of 3-Hydrazonoindolin-2-one Derivatives as Novel HIV-1 RNase H Inhibitors
2025-01-01 Zhang, Yiying; Wang, Rao; Bu, Yueyue; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Pannecouque, Christophe; De Clercq, Erik; Wang, Shuai; Meng, Ge; Chen, Fen-Er
Dual-Site Inhibition of SARS-CoV2 RNA-Dependent RNA Polymerase by Small Molecules Able to Block Viral Replication Identified through a Computer-Aided Drug Discovery Approach
2025-01-01 Malune, Paolo; Iaconis, Daniela; Manelfi, Candida; Giunta, Stefano; Emmolo, Roberta; Lunghini, Filippo; Paulis, Annalaura; Talarico, Carmine; Corona, Angela; Rosario Beccari, Andrea; Tramontano, Enzo; Esposito, Francesca
HERV Modulation in Colorectal Carcinoma Patients: A Snapshot of Endogenous Retroviral Transcriptome
2025-01-01 Grandi, Nicole; Liu, Ching‐hsuan; Chabukswar, Saili; Carta, Daniele; Yen, Yun; Lin, Liang‐tzung; Tramontano, Enzo
Identification of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Inhibitors Based on 2-Hydroxy-1,4-naphthoquinone Mannich Bases
2025-01-01 Tu, Nhat Quang; Richetta, Clémence; Putzu, Federica; Delelis, Olivier; Ahmed, Khursheed; Masand, Vijay H.; Schobert, Rainer; Tramontano, Enzo; Corona, Angela; Biersack, Bernhard
Impact of Pre-lockdown Hyper-energy on Mood and Rhythm Dysregulation in Older Adults During the COVID-19 Pandemic
2025-01-01 Primavera, Diego; Kalcev, Goce; Bert, Fabrizio; Cantone, Elisa; Perra, Alessandra; Tusconi, Massimo; Pinna, Samantha; Orrù, Germano; Scano, Alessandra; Tramontano, Enzo; Barbov, Ivan; Nonnis, Marcello; Nardi, Antonio Egidio; Cossu, Giulia; Sancassiani, Federica; Carta, Mauro Giovanni
Meeting report: Seventh summer school on innovative approaches for identification of antiviral agents (IAAASS)
2025-01-01 Corona, Angela; Cagno, Valeria; Grandi, Nicole; Fanunza, Elisa; Esposito, Francesca; Seley-Radtke, Kathie L.; Tramontano, Enzo
N -alkyl and N-benzyl indoles are anti-SARS-CoV-2 agents and nsp13 inhibitors
2025-01-01 Albano, Aurora; Emmolo, Roberta; De Santis, Riccardo; Patacchini, Elisa; Madia, Valentina Noemi; Maloccu, Stefania; Ialongo, Davide; Ruggieri, Giuseppe; Arpacioglu, Merve; Scipione, Luigi; Saccoliti, Francesco; Amatore, Donatella; Grilli, Giorgia; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta
Resilience to depression and unchanged quality of life in Sardinian old adults during COVID-19 lockdown
2025-01-01 Cossu, G.; Atzeni, M.; Cantone, E.; Forte, V.; Tusconi, M.; Kalcev, G.; Maleci, A.; Montisci, R.; Ferreli, C.; Atzori, L.; Primavera, D.; Dursun, S. M.; Bert, F.; Tramontano, E.; Carta, M. G.
