UNICA IRIS Institutional Research Information System

MELEDDU, RITA
 Distribuzione geografica
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Continente #
EU - Europa 171.613
NA - Nord America 3.972
AS - Asia 615
AF - Africa 10
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 2
Totale 176.216
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Nazione #
IT - Italia 170.435
US - Stati Uniti d'America 3.950
CN - Cina 450
UA - Ucraina 374
SE - Svezia 360
DE - Germania 183
FI - Finlandia 99
GB - Regno Unito 86
SG - Singapore 78
FR - Francia 26
VN - Vietnam 24
IN - India 19
CA - Canada 17
RU - Federazione Russa 14
HK - Hong Kong 13
PK - Pakistan 13
KR - Corea 9
BE - Belgio 8
CZ - Repubblica Ceca 8
PT - Portogallo 6
MX - Messico 5
ES - Italia 4
IR - Iran 4
ZA - Sudafrica 4
EU - Europa 3
TN - Tunisia 3
EG - Egitto 2
HU - Ungheria 2
ID - Indonesia 2
NL - Olanda 2
PL - Polonia 2
RO - Romania 2
A1 - Anonimo 1
BR - Brasile 1
CM - Camerun 1
CO - Colombia 1
IE - Irlanda 1
IM - Isola di Man 1
JP - Giappone 1
KW - Kuwait 1
LA - Repubblica Popolare Democratica del Laos 1
Totale 176.216
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Città #
Cagliari 168.345
Uta 1.811
Fairfield 463
Woodbridge 399
Chandler 348
Ashburn 265
Nyköping 261
Houston 245
Ann Arbor 238
Wilmington 224
Boardman 205
Seattle 204
Jacksonville 183
Cambridge 149
Dearborn 136
New York 95
Shanghai 87
Nanjing 75
Beijing 57
Boston 52
Helsinki 45
Redwood City 34
Singapore 31
San Diego 30
Shenyang 26
Dong Ket 24
Changsha 20
Los Angeles 19
Nanchang 19
Verona 17
Jiaxing 16
Sassari 16
Hebei 15
Milan 15
Guangzhou 14
Herndon 14
Mountain View 13
Zhengzhou 13
Hong Kong 12
Jinan 12
Gujranwala 11
Norwalk 11
Toronto 11
Kunming 10
London 9
Seoul 9
Tianjin 9
Auburn Hills 8
Brussels 8
Wuhan 8
Rome 7
Washington 7
Atlanta 6
Brno 6
Ningbo 6
Orange 6
Walnut 6
Zerfalìu 6
Falls Church 5
Hangzhou 5
Mumbai 5
Olbia 5
Paris 5
Redmond 5
Saint Petersburg 5
Bengaluru 4
Durban 4
Hefei 4
Indiana 4
Ottawa 4
Phoenix 4
Taizhou 4
Chicago 3
Munich 3
Pisa 3
Pune 3
Quartu Sant'Elena 3
Villanovafranca 3
Acton 2
Barcelona 2
Berlin 2
Borås 2
Chiswick 2
Dolianova 2
Frankfurt am Main 2
Hanover 2
Jakarta 2
Kilburn 2
La Jolla 2
Madrid 2
Mohegan Lake 2
Monserrato 2
Nanning 2
Nürnberg 2
Oristano 2
Porto 2
Püttlingen 2
Quartu Sant'elena 2
San Francisco 2
San Mateo 2
Totale 174.516
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Nome #
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 14.508
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida 4.871
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase 4.507
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders 4.506
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase 4.300
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors 4.255
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents 4.232
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6 4.163
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B 4.138
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase 4.010
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII 3.771
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold 3.629
A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition 3.610
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors 3.388
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators 3.367
Systemic lupus erythematosus occurring in a patient with Niemann-Pick type B disease. 3.353
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B 3.205
Design and synthesis of new isatin derivatives as HIV-1 reverse transcriptase associated ribonuclease H inhibitors 3.157
Molecular Aspects of the RT/drug Interactions. Perspective of Dual Inhibitors 3.156
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B 3.109
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation 3.109
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase 3.093
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms 3.038
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 RT. 2.886
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides 2.861
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids 2.831
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) enlighten the mechanism of action of a new Ribonuclease H/DNA polymerase RT dual inhibitor 2.779
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) shed light on the mechanism of action of a new Ribonuclease H/ DNA polymerase RT dual inhibitor 2.776
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Single Site Dual Inhibitors of HIV-1 RT 2.752
Mutagenic study on HIV-1 reverse transcriptase to explore the mechanism of action of HIV-1 reverse transcriptase dual inhibitors 2.614
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function 2.483
Synthesis and biological activity evaluation of new dual-inhibitors of both associated functions of HIV-1 RT 2.481
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases 2.392
Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase 2.312
New promising scaffolds for the inhibition of monoamine oxidase B 2.163
Exploring new scaffolds for the inibition of the Ribonuclease H function of RT HIV-1 2.129
Design and synthesis of new Isatin derivatives as HIV-1 Reverse Transcriptase associated Ribonuclease H inhibitors twenty-fourth 2.028
Isatin derivatives as new scaffolds for HIV-1 reverse transcriptase associated RNase H and RDDP dual inhibitors 1.992
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis 1.968
Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors 1.952
2-Acylhydrazino-5-arylpyrrole derivatives: Synthesis and antifungal activity evaluation 1.878
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis and microbiological evaluation 1.834
Design, synthesis and biological activity evaluation of new HIV-1 reverse transcriptase dual inhibitors 1.828
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones 1.800
Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach 1.760
1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings 1.715
Identification of new scaffolds for the inhibition of HIV-1 Reverse Transcriptase associated Ribonuclease H function by means of shape based similarity screening 1.687
SITE DIRECT MUTAGENESIS AND KINETIC STUDIES TO EXPLORE THE MECHANISM OF ACTION OF ISATIN DERIVATIVES AS HIV-1 REVERSE TRANSCRIPTASE DUAL INHIBITORS 1.634
Exploring new scaffolds for the inhibition of the Ribonuclease H function of RT HIV-1 1.593
SYNTHESIS, MOLECULAR MODELLING, INHIBITORY ACTIVITY, AND SELECTIVITY TOWARDS MONOAMINE OXIDASE OF NEW HETEROCYCLIC SCAFFOLDS 1.564
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII 1.522
Semicarbazide-sensitive amine oxidase/vascular adhesion protein-1: a patent survey 1.516
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis 1.485
Synthesis and biological evaluation of new dual inhibitors of HIV-1 associated functions 1.478
Novel N-aryl- and N-heteryl-phenazine-1-carboxamides as potential agents for the treatment of infections sustained by drug-resistant and MDR Mycobacterium tuberculosis 1.452
From classic to innovative approaches in HIV-1 infection treatment 1.426
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function 1.426
Novel N-aryl- and N-heteryl phenazine-1-carboxamides as potential agents for the treatment of infections sustained by drug-resistant and multidrug-resistant Mycobacterium tuberculosis 1.385
2-methoxynaphthalen thiazole derivate : a new HIV-1 RT Ribonuclease H/DNA polymerase dual inhibitor active on viral replication 1.380
Synthesis, molecular modelling, inhibitory acivity, and selectivity towards monoamine oxidase of new heterocyclic scaffold 1.004
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents 986
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions 943
L’OLIO ESSENZIALE DI ARTEMISIA ARBORESCENS INATTIVA HSV1 E HSV2 E INIBISCE LA DIFFUSIONE LATERALE DI CELLULE VERO 916
Synthesis of different series of small molecules targeting HIV-1 RT, Candida albicans, MAO and G-Quadruplex 867
Tri-substituted thiazolines as promising scaffolds for the design of efficient COX inhibitors 821
L’olio essenziale di Artemisia arborescens inattiva HSV-1 e HSV-2 e inibisce la diffusione laterale in cellule Vero 698
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action 648
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives 564
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPβ phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea 432
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms 204
Privileged Scaffold Hybridization in the Design of Carbonic Anhydrase Inhibitors 68
New Structural Features of Isatin Dihydrothiazole Hybrids for Selective Carbonic Anhydrase Inhibitors 62
Totale 176.450
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Categoria #
all - tutte 194.620
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 194.620
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/202024.830 0 0 0 597 8.832 7.053 3.700 792 648 945 801 1.462
2020/202139.479 1.369 1.508 2.136 10.305 7.169 4.124 3.003 2.371 1.146 2.434 2.581 1.333
2021/20228.064 1.004 734 401 542 710 557 445 382 689 764 894 942
2022/202312.945 1.117 1.853 1.685 1.379 868 1.346 675 1.036 762 691 1.076 457
2023/202411.424 523 367 816 816 1.081 2.108 1.464 934 723 706 858 1.028
2024/202530.395 13.803 11.583 4.410 599 0 0 0 0 0 0 0 0
Totale 176.450