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Titolo Data di pubblicazione Autore(i) Rivista Editore
S-layer proteins as a source of carotenoids: Isolation of the carotenoid cofactor deinoxanthin from its S-layer protein DR_2577 1-gen-2017 Farci, Domenica; Esposito, Francesca; El Alaoui, Sabah; Piano, Dario FOOD RESEARCH INTERNATIONAL -
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action 1-gen-2017 Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo PATHOGENS AND DISEASE -
Chelation motifs affecting metal-dependent viral enzymes: N′-acylhydrazone ligands as dual target inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H domain 1-gen-2017 Carcelli, Mauro; Rogolino, Dominga; Gatti, Anna; Pala, Nicolino; Corona, Angela; Caredda, Alessia; Tramontano, Enzo; Pannecouque, Christophe; Naesens, Lieve; Esposito, Francesca FRONTIERS IN MICROBIOLOGY -
Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding 1-gen-2017 Martini, Riccardo; Esposito, Francesca; Corona, Angela; Ferrarese, Roberto; Ceresola, Elisa Rita; Visconti, Laura; Tintori, Cristina; Barbieri, Alessandro; Calcaterra, Andrea; Iovine, Valentina; Canducci, Filippo; Tramontano, Enzo; Botta, Maurizio CHEMBIOCHEM -
Inhibition of HIV-1 reverse transcriptase dimerization by small molecules 1-gen-2016 Tintori, C; Corona, Angela; Esposito, Francesca; Brai, A; Grandi, Nicole; Ceresola, Er; Clementi, M; Canducci, F; Tramontano, Enzo; Botta, M. CHEMBIOCHEM -
Inhibitory effect of 2,3,5,6-tetrafluoro-4-[4-(Aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide derivatives on HIV reverse transcriptase associated rnase H activities 1-gen-2016 Pala, Nicolino; Esposito, Francesca; Rogolino, Dominga; Carcelli, Mauro; Sanna, Vanna; Palomba, Michele; Naesens, Lieve; Corona, Angela; Grandi, Nicole; Tramontano, Enzo; Sechi, Mario INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES -
RhVI1 is a membrane-anchored vacuolar invertase highly expressed in Rosa hybrida L. petals 1-gen-2016 Farci, Domenica; Collu, Gabriella; Kirkpatrick, Joanna; Esposito, Francesca; Piano, Dario JOURNAL OF EXPERIMENTAL BOTANY -
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H 1-gen-2016 Corona, Angela; di Leva, Francesco Saverio; Rigogliuso, Giuseppe; Pescatori, Luca; Madia, Valentina Noemi; Subra, Frederic; Delelis, Olivier; Esposito, Francesca; Cadeddu, Marta; Costi, Roberta; Cosconati, Sandro; Novellino, Ettore; di Santo, Roberto; Tramontano, Enzo ANTIVIRAL RESEARCH -
Biological activities of aerial parts extracts of Euphorbia characias 1-gen-2016 Pisano, MARIA BARBARA; Cosentino, Sofia; Viale, Silvia; Spano', Delia; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; Montoro, P; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca BIOMED RESEARCH INTERNATIONAL -
Sennoside A, derived from the traditional chinese medicine plant Rheum L., is a new dual HIV-1 inhibitor effective on HIV-1 replication 1-gen-2016 Esposito, Francesca; Carli, Ilaria; Del Vecchio, Claudia; Xu, Lijia; Corona, Angela; Grandi, Nicole; Piano, Dario; Maccioni, Elias; Distinto, Simona; Parolin, Cristina; Tramontano, Enzo PHYTOMEDICINE -
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6 1-gen-2016 Corona, Angela; Meleddu, Rita; Esposito, Francesca; Distinto, Simona; Bianco, Giulia; Masaoka, T; Maccioni, Elias; Menéndez Arias, L; Alcaro, S; Le Grice, Sfj; Tramontano, Enzo PLOS ONE -
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors 1-gen-2016 Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J; Tramontano, Enzo; Tabarrini, Oriana CHEMMEDCHEM -
Development and identification of a novel anti-HIV-1 peptide derived by modification of the N-terminal domain of HIV-1 integrase 1-gen-2016 Sala, M; Spensiero, A; Esposito, Francesca; Scala, Mc; Vernieri, E; Bertamino, A; Manfra, M; Carotenuto, A; Grieco, P; Novellino, E; Cadeddu, Marta; Tramontano, Enzo; Schols, D; Campiglia, P; Gomez Monterrey, Im FRONTIERS IN MICROBIOLOGY -
From the traditional Chinese medicine plant Schisandra chinensis new scaffolds effective on HIV-1 reverse transcriptase resistant to non-nucleoside inhibitors 1-gen-2015 Xu, L; Grandi, Nicole; Del Vecchio, C; Mandas, D; Corona, Angela; Piano, Dario; Esposito, Francesca; Parolin, C; Tramontano, Enzo JOURNAL OF MICROBIOLOGY -
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 1-gen-2015 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
An efficient route to novel uracil-based drug-like molecules 1-gen-2015 Babkov, Da; Chizhov, Ao; Khandazhinskaya, Al; Corona, Angela; Esposito, Francesca; Tramontano, Enzo; SELEY RADTKE, Kl; Novikov, Ms SYNTHESIS -
Structure-Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain 1-gen-2015 Cuzzucoli Crucitti, G; Métifiot, M; Pescatori, L; Messore, A; Madia V., N; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S; Esposito, Francesca; Corona, Angela; Cadeddu, M; Marchand, C; Pommier, Y; Tramontano, Enzo; Costi, R; Di Santo, R. JOURNAL OF MEDICINAL CHEMISTRY -
Kuwanon-L as a new allosteric HIV-1 integrase inhibitor: molecular modeling and biological evaluation 1-gen-2015 Esposito, Francesca; Tintori, C; Martini, R; Christ, F; Debyser, Z; Ferrarese, R; Cabiddu, Gianluigi; Corona, Angela; Ceresola E., R; Calcaterra, A; Iovine, V; Botta, B; Clementi, M; Canducci, F; Botta, M; Tramontano, Enzo CHEMBIOCHEM -
Euphorbia characias latex: Micromorphology of rubber particles and rubber transferase activity 1-gen-2015 Spanò, D; Pintus, Francesca; Esposito, Francesca; Loche, Danilo; Floris, Giovanni; Medda, Rosaria PLANT PHYSIOLOGY AND BIOCHEMISTRY -
Investigation on the sucrose binding pocket of HIV-1 Integrase by molecular dynamics and synergy experiments 1-gen-2015 Tintori, C; Esposito, Francesca; Morreale, F; Martini, R; Tramontano, Enzo; Botta, M. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS -
Mostrati risultati da 41 a 60 di 127
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