Structure-Based Discovery of Novel Diarylpyrimidines as Potent and Selective Non-Nucleoside Reverse Transcriptase Inhibitors: From CH(CN)-Biphenyl-Diarylpyrimidines to C=NNH2-Biphenyl-Diarylpyrimidines
2025-01-01 Chen, Xiao-Mei; Pannecouque, Christophe; De Clercq, Erik; Lian, Yu-Xuan; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Wang, Shuai; Chen, Fen-Er
Structure−Activity Relationships of New 1‐Aryl‐1H‐Indole Derivatives as SARS‐CoV‐2 Nsp13 Inhibitors
2025-01-01 Madia, Valentina Noemi; Emmolo, Roberta; Patacchini, Elisa; Amatore, Donatella; Maloccu, Stefania; Ialongo, Davide; Albano, Aurora; Ruggieri, Giuseppe; Cara, Emanuele; Zarbo, Laura; Messore, Antonella; De Santis, Riccardo; Amoroso, Alessandra; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta
Suicidality and/or Death-Related Thoughts in Health Workers After Pandemics: The Role of DYMERS
2025-01-01 Urban, Antonio; Cantone, Elisa; Forte, Viviana; Atzeni, Michela; Lorrai, Stefano; Carzedda, Mauro; Finco, Gabriele; Gonzalez, Cesar Ivan Aviles; Machado, Sergio; Montisci, Roberta; Tramontano, Enzo; Marra, Orsola; Muscas, Francesco; Bert, Fabrizio; Cossu, Giulia; Carta, Mauro Giovanni
The efficiency of high-throughput screening (HTS) and in-silico data analysis during medical emergencies: Identification of effective antiviral 3CLpro inhibitors
2025-01-01 Zian, D.; Iaconis, D.; Nenci, S.; Crusco, A.; Tawde, S.; Sodano, M.; Vitalone, R.; Raje, A.; Palamini, M.; Carettoni, D.; Molteni, A.; Manelfi, C.; Tazzari, V.; Beccari, A. R.; Malune, P.; Maloccu, S.; Paulis, Annalaura; Corona, Angela; Nieddu, Salvatore; Coletti, S.; Scarabottolo, L.; Tramontano, Enzo; Esposito, Francesca; Catalani, M.
The Use of Heart Rate Variability-Biofeedback (HRV-BF) as an Adjunctive Intervention in Chronic Fatigue Syndrome (CSF/ME) in Long COVID: Results of a Phase II Controlled Feasibility Trial
2025-01-01 Cossu, Giulia; Kalcev, Goce; Primavera, Diego; Lorrai, Stefano; Perra, Alessandra; Galetti, Alessia; Demontis, Roberto; Tramontano, Enzo; Bert, Fabrizio; Montisci, Roberta; Maleci, Alberto; Castilla, Pedro José Fragoso; Jaramillo, Shellsyn Giraldo; Kurotschka, Peter K.; Rocha, Nuno Barbosa; Carta, Mauro Giovanni
Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2
2025-01-01 Kuzikov, Maria; Morasso, Stefano; Reinshagen, Jeanette; Wolf, Markus; Monaco, Vittoria; Cozzolino, Flora; Golič Grdadolnik, Simona; Šket, Primož; Plavec, Janez; Iaconis, Daniela; Summa, Vincenzo; Corona, Angela; Paulis, Annalaura; Esposito, Francesca; Tramontano, Enzo; Monti, Maria; Beccari, Andrea R.; Manelfi, Candida; Windshügel, Björn; Gribbon, Philip; Storici, Paola; Zaliani, Andrea
Tiazolidinoni come agenti antivirali
2025-01-01 Distinto, Simona; Corona, Angela; Sanna, Erica; Tramontano, Enzo; Maccioni, Elias; Scognamiglio, Sante; Onali, Alessia; Cottiglia, Filippo; Meleddu, Rita; Secci, Daniela; Maloccu, Stefania
Unveiling SARS-CoV-2's heart: role, structure and inhibition of SARS-CoV-2 RNA-dependent RNA polymerase
2025-01-01 Malune, P.; Esposito, Francesca; Tramontano, E.
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Rational structure-based design and optimization of next-generation biphenyl-piperidine-triazine derivatives as potent non-nucleoside reverse transcriptase inhibitors | 1-gen-2026 | Zhang, Kun; Zhao, Li-Min; Xing, Tianhao; Bu, Yueyue; Wang, Qingyun; Pannecouque, Christophe; De Clercq, Erik; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Wang, Shuai; Chen, Fen-Er | CHINESE CHEMICAL LETTERS | - |
| Characterization of SARS-CoV-2 nucleocapsid protein oligomers | 1-gen-2025 | Farci, Domenica; Graça, André T; Hall, Michael; Haniewicz, Patrycja; Kereïche, Sami; Faull, Peter; Kirkpatrick, Joanna; Tramontano, Enzo; Schröder, Wolfgang P; Piano, Dario | JOURNAL OF STRUCTURAL BIOLOGY | - |
| Cys44 of SARS-CoV-2 3CLpro affects its catalytic activity | 1-gen-2025 | Iacobucci, I.; Cipollone, I.; Cozzolino, F.; Iaconis, D.; Talarico, C.; Coppola, G.; Morasso, S.; Costanzi, E.; Malune, Paolo; Storici, P.; Tramontano, E.; Esposito, Francesca; Monti, M. | INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES | - |
| Design, and synthesis of 2,4-thiazolidinedione substituted 1–3-5-triazine derivatives as anti-HIV agent via inhibition of reverse transcriptase along with anti-SARS CoV-2, antibacterial and antibiofilm activity | 1-gen-2025 | Singh, Saumya; Srivastava, Kumar Saurabh; Gahtori, Prashant; Anand, Ananya Anurag; Samanta, Sintu Kumar; Kumawat, Mukesh Kumar; Bhat, Hans Raj; Corona, Angela; Tramontano, Enzo; Mitra, Debashis; Singh, Udaya Pratap | BIOORGANIC CHEMISTRY | - |
| Design, Synthesis and Biological Evaluation of 3-Hydrazonoindolin-2-one Derivatives as Novel HIV-1 RNase H Inhibitors | 1-gen-2025 | Zhang, Yiying; Wang, Rao; Bu, Yueyue; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Pannecouque, Christophe; De Clercq, Erik; Wang, Shuai; Meng, Ge; Chen, Fen-Er | MOLECULES | - |
| Dual-Site Inhibition of SARS-CoV2 RNA-Dependent RNA Polymerase by Small Molecules Able to Block Viral Replication Identified through a Computer-Aided Drug Discovery Approach | 1-gen-2025 | Malune, Paolo; Iaconis, Daniela; Manelfi, Candida; Giunta, Stefano; Emmolo, Roberta; Lunghini, Filippo; Paulis, Annalaura; Talarico, Carmine; Corona, Angela; Rosario Beccari, Andrea; Tramontano, Enzo; Esposito, Francesca | ACS INFECTIOUS DISEASES | - |
| HERV Modulation in Colorectal Carcinoma Patients: A Snapshot of Endogenous Retroviral Transcriptome | 1-gen-2025 | Grandi, Nicole; Liu, Ching‐hsuan; Chabukswar, Saili; Carta, Daniele; Yen, Yun; Lin, Liang‐tzung; Tramontano, Enzo | JOURNAL OF MEDICAL VIROLOGY | - |
| Identification of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Inhibitors Based on 2-Hydroxy-1,4-naphthoquinone Mannich Bases | 1-gen-2025 | Tu, Nhat Quang; Richetta, Clémence; Putzu, Federica; Delelis, Olivier; Ahmed, Khursheed; Masand, Vijay H.; Schobert, Rainer; Tramontano, Enzo; Corona, Angela; Biersack, Bernhard | MOLECULES | - |
| Impact of Pre-lockdown Hyper-energy on Mood and Rhythm Dysregulation in Older Adults During the COVID-19 Pandemic | 1-gen-2025 | Primavera, Diego; Kalcev, Goce; Bert, Fabrizio; Cantone, Elisa; Perra, Alessandra; Tusconi, Massimo; Pinna, Samantha; Orrù, Germano; Scano, Alessandra; Tramontano, Enzo; Barbov, Ivan; Nonnis, Marcello; Nardi, Antonio Egidio; Cossu, Giulia; Sancassiani, Federica; Carta, Mauro Giovanni | CLINICAL PRACTICE AND EPIDEMIOLOGY IN MENTAL HEALTH | - |
| Meeting report: Seventh summer school on innovative approaches for identification of antiviral agents (IAAASS) | 1-gen-2025 | Corona, Angela; Cagno, Valeria; Grandi, Nicole; Fanunza, Elisa; Esposito, Francesca; Seley-Radtke, Kathie L.; Tramontano, Enzo | ANTIVIRAL RESEARCH | - |
| N -alkyl and N-benzyl indoles are anti-SARS-CoV-2 agents and nsp13 inhibitors | 1-gen-2025 | Albano, Aurora; Emmolo, Roberta; De Santis, Riccardo; Patacchini, Elisa; Madia, Valentina Noemi; Maloccu, Stefania; Ialongo, Davide; Ruggieri, Giuseppe; Arpacioglu, Merve; Scipione, Luigi; Saccoliti, Francesco; Amatore, Donatella; Grilli, Giorgia; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Resilience to depression and unchanged quality of life in Sardinian old adults during COVID-19 lockdown | 1-gen-2025 | Cossu, G.; Atzeni, M.; Cantone, E.; Forte, V.; Tusconi, M.; Kalcev, G.; Maleci, A.; Montisci, R.; Ferreli, C.; Atzori, L.; Primavera, D.; Dursun, S. M.; Bert, F.; Tramontano, E.; Carta, M. G. | FRONTIERS IN PSYCHIATRY | - |
