MOI, DAVIDE
MOI, DAVIDE
DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE
Anticancer potential of chalcones
2026-01-01 Moi, Davide; Onnis, Valentina; Deplano, Alberto
Catalytic Enantioselective Synthesis of Conformationally Stable C(sp2)−C(sp3) Naphthocoumarin Atropisomers
2026-01-01 Cabua, M. Chiara; Moi, Davide; Cocco, Emanuele; Onnis, Valentina; Podda, Enrico; Aitken, David J.; Carlone, Armando; Luisi, Renzo; Tuveri, Enrica; Parsons, Drew F.; Secci, Francesco
Chalcones. From Drug Discovery to Pharmaceutical Applications
2026-01-01 Carradori, Simone; Moi, Davide; D’Agostino, Ilaria
Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential
2026-01-01 Saravanan, Venkatesan; Angeli, Andrea; Melfi, Francesco; Amodio, Nicola; Valentino, Ilenia; Gentile, Massimo; D'Agostino, Ilaria; Muthukumaradoss, Kathiravan; Zengin, Gokhan; Moi, Davide; Simsek, Rahime; Supuran, Claudiu T.; Carradori, Simone
Prokineticin 2 regulates the electrophysiological activity of gonadotropin-releasing hormone neurons via direct signalling in adult female mice
2026-01-01 Farkas, Imre; Göblyös, Barbara; Moi, Davide; Onnis, Valentina; Kalló, Imre; Liposits, Zsolt
Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity
2026-01-01 Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina
The prokineticin system and glia cells as pharmacological targets to control neuroinflammation and to relieve pain in a murine model of Fabry–Anderson disease
2026-01-01 Galimberti, Giulia; Franchi, Silvia; Amodeo, Giada; Romualdi, Patrizia; Candeletti, Sanzio; Rullo, Laura; Losapio, Loredana Maria; Onnis, Valentina; Moi, Davide; Riboldi, Benedetta; Magni, Giulia; Ceruti, Stefania; Sacerdote, Paola
Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides
2025-01-01 Moi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025-01-01 Citarella, Andrea; Belluti, Silvia; Bonanni, Davide; Moi, Davide; Piccinini, Isabella; Rinaldi, Arianna; Papulino, Chiara; Benedetti, Rosaria; Cuoghi, Laura; Ciolo, Stefano Di; Silvani, Alessandra; Altucci, Lucia; Pinzi, Luca; Franchini, Silvia; Passarella, Daniele; Sorbi, Claudia; Giannini, Clelia; Imbriano, Carol; Rastelli, Giulio
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025-01-01 Citarella, Andrea; Sibille, Giulia; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Col, Lorenzo Dal; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Gribaudo, Giorgio; Passarella, Daniele
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors
2024-01-01 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina
Exploring the Antiviral Potential of Esters of Cinnamic Acids with Quercetin
2024-01-01 Manca, Valeria; Chianese, Annalisa; Palmas, Vanessa; Etzi, Federica; Zannella, Carla; Moi, Davide; Secci, Francesco; Serreli, Gabriele; Sarais, Giorgia; Morone, Maria Vittoria; Galdiero, Massimiliano; Onnis, Valentina; Manzin, Aldo; Sanna, Giuseppina
Low‐Impact Synthesis of γ‐Lactones through Photoinduced Baeyer‐Villiger Oxidation of Cyclic Ketones
2024-01-01 Cabua, Maria Chiara; Velichko, Viktoria; Pilia, Luca; Moi, Davide; Secci, Francesco
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024-01-01 Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele
Two-step continuous flow-driven synthesis of 1,1-cyclopropane aminoketones
2024-01-01 Velichko, Viktoria; Moi, Davide; Soddu, Francesco; Scipione, Roberto; Podda, Enrico; Luridiana, Alberto; Cambie, Dario; Secci, Francesco; Cabua, Maria Chiara
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro
2023-01-01 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer
2023-01-01 Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors
2023-01-01 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives
2023-01-01 Citarella, Andrea; Dimasi, Alessandro; Moi, Davide; Passarella, Daniele; Scala, Angela; Piperno, Anna; Micale, Nicola
Synthesis of SARS-CoV-2 Mpro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses
2023-01-01 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Dimasi, Alessandro; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Anticancer potential of chalcones | 1-gen-2026 | Moi, Davide; Onnis, Valentina; Deplano, Alberto | - | Elsevier |
| Catalytic Enantioselective Synthesis of Conformationally Stable C(sp2)−C(sp3) Naphthocoumarin Atropisomers | 1-gen-2026 | Cabua, M. Chiara; Moi, Davide; Cocco, Emanuele; Onnis, Valentina; Podda, Enrico; Aitken, David J.; Carlone, Armando; Luisi, Renzo; Tuveri, Enrica; Parsons, Drew F.; Secci, Francesco | ADVANCED SYNTHESIS & CATALYSIS | - |
| Chalcones. From Drug Discovery to Pharmaceutical Applications | 1-gen-2026 | Carradori, Simone; Moi, Davide; D’Agostino, Ilaria | - | Elsevier |
| Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential | 1-gen-2026 | Saravanan, Venkatesan; Angeli, Andrea; Melfi, Francesco; Amodio, Nicola; Valentino, Ilenia; Gentile, Massimo; D'Agostino, Ilaria; Muthukumaradoss, Kathiravan; Zengin, Gokhan; Moi, Davide; Simsek, Rahime; Supuran, Claudiu T.; Carradori, Simone | PHARMACEUTICALS | - |
| Prokineticin 2 regulates the electrophysiological activity of gonadotropin-releasing hormone neurons via direct signalling in adult female mice | 1-gen-2026 | Farkas, Imre; Göblyös, Barbara; Moi, Davide; Onnis, Valentina; Kalló, Imre; Liposits, Zsolt | FRONTIERS IN ENDOCRINOLOGY | - |
| Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity | 1-gen-2026 | Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina | PHARMACEUTICALS | - |
| The prokineticin system and glia cells as pharmacological targets to control neuroinflammation and to relieve pain in a murine model of Fabry–Anderson disease | 1-gen-2026 | Galimberti, Giulia; Franchi, Silvia; Amodeo, Giada; Romualdi, Patrizia; Candeletti, Sanzio; Rullo, Laura; Losapio, Loredana Maria; Onnis, Valentina; Moi, Davide; Riboldi, Benedetta; Magni, Giulia; Ceruti, Stefania; Sacerdote, Paola | PAIN | - |
| Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides | 1-gen-2025 | Moi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina | PHARMACEUTICALS | - |
| Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer | 1-gen-2025 | Citarella, Andrea; Belluti, Silvia; Bonanni, Davide; Moi, Davide; Piccinini, Isabella; Rinaldi, Arianna; Papulino, Chiara; Benedetti, Rosaria; Cuoghi, Laura; Ciolo, Stefano Di; Silvani, Alessandra; Altucci, Lucia; Pinzi, Luca; Franchini, Silvia; Passarella, Daniele; Sorbi, Claudia; Giannini, Clelia; Imbriano, Carol; Rastelli, Giulio | JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity | 1-gen-2025 | Citarella, Andrea; Sibille, Giulia; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Col, Lorenzo Dal; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Gribaudo, Giorgio; Passarella, Daniele | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors | 1-gen-2024 | Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina | ACS MEDICINAL CHEMISTRY LETTERS | - |
| Exploring the Antiviral Potential of Esters of Cinnamic Acids with Quercetin | 1-gen-2024 | Manca, Valeria; Chianese, Annalisa; Palmas, Vanessa; Etzi, Federica; Zannella, Carla; Moi, Davide; Secci, Francesco; Serreli, Gabriele; Sarais, Giorgia; Morone, Maria Vittoria; Galdiero, Massimiliano; Onnis, Valentina; Manzin, Aldo; Sanna, Giuseppina | VIRUSES | - |
| Low‐Impact Synthesis of γ‐Lactones through Photoinduced Baeyer‐Villiger Oxidation of Cyclic Ketones | 1-gen-2024 | Cabua, Maria Chiara; Velichko, Viktoria; Pilia, Luca; Moi, Davide; Secci, Francesco | EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | - |
| Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells | 1-gen-2024 | Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Two-step continuous flow-driven synthesis of 1,1-cyclopropane aminoketones | 1-gen-2024 | Velichko, Viktoria; Moi, Davide; Soddu, Francesco; Scipione, Roberto; Podda, Enrico; Luridiana, Alberto; Cambie, Dario; Secci, Francesco; Cabua, Maria Chiara | CHEMICAL COMMUNICATIONS | - |
| Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro | 1-gen-2023 | Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia | MOLECULES | - |
| Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer | 1-gen-2023 | Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors | 1-gen-2023 | Moi, Davide; Vittorio, Serena; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | MOLECULES | - |
| Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives | 1-gen-2023 | Citarella, Andrea; Dimasi, Alessandro; Moi, Davide; Passarella, Daniele; Scala, Angela; Piperno, Anna; Micale, Nicola | BIOMOLECULES | - |
| Synthesis of SARS-CoV-2 Mpro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses | 1-gen-2023 | Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Dimasi, Alessandro; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele | ORGANIC & BIOMOLECULAR CHEMISTRY | - |