DEPLANO, ALESSANDRO

DEPLANO, ALESSANDRO  

Mostra records
Risultati 1 - 20 di 33 (tempo di esecuzione: 0.027 secondi).
Titolo Data di pubblicazione Autore(i) Rivista Editore
Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity 1-gen-2023 Moi, Davide; Deplano, Alessandro; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina MOLECULES -
Molecular Basis for Non-Covalent, Non-Competitive FAAH Inhibition 1-gen-2022 Morgillo, Carmine Marco; Lupia, Antonio; Deplano, Alessandro; Pirone, Luciano; Fiorillo, Bianca; Pedone, Emilia; Luque, F. Javier; Onnis, Valentina; Moraca, Federica; Catalanotti, Bruno INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES -
Design, synthesis and in vitro and in vivo biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents 1-gen-2021 Deplano, Alessandro; Karlsson, Jessica; Moraca, Federica; Svensson, Mona; Cristiano, Claudia; Morgillo, Carmine Marco; Fowler, Christopher J.; Russo, Roberto; Catalanotti, Bruno; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors 1-gen-2020 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Piras, Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina BIOORGANIC CHEMISTRY -
Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen 1-gen-2020 Deplano, Alessandro; Karlsson, Jessica; Svensson, Mona; Moraca, Federica; Catalanotti, Bruno; Fowler, Christopher J.; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors 1-gen-2020 Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen 1-gen-2020 Deplano, Alessandro; Karlsson, Jessica; Fowler, Christopher J.; Onnis, Valentina BIOORGANIC CHEMISTRY -
Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors 1-gen-2019 Deplano, Alessandro; Cipriano, Mariateresa; Moraca, Federica; Novellino, Ettore; Catalanotti, Bruno; Fowler, Christopher J.; Onnis, Valentina JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation 1-gen-2019 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors 1-gen-2019 Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gianfranco; Onnis, Valentina; Potter, Barry V. L. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Development and Validation of Molecular Overlays Derived from Three-Dimensional Hydrophobic Similarity with PharmScreen 1-gen-2018 Vázquez, J.; Deplano, A.; Herrero, A.; Ginex, T.; Gibert, E.; Rabal, O.; Oyarzabal, J.; Herrero, E.; Luque, F. J. JOURNAL OF CHEMICAL INFORMATION AND MODELING -
Hydrophobic similarity between molecules: Application to three-dimensional molecular overlays with PharmScreen 1-gen-2018 Vazquez, Javier; Deplano, Alessandro; Herrero, Albert; Gibert, Enric; Ginex, Tiziana; Rabal, Obdulia; Oyarzabal, Julen; Herrero, Enric; Luque, F Javier - American Chemical Society
Onthe use (QM) IEF/PMC-MST-derived hydrophobic contributions as physicochemical descriptors in 3D-QSAR: the PHARMSQSARTM approach 1-gen-2018 Rey, Oscar; Ginex, Tiziana; Vazquez, Javier; Deplano, Alessandro; Herrero, Albert; Gibert, Enric; Herrero, Enric; Javier Luque, Francisco - -
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions 1-gen-2017 Corona, Angela; Onnis, Valentina; Deplano, Alessandro; Bianco, Giulia; Demurtas, Monica; Distinto, Simona; Cheng, Yung Chi; Alcaro, Stefano; Esposito, Francesca; Tramontano, Enzo PATHOGENS AND DISEASE -
Novel propanamides as fatty acid amide hydrolase inhibitors 1-gen-2017 Deplano, Alessandro; Morgillo, Carmine Marco; Demurtas, Monica; Björklund, Emmelie; Cipriano, Mariateresa; Svensson, Mona; Hashemian, Sanaz; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Cabiddu, MARIA GRAZIA; Novellino, Ettore; Fowler, Christopher J.; Catalanotti, Bruno; Onnis, Valentina EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones 1-gen-2016 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, A; Manfredini, S; Pacifico, S; Liekens, S; Balzarini, J. MOLECULES -
DESIGN, SYNTHESIS AND PHARMACOLOGICAL INVESTIGATION OF NEW DNA METHYLTRANSFERASE INHIBITORS 1-gen-2016 Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Arimondo, Paola B.; Masson, Veronique; Onnis, Valentina - -
Design, synthesis and SAR of small molecules acting on pain pathways 24-mar-2016 - - Università degli Studi di Cagliari
DIHYDROQUINAZOLINE BENZYLAMIDES AS ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE INHIBITORS 1-gen-2016 Onnis, Valentina; Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol; Catto, Marco; Pisani, Leonardo; Carotti, Angelo - -
Discovery of a novel class of profen derivatives as FAAH inhibitors: MD and QM/MM studies of the binding mode and 3D SAR 1-gen-2016 Morgillo, Cm; Deplano, Alessandro; Karlsson, J; Cipriano, M; Björklund, E; Fowler, Cj; Onnis, Valentina; Luque, Fj; Catalanotti, B. - -