UNICA IRIS Institutional Research Information System

MELEDDU, RITA
 Distribuzione geografica
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Continente #
EU - Europa 139.730
NA - Nord America 3.810
AS - Asia 475
AF - Africa 10
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 2
Totale 144.031
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Nazione #
IT - Italia 138.566
US - Stati Uniti d'America 3.788
CN - Cina 385
UA - Ucraina 374
SE - Svezia 360
DE - Germania 179
FI - Finlandia 97
GB - Regno Unito 86
FR - Francia 26
VN - Vietnam 24
CA - Canada 17
SG - Singapore 16
IN - India 15
HK - Hong Kong 13
PK - Pakistan 13
RU - Federazione Russa 12
BE - Belgio 8
PT - Portogallo 6
MX - Messico 5
ES - Italia 4
IR - Iran 4
ZA - Sudafrica 4
EU - Europa 3
TN - Tunisia 3
CZ - Repubblica Ceca 2
EG - Egitto 2
HU - Ungheria 2
ID - Indonesia 2
NL - Olanda 2
PL - Polonia 2
RO - Romania 2
A1 - Anonimo 1
BR - Brasile 1
CM - Camerun 1
CO - Colombia 1
IE - Irlanda 1
IM - Isola di Man 1
JP - Giappone 1
KW - Kuwait 1
LA - Repubblica Popolare Democratica del Laos 1
Totale 144.031
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Città #
Cagliari 138.305
Fairfield 463
Woodbridge 399
Chandler 348
Nyköping 261
Ashburn 258
Houston 245
Ann Arbor 238
Wilmington 224
Seattle 204
Jacksonville 183
Cambridge 149
Dearborn 136
New York 95
Nanjing 74
Boardman 61
Shanghai 59
Beijing 55
Boston 52
Helsinki 43
Redwood City 34
San Diego 30
Shenyang 26
Dong Ket 24
Changsha 20
Nanchang 19
Verona 17
Hebei 15
Herndon 14
Jiaxing 14
Guangzhou 13
Mountain View 13
Zhengzhou 13
Hong Kong 12
Jinan 12
Milan 12
Gujranwala 11
Norwalk 11
Toronto 11
Kunming 10
Los Angeles 10
Sassari 10
London 9
Tianjin 9
Auburn Hills 8
Brussels 8
Washington 7
Atlanta 6
Ningbo 6
Orange 6
Walnut 6
Zerfalìu 6
Falls Church 5
Hangzhou 5
Mumbai 5
Olbia 5
Paris 5
Redmond 5
Saint Petersburg 5
Durban 4
Hefei 4
Indiana 4
Ottawa 4
Phoenix 4
Rome 4
Taizhou 4
Chicago 3
Pune 3
Quartu Sant'Elena 3
Villanovafranca 3
Wuhan 3
Acton 2
Barcelona 2
Berlin 2
Borås 2
Chiswick 2
Dolianova 2
Hanover 2
Jakarta 2
Kilburn 2
La Jolla 2
Madrid 2
Mohegan Lake 2
Monserrato 2
Nanning 2
Nürnberg 2
Oristano 2
Porto 2
Püttlingen 2
Quartu Sant'elena 2
San Francisco 2
San Mateo 2
Sovicille 2
Vila Nova de Gaia 2
Warsaw 2
Xian 2
Yellow Springs 2
Alghero 1
Ardabil 1
Arlington 1
Totale 142.407
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Nome #
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida 4.414
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase 4.129
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase 4.079
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6 3.964
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase 3.838
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase 3.785
3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B 3.700
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII 3.603
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders 3.546
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors 3.546
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold 3.497
A novel series of 3,4-disubstituted dihydropyrazoles: Synthesis and evaluation for MAO enzyme inhibition 3.352
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents 3.164
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators 3.136
Systemic lupus erythematosus occurring in a patient with Niemann-Pick type B disease. 3.075
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B 3.059
Design and synthesis of new isatin derivatives as HIV-1 reverse transcriptase associated ribonuclease H inhibitors 2.952
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms 2.912
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B 2.909
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase 2.822
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors 2.662
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) shed light on the mechanism of action of a new Ribonuclease H/ DNA polymerase RT dual inhibitor 2.659
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids 2.646
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Single Site Dual Inhibitors of HIV-1 RT 2.618
Site directed mutagenesis studies on HIV-1 reverse transcriptase (RT) enlighten the mechanism of action of a new Ribonuclease H/DNA polymerase RT dual inhibitor 2.618
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation 2.581
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides 2.490
Design, Synthesis and Biological Evaluation of New 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 RT. 2.329
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases 2.268
Molecular Aspects of the RT/drug Interactions. Perspective of Dual Inhibitors 2.244
