DEPLANO, ALESSANDRO

DEPLANO, ALESSANDRO  

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Risultati 1 - 20 di 33 (tempo di esecuzione: 0.039 secondi).
Titolo Data di pubblicazione Autore(i) Rivista Editore
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors 1-gen-2020 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Piras, Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina BIOORGANIC CHEMISTRY -
Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors 1-gen-2019 Deplano, Alessandro; Cipriano, Mariateresa; Moraca, Federica; Novellino, Ettore; Catalanotti, Bruno; Fowler, Christopher J.; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor 1-gen-2015 Gouveia Figueira, S; Karlsson, J; Deplano, Alessandro; Hashemian, S; Svensson, M; Fredriksson Sundbom, M; Congiu, Cenzo; Onnis, Valentina; Fowler, Cj PLOS ONE -
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions 1-gen-2017 Corona, Angela; Onnis, Valentina; Deplano, Alessandro; Bianco, Giulia; Demurtas, Monica; Distinto, Simona; Cheng, Yung Chi; Alcaro, Stefano; Esposito, Francesca; Tramontano, Enzo PATHOGENS AND DISEASE -
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones 1-gen-2016 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, A; Manfredini, S; Pacifico, S; Liekens, S; Balzarini, J. MOLECULES -
Design, Synthesis and Evaluation of new 2-(Arylidenehydrazino)pyrrole Derivatives as Potential Antitumor Agents 1-gen-2014 Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Demurtas, M; Balboni, Gianfranco CHEMMEDCHEM -
Design, synthesis and in vitro and in vivo biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents 1-gen-2021 Deplano, Alessandro; Karlsson, Jessica; Moraca, Federica; Svensson, Mona; Cristiano, Claudia; Morgillo, Carmine Marco; Fowler, Christopher J.; Russo, Roberto; Catalanotti, Bruno; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
DESIGN, SYNTHESIS AND PHARMACOLOGICAL INVESTIGATION OF NEW DNA METHYLTRANSFERASE INHIBITORS 1-gen-2016 Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Arimondo, Paola B.; Masson, Veronique; Onnis, Valentina - -
Design, synthesis and pharmacological investigation on new FAAH inhibitors 1-gen-2014 Onnis, Valentina; Congiu, Cenzo; Deplano, Alessandro; Demurtas, M; Cipriano, M; Fowler C., J; Morgillo C., M; Catalanotti, B. CHEMMEDCHEM -
Design, synthesis and SAR of small molecules acting on pain pathways 24-mar-2016 - - Università degli Studi di Cagliari
Development and Validation of Molecular Overlays Derived from Three-Dimensional Hydrophobic Similarity with PharmScreen 1-gen-2018 Vázquez, J.; Deplano, A.; Herrero, A.; Ginex, T.; Gibert, E.; Rabal, O.; Oyarzabal, J.; Herrero, E.; Luque, F. J. JOURNAL OF CHEMICAL INFORMATION AND MODELING -
Dihydroquinazoline and Triazinedione Derivatives as Prok1 and Prok2 receptor antagonists in HEK-293 transfected cells 1-gen-2015 Balboni, Gianfranco; Congiu, Cenzo; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Sbai, Oualid; Rondard, Philippe; Onnis, Valentina - -
DIHYDROQUINAZOLINE BENZYLAMIDES AS ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE INHIBITORS 1-gen-2016 Onnis, Valentina; Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Catto, Marco; Pisani, Leonardo; Carotti, Angelo - -
Discovery of a novel class of profen derivatives as FAAH inhibitors: MD and QM/MM studies of the binding mode and 3D SAR 1-gen-2016 Morgillo, Cm; Deplano, Alessandro; Karlsson, J; Cipriano, M; Björklund, E; Fowler, Cj; Onnis, Valentina; Luque, Fj; Catalanotti, B. - -
Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen 1-gen-2020 Deplano, Alessandro; Karlsson, Jessica; Svensson, Mona; Moraca, Federica; Catalanotti, Bruno; Fowler, Christopher J.; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen 1-gen-2020 Deplano, Alessandro; Karlsson, Jessica; Fowler, Christopher J.; Onnis, Valentina BIOORGANIC CHEMISTRY -
Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization 1-gen-2014 Lattanzi, R; Congiu, Cenzo; Onnis, Valentina; Deplano, Alessandro; Salvadori, S; Marconi, V; Maftei, D; Francioso, A; Ambrosio, C; Casella, I; Costa, T; Caltabiano, G; Matsoukas M., T; Balboni, Gianfranco; Negri, L. INTERNATIONAL JOURNAL OF PHARMACEUTICAL SCIENCES AND RESEARCH -
Homology modeling of a Class A GPCR in the inactive conformation: A quantitative analysis of the correlation between model/template sequence identity and model accuracy 1-gen-2016 Costanzi, Stefano; Skorski, Matthew; Deplano, Alessandro; Habermehl, Brett; Mendoza, Mary; Wang, Keyun; Biederman, Michelle; Dawson, Jessica; Gaoa, Jia JOURNAL OF MOLECULAR GRAPHICS & MODELLING -
Hydrophobic similarity between molecules: Application to three-dimensional molecular overlays with PharmScreen 1-gen-2018 Vazquez, Javier; Deplano, Alessandro; Herrero, Albert; Gibert, Enric; Ginex, Tiziana; Rabal, Obdulia; Oyarzabal, Julen; Herrero, Enric; Luque, F Javier - American Chemical Society
In vitro nematicidal activity of aryl hydrazones and comparative GC-MS metabolomics analysis 1-gen-2015 Eloh, Kodjo; Demurtas, Monica; Deplano, Alessandro; Ngoutane Mfopa, A; Murgia, Antonio; Maxia, Andrea; Onnis, Valentina; Caboni, Pierluigi JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -