Sfoglia per Autore
In Vitro Anti-HIV-1 Reverse Transcriptase and Integrase Properties of Punica granatum L. Leaves, Bark, and Peel Extracts and Their Main Compounds
2021-01-01 Sanna, C.; Marengo, A.; Acquadro, S.; Caredda, A.; Lai, R.; Corona, A.; Tramontano, E.; Rubiolo, P.; Esposito, F.
Integration of SARS-CoV-2 RNA in infected human cells by retrotransposons: an unlikely hypothesis and old viral relationships
2021-01-01 Grandi, N.; Tramontano, E.; Berkhout, B.
Zika virus NS2A inhibits interferon signaling by degradation of STAT1 and STAT2
2021-01-01 Fanunza, Elisa; Carletti, Fabrizio; Quartu, Marina; Grandi, Nicole; Ermellino, Laura; Milia, Jessica; Corona, Angela; Capobianchi, Maria Rosaria; Ippolito, Giuseppe; Tramontano, Enzo
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function
2021-01-01 Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo
Inhibitors of Ebolavirus targeting innate immune evasion
2021-01-01 Paulis, A. L.; Corona, A.; Tramontano, E.
Early Diffusion of SARS-CoV-2 Infection in the Inner Area of the Italian Sardinia Island
2021-01-01 Piras, Giovanna; Grandi, Nicole; Monne, Maria; Asproni, Rosanna; Fancello, Tatiana; Fiamma, Maura; Mameli, Giuseppe; Casu, Gavino; lo Maglio, Iana; Palmas, Angelo D.; Tramontano, Enzo
Natural and Nature-Derived Products Targeting Human Coronaviruses
2021-01-01 Vougogiannopoulou, Konstantina; Corona, Angela; Tramontano, Enzo; Alexis, Michael N.; Skaltsounis, Alexios-Leandros
Garcinol from Garcinia indica inhibits HIV-1 reverse transcriptase-associated ribonuclease H
2021-01-01 Corona, Angela; Seibt, Sebastian; Schaller, David; Schobert, Rainer; Volkamer, Andrea; Biersack, Bernhard; Tramontano, Enzo
INMI1 Zika Virus NS4B Antagonizes the Interferon Signaling by Suppressing STAT1 Phosphorylation
2021-01-01 Fanunza, Elisa; Grandi, Nicole; Quartu, Marina; Carletti, Fabrizio; Ermellino, Laura; Milia, Jessica; Corona, Angela; Rosaria Capobianchi, Maria; Ippolito, Giuseppe; Tramontano, Enzo
Diagnosi in vitro della Sclerosi Multipla
2020-01-01 Grandi, Nicole; Pisano, MARIA PAOLA; Tramontano, Enzo
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture
2020-01-01 Pala, Nicolino; Esposito, Francesca; Tramontano, Enzo; Kumar Singh, Pankaj; Sanna, Vanna; Carcelli, Mauro; Haigh, Lisa D.; Satta, Sandro; Mario Sechi, And
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity
2020-01-01 Desantis, Jenny; Massari, Serena; Corona, Angela; Astolfi, Andrea; Sabatini, Stefano; Manfroni, Giuseppe; Palazzotti, Deborah; Cecchetti, Violetta; Pannecouque, Christophe; Tramontano, Enzo; Tabarrini, Oriana
Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition
2020-01-01 Hayek, S.; Pietrancosta, N.; Hovhannisyan, A. A.; Alves de Sousa, R.; Bekaddour, N.; Ermellino, L.; Tramontano, E.; Arnould, S.; Sardet, C.; Dairou, J.; Diaz, O.; Lotteau, V.; Nisole, S.; Melikyan, G.; Herbeuval, J. -P.; Vidalain, P. -O.
Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitors
2020-01-01 Esposito, Francesca; Sechi, Mario; Pala, Nicolino; Sanna, Adele; Koneru, Pratibha Chowdary; Kvaratskhelia, Mamuka; Naesens, Lieve; Corona, Angela; Grandi, Nicole; di Santo, Roberto; D'Amore, Vincenzo Maria; Di Leva, Francesco Saverio; Novellino, Ettore; Cosconati, Sandro; Tramontano, Enzo
Peptides Mimicking the β7/β8 loop of HIV-1 Reverse Transcriptase p51 as “Hotspot-Targeted” Dimerization Inhibitors
2020-01-01 Sánchez-Murcia, Pedro A.; de Castro, Sonia; García-Aparicio, Carlos; Jimenez, M. Angeles; Corona, Angela; Tramontano, Enzo; Sluis-Cremer, Nicolas; Menendez Arias, Luis; Velazquez, Sonsoles; Gago, Federico; Camarasa, María-José
2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication
2020-01-01 Corona, Angela; Onnis, Valentina; Del Vecchio, Claudia; Esposito, Francesca; Cheng, Yung-Chi; Tramontano, Enzo
Quercetin blocks Ebola Virus infection by counteracting the VP24 Interferon inhibitory function
2020-01-01 Fanunza, Elisa; Iampietro, Mathieu; Distinto, Simona; Corona, Angela; Quartu, Marina; Maccioni, Elias; Horvat, Branka; Tramontano, Enzo
A human MMTV-like betaretrovirus linked to breast cancer has been present in humans at least since the Copper Age
2020-01-01 Lessi, F.; Grandi, N.; Mazzanti, C. M.; Civita, P.; Scatena, C.; Aretini, P.; Bandiera, P.; Fornaciari, A.; Giuffra, V.; Fornaciari, G.; Naccarato, A. G.; Tramontano, E.; Bevilacqua, G.
Targeting HIV-1 RNase H: N'-(2-Hydroxy-benzylidene)-3,4,5-Trihydroxybenzoylhydrazone as Selective Inhibitor Active against NNRTIs-Resistant Variants
2020-01-01 Corona, Angela; Ballana, Ester; Distinto, Simona; Rogolino, Dominga; Del Vecchio, Claudia; Carcelli, Mauro; Badia, Roger; Riveira-Muñoz, Eva; Esposito, Francesca; Parolin, Cristina; Esté, José A; Grandi, Nicole; Tramontano, Enzo
Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase
2020-01-01 Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Di Maro, Salvatore; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Valenti, Piera; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
In Vitro Anti-HIV-1 Reverse Transcriptase and Integrase Properties of Punica granatum L. Leaves, Bark, and Peel Extracts and Their Main Compounds | 1-gen-2021 | Sanna, C.; Marengo, A.; Acquadro, S.; Caredda, A.; Lai, R.; Corona, A.; Tramontano, E.; Rubiolo, P.; Esposito, F. | PLANTS | - |
Integration of SARS-CoV-2 RNA in infected human cells by retrotransposons: an unlikely hypothesis and old viral relationships | 1-gen-2021 | Grandi, N.; Tramontano, E.; Berkhout, B. | RETROVIROLOGY | - |
Zika virus NS2A inhibits interferon signaling by degradation of STAT1 and STAT2 | 1-gen-2021 | Fanunza, Elisa; Carletti, Fabrizio; Quartu, Marina; Grandi, Nicole; Ermellino, Laura; Milia, Jessica; Corona, Angela; Capobianchi, Maria Rosaria; Ippolito, Giuseppe; Tramontano, Enzo | VIRULENCE | - |
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function | 1-gen-2021 | Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Inhibitors of Ebolavirus targeting innate immune evasion | 1-gen-2021 | Paulis, A. L.; Corona, A.; Tramontano, E. | ANNUAL REPORTS IN MEDICINAL CHEMISTRY | - |
Early Diffusion of SARS-CoV-2 Infection in the Inner Area of the Italian Sardinia Island | 1-gen-2021 | Piras, Giovanna; Grandi, Nicole; Monne, Maria; Asproni, Rosanna; Fancello, Tatiana; Fiamma, Maura; Mameli, Giuseppe; Casu, Gavino; lo Maglio, Iana; Palmas, Angelo D.; Tramontano, Enzo | FRONTIERS IN MICROBIOLOGY | - |
Natural and Nature-Derived Products Targeting Human Coronaviruses | 1-gen-2021 | Vougogiannopoulou, Konstantina; Corona, Angela; Tramontano, Enzo; Alexis, Michael N.; Skaltsounis, Alexios-Leandros | MOLECULES | - |
Garcinol from Garcinia indica inhibits HIV-1 reverse transcriptase-associated ribonuclease H | 1-gen-2021 | Corona, Angela; Seibt, Sebastian; Schaller, David; Schobert, Rainer; Volkamer, Andrea; Biersack, Bernhard; Tramontano, Enzo | ARCHIV DER PHARMAZIE | - |
INMI1 Zika Virus NS4B Antagonizes the Interferon Signaling by Suppressing STAT1 Phosphorylation | 1-gen-2021 | Fanunza, Elisa; Grandi, Nicole; Quartu, Marina; Carletti, Fabrizio; Ermellino, Laura; Milia, Jessica; Corona, Angela; Rosaria Capobianchi, Maria; Ippolito, Giuseppe; Tramontano, Enzo | VIRUSES | - |
Diagnosi in vitro della Sclerosi Multipla | 1-gen-2020 | Grandi, Nicole; Pisano, MARIA PAOLA; Tramontano, Enzo | - | - |
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture | 1-gen-2020 | Pala, Nicolino; Esposito, Francesca; Tramontano, Enzo; Kumar Singh, Pankaj; Sanna, Vanna; Carcelli, Mauro; Haigh, Lisa D.; Satta, Sandro; Mario Sechi, And | ACS MEDICINAL CHEMISTRY LETTERS | - |
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity | 1-gen-2020 | Desantis, Jenny; Massari, Serena; Corona, Angela; Astolfi, Andrea; Sabatini, Stefano; Manfroni, Giuseppe; Palazzotti, Deborah; Cecchetti, Violetta; Pannecouque, Christophe; Tramontano, Enzo; Tabarrini, Oriana | MOLECULES | - |
Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition | 1-gen-2020 | Hayek, S.; Pietrancosta, N.; Hovhannisyan, A. A.; Alves de Sousa, R.; Bekaddour, N.; Ermellino, L.; Tramontano, E.; Arnould, S.; Sardet, C.; Dairou, J.; Diaz, O.; Lotteau, V.; Nisole, S.; Melikyan, G.; Herbeuval, J. -P.; Vidalain, P. -O. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitors | 1-gen-2020 | Esposito, Francesca; Sechi, Mario; Pala, Nicolino; Sanna, Adele; Koneru, Pratibha Chowdary; Kvaratskhelia, Mamuka; Naesens, Lieve; Corona, Angela; Grandi, Nicole; di Santo, Roberto; D'Amore, Vincenzo Maria; Di Leva, Francesco Saverio; Novellino, Ettore; Cosconati, Sandro; Tramontano, Enzo | ANTIVIRAL RESEARCH | - |
Peptides Mimicking the β7/β8 loop of HIV-1 Reverse Transcriptase p51 as “Hotspot-Targeted” Dimerization Inhibitors | 1-gen-2020 | Sánchez-Murcia, Pedro A.; de Castro, Sonia; García-Aparicio, Carlos; Jimenez, M. Angeles; Corona, Angela; Tramontano, Enzo; Sluis-Cremer, Nicolas; Menendez Arias, Luis; Velazquez, Sonsoles; Gago, Federico; Camarasa, María-José | ACS MEDICINAL CHEMISTRY LETTERS | - |
2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication | 1-gen-2020 | Corona, Angela; Onnis, Valentina; Del Vecchio, Claudia; Esposito, Francesca; Cheng, Yung-Chi; Tramontano, Enzo | MOLECULES | - |
Quercetin blocks Ebola Virus infection by counteracting the VP24 Interferon inhibitory function | 1-gen-2020 | Fanunza, Elisa; Iampietro, Mathieu; Distinto, Simona; Corona, Angela; Quartu, Marina; Maccioni, Elias; Horvat, Branka; Tramontano, Enzo | ANTIMICROBIAL AGENTS AND CHEMOTHERAPY | - |
A human MMTV-like betaretrovirus linked to breast cancer has been present in humans at least since the Copper Age | 1-gen-2020 | Lessi, F.; Grandi, N.; Mazzanti, C. M.; Civita, P.; Scatena, C.; Aretini, P.; Bandiera, P.; Fornaciari, A.; Giuffra, V.; Fornaciari, G.; Naccarato, A. G.; Tramontano, E.; Bevilacqua, G. | AGING | - |
Targeting HIV-1 RNase H: N'-(2-Hydroxy-benzylidene)-3,4,5-Trihydroxybenzoylhydrazone as Selective Inhibitor Active against NNRTIs-Resistant Variants | 1-gen-2020 | Corona, Angela; Ballana, Ester; Distinto, Simona; Rogolino, Dominga; Del Vecchio, Claudia; Carcelli, Mauro; Badia, Roger; Riveira-Muñoz, Eva; Esposito, Francesca; Parolin, Cristina; Esté, José A; Grandi, Nicole; Tramontano, Enzo | VIRUSES | - |
Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase | 1-gen-2020 | Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Di Maro, Salvatore; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Valenti, Piera; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto | ACS MEDICINAL CHEMISTRY LETTERS | - |
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