| Structure-Based Discovery of Novel Diarylpyrimidines as Potent and Selective Non-Nucleoside Reverse Transcriptase Inhibitors: From CH(CN)-Biphenyl-Diarylpyrimidines to C=NNH2-Biphenyl-Diarylpyrimidines | 1-gen-2025 | Chen, Xiao-Mei; Pannecouque, Christophe; De Clercq, Erik; Lian, Yu-Xuan; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Wang, Shuai; Chen, Fen-Er | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Structure−Activity Relationships of New 1‐Aryl‐1H‐Indole Derivatives as SARS‐CoV‐2 Nsp13 Inhibitors | 1-gen-2025 | Madia, Valentina Noemi; Emmolo, Roberta; Patacchini, Elisa; Amatore, Donatella; Maloccu, Stefania; Ialongo, Davide; Albano, Aurora; Ruggieri, Giuseppe; Cara, Emanuele; Zarbo, Laura; Messore, Antonella; De Santis, Riccardo; Amoroso, Alessandra; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta | CHEMMEDCHEM | - |
| Suicidality and/or Death-Related Thoughts in Health Workers After Pandemics: The Role of DYMERS | 1-gen-2025 | Urban, Antonio; Cantone, Elisa; Forte, Viviana; Atzeni, Michela; Lorrai, Stefano; Carzedda, Mauro; Finco, Gabriele; Gonzalez, Cesar Ivan Aviles; Machado, Sergio; Montisci, Roberta; Tramontano, Enzo; Marra, Orsola; Muscas, Francesco; Bert, Fabrizio; Cossu, Giulia; Carta, Mauro Giovanni | JOURNAL OF CLINICAL MEDICINE | - |
| The efficiency of high-throughput screening (HTS) and in-silico data analysis during medical emergencies: Identification of effective antiviral 3CLpro inhibitors | 1-gen-2025 | Zian, D.; Iaconis, D.; Nenci, S.; Crusco, A.; Tawde, S.; Sodano, M.; Vitalone, R.; Raje, A.; Palamini, M.; Carettoni, D.; Molteni, A.; Manelfi, C.; Tazzari, V.; Beccari, A. R.; Malune, P.; Maloccu, S.; Paulis, Annalaura; Corona, Angela; Nieddu, Salvatore; Coletti, S.; Scarabottolo, L.; Tramontano, Enzo; Esposito, Francesca; Catalani, M. | ANTIVIRAL RESEARCH | - |
| The Use of Heart Rate Variability-Biofeedback (HRV-BF) as an Adjunctive Intervention in Chronic Fatigue Syndrome (CSF/ME) in Long COVID: Results of a Phase II Controlled Feasibility Trial | 1-gen-2025 | Cossu, Giulia; Kalcev, Goce; Primavera, Diego; Lorrai, Stefano; Perra, Alessandra; Galetti, Alessia; Demontis, Roberto; Tramontano, Enzo; Bert, Fabrizio; Montisci, Roberta; Maleci, Alberto; Castilla, Pedro José Fragoso; Jaramillo, Shellsyn Giraldo; Kurotschka, Peter K.; Rocha, Nuno Barbosa; Carta, Mauro Giovanni | JOURNAL OF CLINICAL MEDICINE | - |
| Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2 | 1-gen-2025 | Kuzikov, Maria; Morasso, Stefano; Reinshagen, Jeanette; Wolf, Markus; Monaco, Vittoria; Cozzolino, Flora; Golič Grdadolnik, Simona; Šket, Primož; Plavec, Janez; Iaconis, Daniela; Summa, Vincenzo; Corona, Angela; Paulis, Annalaura; Esposito, Francesca; Tramontano, Enzo; Monti, Maria; Beccari, Andrea R.; Manelfi, Candida; Windshügel, Björn; Gribbon, Philip; Storici, Paola; Zaliani, Andrea | ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE | - |
| Tiazolidinoni come agenti antivirali | 1-gen-2025 | Distinto, Simona; Corona, Angela; Sanna, Erica; Tramontano, Enzo; Maccioni, Elias; Scognamiglio, Sante; Onali, Alessia; Cottiglia, Filippo; Meleddu, Rita; Secci, Daniela; Maloccu, Stefania | - | - |
| Unveiling SARS-CoV-2's heart: role, structure and inhibition of SARS-CoV-2 RNA-dependent RNA polymerase | 1-gen-2025 | Malune, P.; Esposito, Francesca; Tramontano, E. | ANTIVIRAL RESEARCH | - |