LAUS, ANTONIO
LAUS, ANTONIO
DIPARTIMENTO DI SCIENZE BIOMEDICHE
Dihydroxyphenyl- and Heteroaromatic-Based Thienopyrimidinones to Tackle HIV-1 LEDGF/p75-Dependent IN Activity
2023-01-01 Tocco, G.; Canton, S.; Laus, A.; Caboni, P.; Le Grice, S. F. J.; Tramontano, E.; Esposito, F.
In silico characterization of ligand–receptor interactions for U-47700, N,N-didesmethyl-U-47700, U-50488 at mu- and kappa-opioid receptors
2023-01-01 Laus, A; Kumar, A; Caboni, P; DE LUCA, MARIA ANTONIETTA; Baumann, Mh; Pieroni, E; Tocco, G.
Off‑target activity of NBOMes and NBOMe analogs at the µ opioid receptor
2023-01-01 Deventer, Marie H.; Persson, Mattias; Laus, Antonio; Pottie, Eline; Cannaert, Annelies; Tocco, Graziella; Gréen, Henrik; Stove, Christophe P.
Structural Elucidation of Relevant Gibberellic Acid Impurities and In Silico Investigation of Their Interaction with Soluble Gibberellin Receptor GID1
2023-01-01 Caboni, Pierluigi; Laus, Antonio; Eloh, Kodjo; Ntalli, Nikoletta G.; Casula, Mattia; Di Giorgi, Sabrina; Tocco, Graziella
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists
2022-01-01 Tocco, Graziella; Laus, Antonio; Vanejevs, Maksims; Ture, Anastasija; Mostallino, Rafaela; Pintori, Nicholas; De Luca, Maria Antonietta; Castelli, M. Paola; Di Chiara, Gaetano
Mukaiyama reagent: An efficient reaction mediator for rapid synthesis of 1,2-disubstituted-1H-benzo[d]imidazoles
2022-01-01 Tocco, G.; Laus, A.; Caboni, P.
Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists
2022-01-01 De Luca, Maria Antonietta; Tocco, Graziella; Mostallino, Rafaela; Laus, Antonio; Caria, Francesca; Musa, Aurora; Pintori, Nicholas; Ucha, Marcos; Poza, Celia; Ambrosio, Emilio; Di Chiara, Gaetano; Castelli, M Paola
Electron-Deficient Alkynes as Powerful Tools against Root-Knot Nematode Melodogyne incognita: Nematicidal Activity and Investigation on the Mode of Action
2020-01-01 Tocco, Graziella; Eloh, Kodjo; Laus, Antonio; Sasanelli, Nicola; Caboni, Pierluigi
Scaffold hopping and optimisation of 3’,4’-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H
2020-01-01 Tocco, Graziella; Esposito, Francesca; Caboni, Pierluigi; Laus, Antonio; Beutler, John A.; Wilson, Jennifer A.; Corona, Angela; Le Grice, Stuart F. J.; Tramontano, Enzo