Chalcones as novel dual inhibitors of HIV-1 reverse transcriptase 2.205
Synthesis and biological activity evaluation of new dual-inhibitors of both associated functions of HIV-1 RT 2.189
3-[2-(4-aryl-1,3-thiazol-2-yl)hydrazin-1-ylidene]-1H-indol-2-ones as new potential dual inhibitors of polimerase and ribonuclease HIV-1 RT associated function 2.104
Exploring new scaffolds for the inibition of the Ribonuclease H function of RT HIV-1 2.023
New promising scaffolds for the inhibition of monoamine oxidase B 2.008
Design and synthesis of new Isatin derivatives as HIV-1 Reverse Transcriptase associated Ribonuclease H inhibitors twenty-fourth 1.924
Mutagenic study on HIV-1 reverse transcriptase to explore the mechanism of action of HIV-1 reverse transcriptase dual inhibitors 1.778
Isatin derivatives as new scaffolds for HIV-1 reverse transcriptase associated RNase H and RDDP dual inhibitors 1.715
Design of new inhibitors of the HIV-1 Reverse Transcriptase associated Ribonuclease H function: a synthetic approach 1.694
Design, synthesis and biolgical activity evaluation of new HIV-1 reverse transcriptase dual inhibitors 1.629
2-Acylhydrazino-5-arylpyrrole derivatives: Synthesis and antifungal activity evaluation 1.522
Identification of new scaffolds for the inhibition of HIV-1 Reverse Transcriptase associated Ribonuclease H function by means of shape based similarity screening 1.515
SITE DIRECT MUTAGENESIS AND KINETIC STUDIES TO EXPLORE THE MECHANISM OF ACTION OF ISATIN DERIVATIVES AS HIV-1 REVERSE TRANSCRIPTASE DUAL INHIBITORS 1.465
Exploring new scaffolds for the inhibition of the Ribonuclease H function of RT HIV-1 1.418
SYNTHESIS, MOLECULAR MODELLING, INHIBITORY ACTIVITY, AND SELECTIVITY TOWARDS MONOAMINE OXIDASE OF NEW HETEROCYCLIC SCAFFOLDS 1.406
Design, synthesis and biological activity evaluation of new HIV-1 reverse transcriptase dual inhibitors 1.391
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis 1.334
From classic to innovative approaches in HIV-1 infection treatment 1.304
Synthesis and biological evaluation of new dual inhibitors of HIV-1 associated functions 1.297
2-methoxynaphthalen thiazole derivate : a new HIV-1 RT Ribonuclease H/DNA polymerase dual inhibitor active on viral replication 1.293
Semicarbazide-sensitive amine oxidase/vascular adhesion protein-1: a patent survey 1.276
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function 1.273
Novel N-aryl- and N-heteryl phenazine-1-carboxamides as potential agents for the treatment of infections sustained by drug-resistant and multidrug-resistant Mycobacterium tuberculosis 1.253
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis and microbiological evaluation 1.216
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones 1.192
Novel N-aryl- and N-heteryl-phenazine-1-carboxamides as potential agents for the treatment of infections sustained by drug-resistant and MDR Mycobacterium tuberculosis 1.130
1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings 1.076
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis 1.059
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents 924
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII 904
Synthesis, molecular modelling, inhibitory acivity, and selectivity towards monoamine oxidase of new heterocyclic scaffold 885
L’OLIO ESSENZIALE DI ARTEMISIA ARBORESCENS INATTIVA HSV1 E HSV2 E INIBISCE LA DIFFUSIONE LATERALE DI CELLULE VERO 829
Tri-substituted thiazolines as promising scaffolds for the design of efficient COX inhibitors 750
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions 746
Synthesis of different series of small molecules targeting HIV-1 RT, Candida albicans, MAO and G-Quadruplex 641
L’olio essenziale di Artemisia arborescens inattiva HSV-1 e HSV-2 e inibisce la diffusione laterale in cellule Vero 616
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives 428
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action 162
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPβ phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea 63
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms 27
Totale 144.261
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Categoria #
all - tutte 159.670
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 159.670
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019952 0 0 0 0 0 0 0 0 0 0 549 403
2019/202027.474 1.286 1.127 231 597 8.832 7.053 3.700 792 648 945 801 1.462
2020/202139.479 1.369 1.508 2.136 10.305 7.169 4.124 3.003 2.371 1.146 2.434 2.581 1.333
2021/20228.064 1.004 734 401 542 710 557 445 382 689 764 894 942
2022/202312.945 1.117 1.853 1.685 1.379 868 1.346 675 1.036 762 691 1.076 457
2023/20249.630 523 367 816 816 1.081 2.108 1.464 934 723 706 92 0
Totale 144.261