FLORIS, COSTANTINO
FLORIS, COSTANTINO
DIPARTIMENTO DI SCIENZE CHIMICHE E GEOLOGICHE
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function
2021-01-01 Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation
2020-01-01 Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F.
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators
2019-01-01 Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACCHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase
2017-01-01 Sonar, VIJAY PRAKASH; Corona, Angela; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Fois, Benedetta; Floris, Costantino; Malpure, Nilesh V.; Alcaro, Stefano; Tramontano, Enzo; Cottiglia, Filippo
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders
2017-01-01 Fois, Benedetta; Bianco, Giulia; Sonar, Vijay P.; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Melis, Claudia; Marras, Luisa; Pompei, Raffaello; Floris, Costantino; Caboni, Pierluigi; Cottiglia, Filippo
Binding of bis-(2-ethylhexyl) phthalate at the surface of hydrozincite nanocrystals: An example of organic molecules absorption onto nanocrystalline minerals
2015-01-01 Sanna, Roberta; Medas, Daniela; Podda, Francesca; Meneghini, C.; Casu, Mariano; Lattanzi, Pierfranco; Scorciapino, MARIANO ANDREA; Floris, Costantino; Cannas, Carla; DE GIUDICI, GIOVANNI BATTISTA
Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies
2015-01-01 Ruiu, S; Anzani, N; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Alcaro, S; Maccioni, Elias; Distinto, Simona; Cottiglia, Filippo
Investigation of the hydrozincite structure by infrared and solid-state NMR spectroscopy
2013-01-01 Sanna, Roberta; DE GIUDICI, GIOVANNI BATTISTA; Scorciapino, MARIANO ANDREA; Floris, Costantino; Casu, Mariano
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors
2013-01-01 Ruiu, S; Anzani, Nicola; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S; Cottiglia, Filippo
N-alkylamides from Otanthus maritimus: structure elucidation, binding affinity for cannabinoid receptors and computational study
2013-01-01 Anzani, N.; Ruiu, S.; Orrù, A.; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S.; Cottiglia, Filippo
Cytotoxic phloroglucinols from the leaves of Myrtus communis
2012-01-01 Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina
Mild Synthetic Approach to Novel Indole-1-Carbinols and Preliminary Evaluation of Their Cytotoxicity in Hepatocarcinoma Cells
2012-01-01 Zedda, G; Simbula, G; Begala, M; Pibiri, M; Floris, C; Casu, M; Casu, L; Tocco, G
Bioguided-isolation of cytotoxic phloroglucinols from the leaves of myrtus communis l.
2011-01-01 Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, P; Aicha, O; Sanna, Giuseppina
Metronidazole prodrugs: Synthesis, physicochemical properties, stability, and ex vivo release studies
2011-01-01 Mura, C; Valenti, Donatella; Floris, Costantino; Sanna, Roberta; DE LUCA, MARIA ANTONIETTA; Fadda, ANNA MARIA; Loy, G.
A chromone from Seseli praecox (Apiaceae)
2010-01-01 Leonti, Marco; Casu, Laura; SOLINAS M., N; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Gertsch, J; Saba, A. R.
A pterocarpan from the seeds of Bituminaria morisiana
2010-01-01 Leonti, Marco; Casu, Laura; Gertsch, J; Bonsignore, L; Floris, Costantino; Casu, Mariano; Cottiglia, Filippo
Benzophenones from the roots of the Popoluca Amerindian medicinal plant Securidaca diversifolia (L.) S.F. Blake
2010-01-01 Casu, Laura; Solinas, Mn; Saba, Ar; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Laconi, S; Pompei, Raffaello; Leonti, Marco
Falcarinol is a covalent cannabinoid CB1 receptor antagonist and induces pro-allergic effects in skin
2010-01-01 Leonti, Marco; Casu, Laura; Raduner, S; Cottiglia, Filippo; Floris, Costantino; ALTMANN K., H; Gertsch, J.
NOVEL 1-[1-(1H-INDOL-3-YL)ALKYL]-1H-INDOLES AND INDOLE-1-CARBINOLS: SYNTHESIS AND EVALUATION OF CYTOTOXICITY IN HEPATOCARCINOMA CELLS.
2010-01-01 Tocco, Graziella; Zedda, G; Simbula, Gabriella; Pibiri, G; Casu, Mariano; Floris, Costantino; Podda, G; Begala, Michela
Easy access to trans-2,3-disubstituted cyclobutanones, 2,4,5-trisubstituted 3,6-dihydro-2H-pyrans and cis-substituted phenylcyclopropylsulfones by using the highly versatile 1-phenylsulfenyl- or 1-phenylsulfonyl-cyclopropylketones
2009-01-01 Alberti, G; Bernard, ANGELA MARIA; Floris, Costantino; Floris, C; Frongia, Angelo; Piras, Pp; Secci, Francesco; Spiga, M.
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function | 1-gen-2021 | Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation | 1-gen-2020 | Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators | 1-gen-2019 | Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACCHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe | JOURNAL OF NATURAL PRODUCTS | - |
| Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2017 | Sonar, VIJAY PRAKASH; Corona, Angela; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Fois, Benedetta; Floris, Costantino; Malpure, Nilesh V.; Alcaro, Stefano; Tramontano, Enzo; Cottiglia, Filippo | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders | 1-gen-2017 | Fois, Benedetta; Bianco, Giulia; Sonar, Vijay P.; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Melis, Claudia; Marras, Luisa; Pompei, Raffaello; Floris, Costantino; Caboni, Pierluigi; Cottiglia, Filippo | JOURNAL OF NATURAL PRODUCTS | - |
| Binding of bis-(2-ethylhexyl) phthalate at the surface of hydrozincite nanocrystals: An example of organic molecules absorption onto nanocrystalline minerals | 1-gen-2015 | Sanna, Roberta; Medas, Daniela; Podda, Francesca; Meneghini, C.; Casu, Mariano; Lattanzi, Pierfranco; Scorciapino, MARIANO ANDREA; Floris, Costantino; Cannas, Carla; DE GIUDICI, GIOVANNI BATTISTA | JOURNAL OF COLLOID AND INTERFACE SCIENCE | - |
| Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies | 1-gen-2015 | Ruiu, S; Anzani, N; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Alcaro, S; Maccioni, Elias; Distinto, Simona; Cottiglia, Filippo | JOURNAL OF NATURAL PRODUCTS | - |
| Investigation of the hydrozincite structure by infrared and solid-state NMR spectroscopy | 1-gen-2013 | Sanna, Roberta; DE GIUDICI, GIOVANNI BATTISTA; Scorciapino, MARIANO ANDREA; Floris, Costantino; Casu, Mariano | AMERICAN MINERALOGIST | - |
| N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors | 1-gen-2013 | Ruiu, S; Anzani, Nicola; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S; Cottiglia, Filippo | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| N-alkylamides from Otanthus maritimus: structure elucidation, binding affinity for cannabinoid receptors and computational study | 1-gen-2013 | Anzani, N.; Ruiu, S.; Orrù, A.; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S.; Cottiglia, Filippo | - | - |
| Cytotoxic phloroglucinols from the leaves of Myrtus communis | 1-gen-2012 | Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina | JOURNAL OF NATURAL PRODUCTS | - |
| Mild Synthetic Approach to Novel Indole-1-Carbinols and Preliminary Evaluation of Their Cytotoxicity in Hepatocarcinoma Cells | 1-gen-2012 | Zedda, G; Simbula, G; Begala, M; Pibiri, M; Floris, C; Casu, M; Casu, L; Tocco, G | ARCHIV DER PHARMAZIE | - |
| Bioguided-isolation of cytotoxic phloroglucinols from the leaves of myrtus communis l. | 1-gen-2011 | Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, P; Aicha, O; Sanna, Giuseppina | - | - |
| Metronidazole prodrugs: Synthesis, physicochemical properties, stability, and ex vivo release studies | 1-gen-2011 | Mura, C; Valenti, Donatella; Floris, Costantino; Sanna, Roberta; DE LUCA, MARIA ANTONIETTA; Fadda, ANNA MARIA; Loy, G. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| A chromone from Seseli praecox (Apiaceae) | 1-gen-2010 | Leonti, Marco; Casu, Laura; SOLINAS M., N; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Gertsch, J; Saba, A. R. | NATURAL PRODUCT COMMUNICATIONS | - |
| A pterocarpan from the seeds of Bituminaria morisiana | 1-gen-2010 | Leonti, Marco; Casu, Laura; Gertsch, J; Bonsignore, L; Floris, Costantino; Casu, Mariano; Cottiglia, Filippo | NATURAL MEDICINES | - |
| Benzophenones from the roots of the Popoluca Amerindian medicinal plant Securidaca diversifolia (L.) S.F. Blake | 1-gen-2010 | Casu, Laura; Solinas, Mn; Saba, Ar; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Laconi, S; Pompei, Raffaello; Leonti, Marco | PHYTOCHEMISTRY LETTERS | - |
| Falcarinol is a covalent cannabinoid CB1 receptor antagonist and induces pro-allergic effects in skin | 1-gen-2010 | Leonti, Marco; Casu, Laura; Raduner, S; Cottiglia, Filippo; Floris, Costantino; ALTMANN K., H; Gertsch, J. | BIOCHEMICAL PHARMACOLOGY | - |
| NOVEL 1-[1-(1H-INDOL-3-YL)ALKYL]-1H-INDOLES AND INDOLE-1-CARBINOLS: SYNTHESIS AND EVALUATION OF CYTOTOXICITY IN HEPATOCARCINOMA CELLS. | 1-gen-2010 | Tocco, Graziella; Zedda, G; Simbula, Gabriella; Pibiri, G; Casu, Mariano; Floris, Costantino; Podda, G; Begala, Michela | - | - |
| Easy access to trans-2,3-disubstituted cyclobutanones, 2,4,5-trisubstituted 3,6-dihydro-2H-pyrans and cis-substituted phenylcyclopropylsulfones by using the highly versatile 1-phenylsulfenyl- or 1-phenylsulfonyl-cyclopropylketones | 1-gen-2009 | Alberti, G; Bernard, ANGELA MARIA; Floris, Costantino; Floris, C; Frongia, Angelo; Piras, Pp; Secci, Francesco; Spiga, M. | ORGANIC & BIOMOLECULAR CHEMISTRY | - |