MOI, DAVIDE

MOI, DAVIDE  

DIPARTIMENTO DI SCIENZE DELLA VITA E DELL'AMBIENTE  

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Risultati 1 - 20 di 39 (tempo di esecuzione: 0.036 secondi).
Titolo Data di pubblicazione Autore(i) Rivista Editore
Anticancer potential of chalcones 1-gen-2026 Moi, Davide; Onnis, Valentina; Deplano, Alberto - Elsevier
Catalytic Enantioselective Synthesis of Conformationally Stable C(sp2)−C(sp3) Naphthocoumarin Atropisomers 1-gen-2026 Cabua, M. Chiara; Moi, Davide; Cocco, Emanuele; Onnis, Valentina; Podda, Enrico; Aitken, David J.; Carlone, Armando; Luisi, Renzo; Tuveri, Enrica; Parsons, Drew F.; Secci, Francesco ADVANCED SYNTHESIS & CATALYSIS -
Chalcones. From Drug Discovery to Pharmaceutical Applications 1-gen-2026 Carradori, Simone; Moi, Davide; D’Agostino, Ilaria - Elsevier
Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential 1-gen-2026 Saravanan, Venkatesan; Angeli, Andrea; Melfi, Francesco; Amodio, Nicola; Valentino, Ilenia; Gentile, Massimo; D'Agostino, Ilaria; Muthukumaradoss, Kathiravan; Zengin, Gokhan; Moi, Davide; Simsek, Rahime; Supuran, Claudiu T.; Carradori, Simone PHARMACEUTICALS -
Prokineticin 2 regulates the electrophysiological activity of gonadotropin-releasing hormone neurons via direct signalling in adult female mice 1-gen-2026 Farkas, Imre; Göblyös, Barbara; Moi, Davide; Onnis, Valentina; Kalló, Imre; Liposits, Zsolt FRONTIERS IN ENDOCRINOLOGY -
Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity 1-gen-2026 Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina PHARMACEUTICALS -
The prokineticin system and glia cells as pharmacological targets to control neuroinflammation and to relieve pain in a murine model of Fabry–Anderson disease 1-gen-2026 Galimberti, Giulia; Franchi, Silvia; Amodeo, Giada; Romualdi, Patrizia; Candeletti, Sanzio; Rullo, Laura; Losapio, Loredana Maria; Onnis, Valentina; Moi, Davide; Riboldi, Benedetta; Magni, Giulia; Ceruti, Stefania; Sacerdote, Paola PAIN -
Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides 1-gen-2025 Moi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina PHARMACEUTICALS -
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer 1-gen-2025 Citarella, Andrea; Belluti, Silvia; Bonanni, Davide; Moi, Davide; Piccinini, Isabella; Rinaldi, Arianna; Papulino, Chiara; Benedetti, Rosaria; Cuoghi, Laura; Ciolo, Stefano Di; Silvani, Alessandra; Altucci, Lucia; Pinzi, Luca; Franchini, Silvia; Passarella, Daniele; Sorbi, Claudia; Giannini, Clelia; Imbriano, Carol; Rastelli, Giulio JOURNAL OF MEDICINAL CHEMISTRY -
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity 1-gen-2025 Citarella, Andrea; Sibille, Giulia; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Col, Lorenzo Dal; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Gribaudo, Giorgio; Passarella, Daniele BIOORGANIC & MEDICINAL CHEMISTRY -
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors 1-gen-2024 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina ACS MEDICINAL CHEMISTRY LETTERS -
Exploring the Antiviral Potential of Esters of Cinnamic Acids with Quercetin 1-gen-2024 Manca, Valeria; Chianese, Annalisa; Palmas, Vanessa; Etzi, Federica; Zannella, Carla; Moi, Davide; Secci, Francesco; Serreli, Gabriele; Sarais, Giorgia; Morone, Maria Vittoria; Galdiero, Massimiliano; Onnis, Valentina; Manzin, Aldo; Sanna, Giuseppina VIRUSES -
Low‐Impact Synthesis of γ‐Lactones through Photoinduced Baeyer‐Villiger Oxidation of Cyclic Ketones 1-gen-2024 Cabua, Maria Chiara; Velichko, Viktoria; Pilia, Luca; Moi, Davide; Secci, Francesco EUROPEAN JOURNAL OF ORGANIC CHEMISTRY -
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells 1-gen-2024 Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele BIOORGANIC & MEDICINAL CHEMISTRY -
Two-step continuous flow-driven synthesis of 1,1-cyclopropane aminoketones 1-gen-2024 Velichko, Viktoria; Moi, Davide; Soddu, Francesco; Scipione, Roberto; Podda, Enrico; Luridiana, Alberto; Cambie, Dario; Secci, Francesco; Cabua, Maria Chiara CHEMICAL COMMUNICATIONS -
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro 1-gen-2023 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia MOLECULES -
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer 1-gen-2023 Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors 1-gen-2023 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina MOLECULES -
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives 1-gen-2023 Citarella, Andrea; Dimasi, Alessandro; Moi, Davide; Passarella, Daniele; Scala, Angela; Piperno, Anna; Micale, Nicola BIOMOLECULES -
Synthesis of SARS-CoV-2 Mpro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses 1-gen-2023 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Dimasi, Alessandro; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele ORGANIC & BIOMOLECULAR CHEMISTRY -