Asymmetric Total Synthesis of (−)‐Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding
2025-01-01 Maiocchi, Alice; Shevelev, Maxim; Boiarska, Zlata; Estévez‐gallego, Juan; Bonato, Francesca; Orlando, Paolo; Chinosi, Alessandra; Marcone, Emanuele; Citarella, Andrea; Horvath, Dragos; Steinmetz, Michel O.; Prota, Andrea E.; Varnek, Alexandre; Fasano, Valerio; Passarella, Daniele
Hydrogels for the Delivery of Plant-Derived (Poly)Phenols
2020-01-01 Micale, Nicola; Citarella, Andrea; Molonia, Maria Sofia; Speciale, Antonio; Cimino, Francesco; Saija, Antonella; Cristani, Mariateresa
Sustainable Synthesis of 1,2,3‐Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry
2025-01-01 Citarella, Andrea; Fiori, Alessandro; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio
A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene
2024-01-01 Citarella, Andrea; Cavinato, Miriam; Amenta, Arianna; Nardini, Marco; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio
Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol
2021-01-01 Micale, N.; Molonia, M. S.; Citarella, A.; Cimino, F.; Saija, A.; Cristani, M.; Speciale, A.
Nirmatrelvir: from discovery to modern and alternative synthetic approaches
2024-01-01 Galli, Michela; Migliano, Francesco; Fasano, Valerio; Silvani, Alessandra; Passarella, Daniele; Citarella, Andrea
Selective noncovalent proteasome inhibiting activity of trifluoromethyl-containing gem-quaternary aziridines
2023-01-01 Ielo, L.; Patamia, V.; Citarella, A.; Schirmeister, T.; Stagno, C.; Rescifina, A.; Micale, N.; Pace, V.
Syntheses, reactivity, and biological applications of coumarins
2024-01-01 Citarella, Andrea; Vittorio, Serena; Dank, Christian; Ielo, Laura
Cyrene: A Green Solvent for the Synthesis of Bioactive Molecules and Functional Biomaterials
2022-01-01 Citarella, Andrea; Amenta, Arianna; Passarella, Daniele; Micale, Nicola
Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines
2022-01-01 Ielo, Laura; Patamia, Vincenzo; Citarella, Andrea; Efferth, Thomas; Shahhamzehei, Nasim; Schirmeister, Tanja; Stagno, Claudio; Langer, Thierry; Rescifina, Antonio; Micale, Nicola; Pace, Vittorio
Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes
2024-01-01 Platella, Chiara; Citarella, Andrea; Manenti, Marco; Spinelli, Guglielmo; Gaglione, Rosa; Arciello, Angela; Riccardi, Claudia; Musumeci, Domenica; Montesarchio, Daniela; Giannini, Clelia; Silvani, Alessandra
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks
2025-01-01 Pedrini, Martina; Pozzi, Luca; Sacchi, Francesca; Citarella, Andrea; Fasano, Valerio; Seneci, Pierfausto; Pieraccini, Stefano; Ruberto, Lorenzo; Perez Peña, Helena; Garzino-Demo, Alfredo; Vitiello, Adriana; Sernicola, Leonardo; Borsetti, Alessandra; Calistri, Arianna; Parolin, Cristina; Passarella, Daniele
SARS-CoV-2 Mpro: A Potential Target for Peptidomimetics and Small-Molecule Inhibitors
2021-01-01 Citarella, Andrea; Scala, Angela; Piperno, Anna; Micale, Nicola
Revisiting the Reduction of Vinpocetine
2025-01-01 Borsoi, Simone; Pozzi, Luca; Fasano, Valerio; Citarella, Andrea; Macetti, Giovanni; Presti, Leonardo Lo; Paladino, Giuseppe; Ciriello, Umberto; Passarella, Daniele
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors
2023-01-01 Fassi, Enrico M. A.; Manenti, Marco; Citarella, Andrea; Dei Cas, Michele; Casati, Sara; Micale, Nicola; Schirmeister, Tanja; Roda, Gabriella; Silvani, Alessandra; Grazioso, Giovanni
Cannabizetol, a Novel Cannabinoid: Chemical Synthesis, Anti-inflammatory Activity and Extraction from Cannabis sativa L
2025-01-01 Pozzi, Luca; Gotti, Andrea; Fumagalli, Marco; Citarella, Andrea; Fasano, Valerio; Paladino, Giuseppe; Ciriello, Umberto; Princiotto, Salvatore; Annunziata, Francesca; Martinelli, Giulia; Sangiovanni, Enrico; Pinto, Andrea; Dell’Agli, Mario; Passarella, Daniele
Chemoselective Homologation-Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes
2020-01-01 Miele, Margherita; Citarella, Andrea; Langer, Thierry; Urban, Ernst; Zehl, Martin; Holzer, Wolfgang; Ielo, Laura; Pace, Vittorio
Peptidyl Fluoromethyl Ketones and Their Applications in Medicinal Chemistry
2020-01-01 Citarella, A.; Micale, N.
Anomalous Magnetism in 3d-4f Double Perovskite Oxide Nd2FeCrO6 with Kramer’s Ion Nd3+
2025-01-01 Kumar, Saurav; Majumder, Shantanu; Congiu, Francesco; Muscas, Giuseppe; Luetkens, H.; Kaushik, S. D.; Pandey, Shishir K.; Lee, Stephen L.; Deshpande, Uday; Sarkar, Tapati; Ray, Soumya Jyoti
PCSK9 Inhibitor Inclisiran Attenuates Cardiotoxicity Induced by Sequential Anthracycline and Trastuzumab Exposure via NLRP3 and MyD88 Pathway Inhibition
2025-01-01 Quagliariello, Vincenzo; Berretta, Massimiliano; Bisceglia, Irma; Iovine, Martina; Barbato, Matteo; Arianna, Raffaele; Canale, Maria Laura; Paccone, Andrea; Inno, Alessandro; Scherillo, Marino; Oliva, Stefano; Cadeddu Dessalvi, Christian; Mauriello, Alfredo; Maurea, Carlo; Fonderico, Celeste; Maratea, Anna Chiara; Gabrielli, Domenico; Maurea, Nicola
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Asymmetric Total Synthesis of (−)‐Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding | 1-gen-2025 | Maiocchi, Alice; Shevelev, Maxim; Boiarska, Zlata; Estévez‐gallego, Juan; Bonato, Francesca; Orlando, Paolo; Chinosi, Alessandra; Marcone, Emanuele; Citarella, Andrea; Horvath, Dragos; Steinmetz, Michel O.; Prota, Andrea E.; Varnek, Alexandre; Fasano, Valerio; Passarella, Daniele | CHEMISTRY-A EUROPEAN JOURNAL | - |
| Hydrogels for the Delivery of Plant-Derived (Poly)Phenols | 1-gen-2020 | Micale, Nicola; Citarella, Andrea; Molonia, Maria Sofia; Speciale, Antonio; Cimino, Francesco; Saija, Antonella; Cristani, Mariateresa | MOLECULES | - |
| Sustainable Synthesis of 1,2,3‐Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry | 1-gen-2025 | Citarella, Andrea; Fiori, Alessandro; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio | CHEMSUSCHEM | - |
| A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene | 1-gen-2024 | Citarella, Andrea; Cavinato, Miriam; Amenta, Arianna; Nardini, Marco; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio | EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | - |
| Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol | 1-gen-2021 | Micale, N.; Molonia, M. S.; Citarella, A.; Cimino, F.; Saija, A.; Cristani, M.; Speciale, A. | MOLECULES | - |
| Nirmatrelvir: from discovery to modern and alternative synthetic approaches | 1-gen-2024 | Galli, Michela; Migliano, Francesco; Fasano, Valerio; Silvani, Alessandra; Passarella, Daniele; Citarella, Andrea | PROCESSES | - |
| Selective noncovalent proteasome inhibiting activity of trifluoromethyl-containing gem-quaternary aziridines | 1-gen-2023 | Ielo, L.; Patamia, V.; Citarella, A.; Schirmeister, T.; Stagno, C.; Rescifina, A.; Micale, N.; Pace, V. | ARCHIV DER PHARMAZIE | - |
| Syntheses, reactivity, and biological applications of coumarins | 1-gen-2024 | Citarella, Andrea; Vittorio, Serena; Dank, Christian; Ielo, Laura | FRONTIERS IN CHEMISTRY | - |
| Cyrene: A Green Solvent for the Synthesis of Bioactive Molecules and Functional Biomaterials | 1-gen-2022 | Citarella, Andrea; Amenta, Arianna; Passarella, Daniele; Micale, Nicola | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
| Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines | 1-gen-2022 | Ielo, Laura; Patamia, Vincenzo; Citarella, Andrea; Efferth, Thomas; Shahhamzehei, Nasim; Schirmeister, Tanja; Stagno, Claudio; Langer, Thierry; Rescifina, Antonio; Micale, Nicola; Pace, Vittorio | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
| Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes | 1-gen-2024 | Platella, Chiara; Citarella, Andrea; Manenti, Marco; Spinelli, Guglielmo; Gaglione, Rosa; Arciello, Angela; Riccardi, Claudia; Musumeci, Domenica; Montesarchio, Daniela; Giannini, Clelia; Silvani, Alessandra | JOURNAL OF MOLECULAR STRUCTURE | - |
| Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks | 1-gen-2025 | Pedrini, Martina; Pozzi, Luca; Sacchi, Francesca; Citarella, Andrea; Fasano, Valerio; Seneci, Pierfausto; Pieraccini, Stefano; Ruberto, Lorenzo; Perez Peña, Helena; Garzino-Demo, Alfredo; Vitiello, Adriana; Sernicola, Leonardo; Borsetti, Alessandra; Calistri, Arianna; Parolin, Cristina; Passarella, Daniele | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| SARS-CoV-2 Mpro: A Potential Target for Peptidomimetics and Small-Molecule Inhibitors | 1-gen-2021 | Citarella, Andrea; Scala, Angela; Piperno, Anna; Micale, Nicola | BIOMOLECULES | - |
| Revisiting the Reduction of Vinpocetine | 1-gen-2025 | Borsoi, Simone; Pozzi, Luca; Fasano, Valerio; Citarella, Andrea; Macetti, Giovanni; Presti, Leonardo Lo; Paladino, Giuseppe; Ciriello, Umberto; Passarella, Daniele | CHEMISTRYSELECT | - |
| Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors | 1-gen-2023 | Fassi, Enrico M. A.; Manenti, Marco; Citarella, Andrea; Dei Cas, Michele; Casati, Sara; Micale, Nicola; Schirmeister, Tanja; Roda, Gabriella; Silvani, Alessandra; Grazioso, Giovanni | MOLECULES | - |
| Cannabizetol, a Novel Cannabinoid: Chemical Synthesis, Anti-inflammatory Activity and Extraction from Cannabis sativa L | 1-gen-2025 | Pozzi, Luca; Gotti, Andrea; Fumagalli, Marco; Citarella, Andrea; Fasano, Valerio; Paladino, Giuseppe; Ciriello, Umberto; Princiotto, Salvatore; Annunziata, Francesca; Martinelli, Giulia; Sangiovanni, Enrico; Pinto, Andrea; Dell’Agli, Mario; Passarella, Daniele | JOURNAL OF NATURAL PRODUCTS | - |
| Chemoselective Homologation-Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes | 1-gen-2020 | Miele, Margherita; Citarella, Andrea; Langer, Thierry; Urban, Ernst; Zehl, Martin; Holzer, Wolfgang; Ielo, Laura; Pace, Vittorio | ORGANIC LETTERS | - |
| Peptidyl Fluoromethyl Ketones and Their Applications in Medicinal Chemistry | 1-gen-2020 | Citarella, A.; Micale, N. | MOLECULES | - |
| Anomalous Magnetism in 3d-4f Double Perovskite Oxide Nd2FeCrO6 with Kramer’s Ion Nd3+ | 1-gen-2025 | Kumar, Saurav; Majumder, Shantanu; Congiu, Francesco; Muscas, Giuseppe; Luetkens, H.; Kaushik, S. D.; Pandey, Shishir K.; Lee, Stephen L.; Deshpande, Uday; Sarkar, Tapati; Ray, Soumya Jyoti | PHYSICAL REVIEW. B | - |
| PCSK9 Inhibitor Inclisiran Attenuates Cardiotoxicity Induced by Sequential Anthracycline and Trastuzumab Exposure via NLRP3 and MyD88 Pathway Inhibition | 1-gen-2025 | Quagliariello, Vincenzo; Berretta, Massimiliano; Bisceglia, Irma; Iovine, Martina; Barbato, Matteo; Arianna, Raffaele; Canale, Maria Laura; Paccone, Andrea; Inno, Alessandro; Scherillo, Marino; Oliva, Stefano; Cadeddu Dessalvi, Christian; Mauriello, Alfredo; Maurea, Carlo; Fonderico, Celeste; Maratea, Anna Chiara; Gabrielli, Domenico; Maurea, Nicola | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
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