COLLU, GABRIELLA
COLLU, GABRIELLA
DIPARTIMENTO DI SCIENZE BIOMEDICHE
Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives
2021-01-01 Ibba, R.; Piras, S.; Corona, P.; Riu, F.; Loddo, R.; Delogu, I.; Collu, G.; Sanna, G.; Caria, P.; Dettori, T.; Carta, A.
Design, synthesis, antiviral evaluation, and SAR studies of new 1-(phenylsulfonyl)-1H-pyrazol -4-yl-methylaniline derivatives.
2019-01-01 Desideri, N.; Fioravanti, R.; Proietti Monaco, L.; Atzori, E. M.; Carta, A.; Delogu, I.; Collu, G.; and Loddo, R
Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation.
2017-01-01 Fioravanti, R.; Desideri, N.; Carta, A.; Atzori E., M.; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta
A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems
2016-01-01 Carta, A; Briguglio, I; Piras, S; Corona, P; Ibba, R; Laurini, E; Fermeglia, M; Pricl, S; Desideri, N; Atzori, Em; La Colla, P; Collu, G; Delogu, I; Loddo, R
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5
2015-01-01 Loddo, Roberta; Novelli, F; Sparatore, A; Tasso, B; Tonelli, M; Boido, V; Sparatore, F; Collu, Gabriella; Delogu, Ilenia; Giliberti, Gabriele; LA COLLA, Paolo
N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents
2015-01-01 Fioravanti, R; Desideri, N; Biava, M; Droghini, P; Atzori, Em; Ibba, Cristina; Collu, Gabriella; Sanna, Giuseppina; Delogu, Ilenia; Loddo, Roberta
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agents
2015-01-01 Spallarossa, Andrea; Caneva, Chiara; Caviglia, Matteo; Alfei, Silvana; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Brindisi, Margherita; Zisterer, Daniela M.; Bright, Sandra A.; Williams, Clive D.; Crespan, Emmanuele; Maga, Giovanni; Sanna, Giuseppina; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Bruno, O; Schenone, S; LA COLLA, P; Collu, Gabriella; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Schenone, S; Bruno, O; Borassi, A; LA COLLA, P; Pezzullo, M; Sanna, Giuseppina; Collu, Gabriella; Secci, Barbara; Loddo, Roberta
Design, synthesis and anti Flaviviridae activity of N6-, 5’,3’-O- and 5’,2’-O-substituted adenine nucleoside analogs
2008-01-01 Angusti, A; Manfredini, S; Durini, E; Ciliberti, N; Vertuani, S; Solaroli, N; Pricl, S; Ferrone, M; Fermeglia, M; Loddo, Roberta; Secci, Barbara; Visioli, A; Sanna, T; Collu, Gabriella; Pezzullo, M; LA COLLA, P.
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Bruno, O; LA COLLA, P; Casula, L; Collu, Gabriella; Sanna, Giuseppina; Loddo, Roberta
Synthesis and anti-HIV-1 evaluation of 1,5-disubstituted pyrimidine-2,4-diones
2008-01-01 Loksha, Ym; Globisch, D; Pedersen, Eb; LA COLLA, P; Collu, Gabriella; Loddo, Roberta
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Bruno, O; LA COLLA, P; Secci, Barbara; Collu, Gabriella; Loddo, Roberta
Synthesis and anti-Picornaviridae in vitro activity of a new class of helicase inhibitors the N,N’-bis[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkyldicarboxamides
2007-01-01 Loddo, Roberta; Loriga, M; Piras, S; Paglietti, G; Ferrone, M; Fermeglia, M; Pricl, S; LA COLLA, P; Collu, Gabriella; Sanna, T.; Loddo, R.
4-Substituted anilino imidazo[1,2-a] and triazolo[4,3-a]quinoxalines. Synthesis and evaluation of in vitro biological activity
2006-01-01 Corona, P; Vitale, G; Loriga, M; Paglietti, G; LA COLLA, P; Collu, Gabriella; Sanna, Giuseppina; Loddo, Roberta
Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 50-a-hydroxyphosphonates
2006-01-01 Szymanska, A; Szymczak, M; Boryski, J; Stawinski, J; Kraszewski, A; Collu, Gabriella; Sanna, Giuseppina; Giliberti, Gabriele; Loddo, Roberta; La Colla, P.
Synthesis and in vitro evaluation of the anti-viral activity of N-[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkylcarboxamides
2006-01-01 Loddo, Roberta; Loriga, G; Piras, S; Paglietti, G; Ferrone, M; Fermeglia, M; Pricl, S; LA COLLA, P; Secci, Barbara; Collu, Gabriella; Loddo, R.
Synthesis of variously substituted 3-phenoxymethyl quinoxalin-2-ones and quinoxalines capable to potenziate in vitro the antiproliferative activity of anticancer drugs in multi-drug resistant cell lines
2006-01-01 Loddo, Roberta; Loriga, M; Piras, S; Paglietti, G; LA COLLA, P; Busonera, B; Collu, Gabriella
Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives
2005-01-01 Ranise, A; Spallarossa, A; Cesarini, S; Bondavalli, F; Schenone, S; Bruno, O; Menozzi, G; Fossa, P; Mosti, L; La Colla, M; Sanna, Giuseppina; Murreddu, M; Collu, Gabriella; Busonera, B; Marongiu, Me; Pani, Alessandra; La Colla, P; Loddo, Roberta