Sfoglia per Autore
S-layer proteins as a source of carotenoids: Isolation of the carotenoid cofactor deinoxanthin from its S-layer protein DR_2577
2017-01-01 Farci, Domenica; Esposito, Francesca; El Alaoui, Sabah; Piano, Dario
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action
2017-01-01 Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo
Chelation motifs affecting metal-dependent viral enzymes: N′-acylhydrazone ligands as dual target inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H domain
2017-01-01 Carcelli, Mauro; Rogolino, Dominga; Gatti, Anna; Pala, Nicolino; Corona, Angela; Caredda, Alessia; Tramontano, Enzo; Pannecouque, Christophe; Naesens, Lieve; Esposito, Francesca
Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding
2017-01-01 Martini, Riccardo; Esposito, Francesca; Corona, Angela; Ferrarese, Roberto; Ceresola, Elisa Rita; Visconti, Laura; Tintori, Cristina; Barbieri, Alessandro; Calcaterra, Andrea; Iovine, Valentina; Canducci, Filippo; Tramontano, Enzo; Botta, Maurizio
Inhibition of HIV-1 reverse transcriptase dimerization by small molecules
2016-01-01 Tintori, C; Corona, Angela; Esposito, Francesca; Brai, A; Grandi, Nicole; Ceresola, Er; Clementi, M; Canducci, F; Tramontano, Enzo; Botta, M.
Inhibitory effect of 2,3,5,6-tetrafluoro-4-[4-(Aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide derivatives on HIV reverse transcriptase associated rnase H activities
2016-01-01 Pala, Nicolino; Esposito, Francesca; Rogolino, Dominga; Carcelli, Mauro; Sanna, Vanna; Palomba, Michele; Naesens, Lieve; Corona, Angela; Grandi, Nicole; Tramontano, Enzo; Sechi, Mario
RhVI1 is a membrane-anchored vacuolar invertase highly expressed in Rosa hybrida L. petals
2016-01-01 Farci, Domenica; Collu, Gabriella; Kirkpatrick, Joanna; Esposito, Francesca; Piano, Dario
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H
2016-01-01 Corona, Angela; di Leva, Francesco Saverio; Rigogliuso, Giuseppe; Pescatori, Luca; Madia, Valentina Noemi; Subra, Frederic; Delelis, Olivier; Esposito, Francesca; Cadeddu, Marta; Costi, Roberta; Cosconati, Sandro; Novellino, Ettore; di Santo, Roberto; Tramontano, Enzo
Biological activities of aerial parts extracts of Euphorbia characias
2016-01-01 Pisano, MARIA BARBARA; Cosentino, Sofia; Viale, Silvia; Spano', Delia; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Montoro, P; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca
Sennoside A, derived from the traditional chinese medicine plant Rheum L., is a new dual HIV-1 inhibitor effective on HIV-1 replication
2016-01-01 Esposito, Francesca; Carli, Ilaria; Del Vecchio, Claudia; Xu, Lijia; Corona, Angela; Grandi, Nicole; Piano, Dario; Maccioni, Elias; Distinto, Simona; Parolin, Cristina; Tramontano, Enzo
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6
2016-01-01 Corona, Angela; Meleddu, Rita; Esposito, Francesca; Distinto, Simona; Bianco, Giulia; Masaoka, T; Maccioni, Elias; Menéndez Arias, L; Alcaro, S; Le Grice, Sfj; Tramontano, Enzo
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors
2016-01-01 Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J; Tramontano, Enzo; Tabarrini, Oriana
Development and identification of a novel anti-HIV-1 peptide derived by modification of the N-terminal domain of HIV-1 integrase
2016-01-01 Sala, M; Spensiero, A; Esposito, Francesca; Scala, Mc; Vernieri, E; Bertamino, A; Manfra, M; Carotenuto, A; Grieco, P; Novellino, E; Cadeddu, Marta; Tramontano, Enzo; Schols, D; Campiglia, P; Gomez Monterrey, Im
From the traditional Chinese medicine plant Schisandra chinensis new scaffolds effective on HIV-1 reverse transcriptase resistant to non-nucleoside inhibitors
2015-01-01 Xu, L; Grandi, Nicole; Del Vecchio, C; Mandas, D; Corona, Angela; Piano, Dario; Esposito, Francesca; Parolin, C; Tramontano, Enzo
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias
An efficient route to novel uracil-based drug-like molecules
2015-01-01 Babkov, Da; Chizhov, Ao; Khandazhinskaya, Al; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; SELEY RADTKE, Kl; Novikov, Ms
Structure-Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain
2015-01-01 Cuzzucoli Crucitti, G; Métifiot, M; Pescatori, L; Messore, A; Madia V., N; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S; Esposito, Francesca; Corona, Angela; Cadeddu, M; Marchand, C; Pommier, Y; Tramontano, Enzo; Costi, R; Di Santo, R.
Kuwanon-L as a new allosteric HIV-1 integrase inhibitor: molecular modeling and biological evaluation
2015-01-01 Esposito, Francesca; Tintori, C; Martini, R; Christ, F; Debyser, Z; Ferrarese, R; Cabiddu, Gianluigi; Corona, Angela; Ceresola E., R; Calcaterra, A; Iovine, V; Botta, B; Clementi, M; Canducci, F; Botta, M; Tramontano, Enzo
Euphorbia characias latex: Micromorphology of rubber particles and rubber transferase activity
2015-01-01 Spanò, D; Pintus, Francesca; Esposito, Francesca; Loche, Danilo; Floris, Giovanni; Medda, Rosaria
Investigation on the sucrose binding pocket of HIV-1 Integrase by molecular dynamics and synergy experiments
2015-01-01 Tintori, C; Esposito, Francesca; Morreale, F; Martini, R; Tramontano, Enzo; Botta, M.
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
S-layer proteins as a source of carotenoids: Isolation of the carotenoid cofactor deinoxanthin from its S-layer protein DR_2577 | 1-gen-2017 | Farci, Domenica; Esposito, Francesca; El Alaoui, Sabah; Piano, Dario | FOOD RESEARCH INTERNATIONAL | - |
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action | 1-gen-2017 | Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo | PATHOGENS AND DISEASE | - |
Chelation motifs affecting metal-dependent viral enzymes: N′-acylhydrazone ligands as dual target inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H domain | 1-gen-2017 | Carcelli, Mauro; Rogolino, Dominga; Gatti, Anna; Pala, Nicolino; Corona, Angela; Caredda, Alessia; Tramontano, Enzo; Pannecouque, Christophe; Naesens, Lieve; Esposito, Francesca | FRONTIERS IN MICROBIOLOGY | - |
Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding | 1-gen-2017 | Martini, Riccardo; Esposito, Francesca; Corona, Angela; Ferrarese, Roberto; Ceresola, Elisa Rita; Visconti, Laura; Tintori, Cristina; Barbieri, Alessandro; Calcaterra, Andrea; Iovine, Valentina; Canducci, Filippo; Tramontano, Enzo; Botta, Maurizio | CHEMBIOCHEM | - |
Inhibition of HIV-1 reverse transcriptase dimerization by small molecules | 1-gen-2016 | Tintori, C; Corona, Angela; Esposito, Francesca; Brai, A; Grandi, Nicole; Ceresola, Er; Clementi, M; Canducci, F; Tramontano, Enzo; Botta, M. | CHEMBIOCHEM | - |
Inhibitory effect of 2,3,5,6-tetrafluoro-4-[4-(Aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide derivatives on HIV reverse transcriptase associated rnase H activities | 1-gen-2016 | Pala, Nicolino; Esposito, Francesca; Rogolino, Dominga; Carcelli, Mauro; Sanna, Vanna; Palomba, Michele; Naesens, Lieve; Corona, Angela; Grandi, Nicole; Tramontano, Enzo; Sechi, Mario | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
RhVI1 is a membrane-anchored vacuolar invertase highly expressed in Rosa hybrida L. petals | 1-gen-2016 | Farci, Domenica; Collu, Gabriella; Kirkpatrick, Joanna; Esposito, Francesca; Piano, Dario | JOURNAL OF EXPERIMENTAL BOTANY | - |
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H | 1-gen-2016 | Corona, Angela; di Leva, Francesco Saverio; Rigogliuso, Giuseppe; Pescatori, Luca; Madia, Valentina Noemi; Subra, Frederic; Delelis, Olivier; Esposito, Francesca; Cadeddu, Marta; Costi, Roberta; Cosconati, Sandro; Novellino, Ettore; di Santo, Roberto; Tramontano, Enzo | ANTIVIRAL RESEARCH | - |
Biological activities of aerial parts extracts of Euphorbia characias | 1-gen-2016 | Pisano, MARIA BARBARA; Cosentino, Sofia; Viale, Silvia; Spano', Delia; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Montoro, P; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca | BIOMED RESEARCH INTERNATIONAL | - |
Sennoside A, derived from the traditional chinese medicine plant Rheum L., is a new dual HIV-1 inhibitor effective on HIV-1 replication | 1-gen-2016 | Esposito, Francesca; Carli, Ilaria; Del Vecchio, Claudia; Xu, Lijia; Corona, Angela; Grandi, Nicole; Piano, Dario; Maccioni, Elias; Distinto, Simona; Parolin, Cristina; Tramontano, Enzo | PHYTOMEDICINE | - |
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6 | 1-gen-2016 | Corona, Angela; Meleddu, Rita; Esposito, Francesca; Distinto, Simona; Bianco, Giulia; Masaoka, T; Maccioni, Elias; Menéndez Arias, L; Alcaro, S; Le Grice, Sfj; Tramontano, Enzo | PLOS ONE | - |
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors | 1-gen-2016 | Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J; Tramontano, Enzo; Tabarrini, Oriana | CHEMMEDCHEM | - |
Development and identification of a novel anti-HIV-1 peptide derived by modification of the N-terminal domain of HIV-1 integrase | 1-gen-2016 | Sala, M; Spensiero, A; Esposito, Francesca; Scala, Mc; Vernieri, E; Bertamino, A; Manfra, M; Carotenuto, A; Grieco, P; Novellino, E; Cadeddu, Marta; Tramontano, Enzo; Schols, D; Campiglia, P; Gomez Monterrey, Im | FRONTIERS IN MICROBIOLOGY | - |
From the traditional Chinese medicine plant Schisandra chinensis new scaffolds effective on HIV-1 reverse transcriptase resistant to non-nucleoside inhibitors | 1-gen-2015 | Xu, L; Grandi, Nicole; Del Vecchio, C; Mandas, D; Corona, Angela; Piano, Dario; Esposito, Francesca; Parolin, C; Tramontano, Enzo | JOURNAL OF MICROBIOLOGY | - |
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
An efficient route to novel uracil-based drug-like molecules | 1-gen-2015 | Babkov, Da; Chizhov, Ao; Khandazhinskaya, Al; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; SELEY RADTKE, Kl; Novikov, Ms | SYNTHESIS | - |
Structure-Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain | 1-gen-2015 | Cuzzucoli Crucitti, G; Métifiot, M; Pescatori, L; Messore, A; Madia V., N; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S; Esposito, Francesca; Corona, Angela; Cadeddu, M; Marchand, C; Pommier, Y; Tramontano, Enzo; Costi, R; Di Santo, R. | JOURNAL OF MEDICINAL CHEMISTRY | - |
Kuwanon-L as a new allosteric HIV-1 integrase inhibitor: molecular modeling and biological evaluation | 1-gen-2015 | Esposito, Francesca; Tintori, C; Martini, R; Christ, F; Debyser, Z; Ferrarese, R; Cabiddu, Gianluigi; Corona, Angela; Ceresola E., R; Calcaterra, A; Iovine, V; Botta, B; Clementi, M; Canducci, F; Botta, M; Tramontano, Enzo | CHEMBIOCHEM | - |
Euphorbia characias latex: Micromorphology of rubber particles and rubber transferase activity | 1-gen-2015 | Spanò, D; Pintus, Francesca; Esposito, Francesca; Loche, Danilo; Floris, Giovanni; Medda, Rosaria | PLANT PHYSIOLOGY AND BIOCHEMISTRY | - |
Investigation on the sucrose binding pocket of HIV-1 Integrase by molecular dynamics and synergy experiments | 1-gen-2015 | Tintori, C; Esposito, Francesca; Morreale, F; Martini, R; Tramontano, Enzo; Botta, M. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile